Full Catalog
GPCRs
| Receptor Family | Receptor | Species | Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Adenosine | A1 | human | HEK293T | C1427B | DC1427B | MC1427B |
| Adenosine | A1 | human | CHO-K1 | C1427-1 | DC1427-1 | MC1427-1 |
| Adenosine | A1 | rat | HEK293T | Cr1427 | DCr1427 | MCr1427 |
| Adenosine | A2A | human | HEK293T | C1428 | DC1428 | MC1428 |
| Adenosine | A2A | human | CHO-K1 | C1428-1 | DC1428-1 | MC1428-1 |
| Adenosine | A2A | mouse | HEK293T | Cm1428A | DCm1428A | MCm1428A |
| Adenosine | A2A | mouse | HEK293T | Cm1428B | DCm1428B | MCm1428B |
| Adenosine | A2A | mouse | CHO-K1 | Cm1428-1 | DCm1428-1 | MCm1428-1 |
| Adenosine | A2A | rat | HEK293T | Cr1428 | DCr1428 | MCr1428 |
| Adenosine | A2B | human | HEK293T | C1429 | DC1429 | MC1429 |
| Adenosine | A2B | human | CHO-K1 | C1429-1 | DC1429-1 | MC1429-1 |
| Adenosine | A2B | human | HEK293T | C1429a | DC1429a | MC1429a |
| Adenosine | A2B | rat | HEK293T | Cr1429 | DCr1429 | MCr1429 |
| Adenosine | A3 | human | HEK293T | C1430 | DC1430 | MC1430 |
| Adenosine | A3 | human | CHO-K1 | C1430-1 | DC1430-1 | MC1430-1 |
| Adenosine | A3 | rat | HEK293T | Cr1430 | DCr1430 | MCr1430 |
| Adhesion Class GPCRs | GPR97 | human | HEK293T | C1396 | DC1396 | MC1396 |
| Adhesion Class GPCRs | GPR110 | human | HEK293T | C1378 | DC1378 | MC1378 |
| Adrenergic | alpha1A | human | CHO-K1 | C1431-1 | DC1431-1 | MC1431-1 |
| Adrenergic | alpha1B | human | CHO-K1 | C1432-1 | DC1432-1 | MC1432-1 |
| Adrenergic | alpha1D | human | CHO-K1 | C1433-1 | DC1433-1 | MC1433-1 |
| Adrenergic | alpha2A | human | CHO-K1 | C1434-1 | DC1434-1 | MC1434-1 |
| Adrenergic | alpha2A | human | CHO-K1 | C1434-1a | DC1434-1a | MC1434-1a |
| Adrenergic | alpha2A | human | CHO-K1 Gqi5 | CG1434-1 | DCG1434-1 | MCG1434-1 |
| Adrenergic | alpha2B | human | CHO-K1 | C1435-1 | DC1435-1 | MC1435-1 |
| Adrenergic | alpha2B | human | CHO-K1 Gqi5 | CG1435-1 | DCG1435-1 | MCG1435-1 |
| Adrenergic | alpha2C | human | CHO-K1 | C1436-1 | DC1436-1 | MC1436-1 |
| Adrenergic | alpha2C | human | CHO-K1 Gqi5 | CG1436-1 | DCG1436-1 | MCG1436-1 |
| Adrenergic | beta1 | human | HEK293T | H1437 | H1437 | H1437 |
| Adrenergic | beta1 | human | CHO-K1 | C1437-1 | DC1437-1 | MC1437-1 |
| Adrenergic | beta2 | human | CHO-K1 | C1438-1a | DC1438-1a | MC1438-1a |
| Adrenergic | beta2 | human | HEK293T β-Arrestin1 | CA1438BA1 | DCA1438BA1 | MCA1438BA1 |
| Adrenergic | beta2 | human | HEK293T β-Arrestin2 | CA1438BA2 | DCA1438BA2 | MCA1438BA2 |
| Adrenergic | beta3 | human | HEK293T | C1439a | DC1439a | MC1439a |
| Anaphylatoxin | C3AR1 | human | HEK293T | C1222 | DC1222 | MC1222 |
| Anaphylatoxin | C5R1 | human | HEK293T | C1221 | DC1221 | MC1221 |
| Angiotensin | AT1 | mouse | CHO-K1 | Cm1417-1 | DCm1417-1 | MCm1417-1 |
| Angiotensin | AT1 | mouse | CHO-K1 | Cm1417-1a | DCm1417-1a | MCm1417-1a |
| Angiotensin | AT1 | human | HEK293T | H1417 | DH1417 | MH1417 |
| Angiotensin | AT1 | human | HEK293T | HA1417- BA1 | DHA1417- BA1 | MHA1417- BA1 |
| Angiotensin | AT1 | human | HEK293T | HA1417-BA2 | DHA1417-BA2 | MHA1417-BA2 |
| Apelin | APJ | human | HEK293T | C1196a | DC1196a | MC1196a |
| Apelin | APJ | human | CHO-K1 | C1196-1 | DC1196-1 | MC1196-1 |
| Bile Acid | GPBA | human | CHO-K1 | C1361-1 | DC1361-1 | MC1361-1 |
| Bile Acid | GPBA | human | CHO-K1 | C1361-1a | DC1361-1a | MC1361-1a |
| Bile Acid | GPBA | rat | CHO-K1 | Cr1361-1 | DCr1361-1 | MCr1361-1 |
| Bile Acid | GPBA | mouse | CHO-K1 | Cm1361-1 | DCm1361-1 | MCm1361-1 |
| Bile Acid | GPBA Mutant W83G | human | CHO-K1 | C1361-1MT1 | DC1361-1MT1 | MC1361-1MT1 |
| Bile Acid | GPBA Mutant W83A | human | CHO-K1 | C1361-1MT2 | DC1361-1MT2 | MC1361-1MT2 |
| Bile Acid | GPBA Mutant V88L | human | CHO-K1 | C1361-1MT3 | DC1361-1MT3 | MC1361-1MT3 |
| Bile Acid | GPBA Mutant Y89A | human | CHO-K1 | C1361-1MT4 | DC1361-1MT4 | MC1361-1MT4 |
| Bile Acid | GPBA Mutant Y89H | human | CHO-K1 | C1361-1MT5 | DC1361-1MT5 | MC1361-1MT5 |
| Bile Acid | GPBA Mutant F96A | human | CHO-K1 | C1361-1MT6 | DC1361-1MT6 | MC1361-1MT6 |
| Bile Acid | GPBA Mutant W237A | human | CHO-K1 | C1361-1MT7 | DC1361-1MT7 | MC1361-1MT7 |
| Bile Acid | GPBA Mutant W240A | human | CHO-K1 | C1361-1MT8 | DC1361-1MT8 | MC1361-1MT8 |
| Bombesin | BB1 | human | HEK293T | C1211 | DC1211 | MC1211 |
| Bombesin | BB1 | rat | C6 | C1211-1 | DC1211-1 | MC1211-1 |
| Bombesin | BB2 | human | HEK293T | C1215 | DC1215 | MC1215 |
| Bombesin | BB3 | human | HEK293T | C1214 | DC1214 | MC1214 |
| Bombesin | BB3 | human | HEK293T | H1214 | DH1214 | MH1214 |
| Bradykinin | B1 | human | HEK293T | C1198a | DC1198a | MC1198a |
| Bradykinin | B1 | mouse | HEK293T | Cm1198 | DCm1198 | MCm1198 |
| Bradykinin | B2 | human | HEK293T | H1199 | DH1199 | MH1199 |
| Bradykinin | B2 | mouse | HEK293T | Cm1199 | DCm1199 | MCm1199 |
| Bradykinin | B2 | rat | HEK293T | Cr1199 | DCr1199 | MCr1199 |
| Bradykinin | B2 | dog | HEK293T | cd1199 | DCd1199 | MCd1199 |
| Bradykinin | B2 | rhesus monkey | HEK293T | Cpr1199 | DCpr1199 | MCpr1199 |
| Bradykinin | B2 | guinea pig | HEK293T | Cc1199 | DCc1199 | MCc1199 |
| Bradykinin | B2 | rabbit | HEK293T | Cb1199 | DCb1199 | MCb1199 |
| Calcitonin | CALCRL | human | HEK293T | C1232 | DC1232 | MC1232 |
| Calcitonin | CALCRL | human | CHO-K1 | C1232-1 | DC1232-1 | MC1232-1 |
| Calcitonin | CGRP | human | CHO-K1 | C1515-1 | DC1515-1 | MC1515-1 |
| Calcitonin | AM1 | human | CHO-K1 | C1516-1 | DC1516-1 | MC1516-1 |
| Calcitonin | AM2 | human | CHO-K1 | C1517-1 | DC1517-1 | MC1517-1 |
| Calcitonin | CT | human | HEK293T | H1231 | DH1231 | MH1231 |
| Calcitonin | CT | human | CHO-K1 | C1231-1A | DC1231-1A | MC1231-1A |
| Calcitonin | CT | human | CHO-K1 | C1231-1B | DC1231-1B | MC1231-1B |
| Calcitonin | AMY1 | human | CHO-K1 | C1509-1 | DC1509-1 | MC1509-1 |
| Calcitonin | AMY1 | human | CHO-K1 | C1509-1a | DC1509-1a | MC1509-1a |
| Calcitonin | AMY2 | human | CHO-K1 | C1510-1a | DC1510-1a | MC1510-1a |
| Calcitonin | AMY2 | human | CHO-K1 | C1510-1b | DC1510-1b | MC1510-1b |
| Calcitonin | AMY3 | human | CHO-K1 | C1511-1a | DC1511-1a | MC1511-1a |
| Calcium-Sensing | CaSR | human | HEK293T | C1233 | DC1233 | MC1233 |
| Calcium-Sensing | CaSR | rat | HEK293T | Hr1233 | DHr1233 | MHr1233 |
| Cannabinoid | CB1 | human | HEK293T | C1229 | DC1229 | MC1229 |
| Cannabinoid | CB1 | human | CHO-K1 | C1229-1a | DC1229-1a | MC1229-1a |
| Cannabinoid | CB1 | human | CHO-K1 | C1229-1 | DC1229-1 | MC1229-1 |
| Cannabinoid | CB1a | human | CHO-K1 | C1512-1 | DC1512-1 | MC1512-1 |
| Cannabinoid | CB1b | human | CHO-K1 | C1513-1 | DC1513-1 | MC1513-1 |
| Cannabinoid | CB1 | mouse | CHO-K1 | Cm1229-1A | DCm1229-1A | MCm1229-1A |
| Cannabinoid | CB1 | mouse | CHO-K1 | Cm1229-1B | DCm1229-1B | MCm1229-1B |
| Cannabinoid | CB1 | dog | HEK293T | Cd1229 | DCd1229 | MCd1229 |
| Cannabinoid | CB1 | dog | HEK293T | Cd1229a | DCd1229a | MCd1229a |
| Cannabinoid | CB1 | dog | HEK293T | Cd1229b | DCd1229b | MCd1229b |
| Cannabinoid | CB1 MUTANT B | human | CHO-K1 β-Arrestin2 | CA1513BA2-1 | DCA1513BA2-1 | MCA1513BA2-1 |
| Cannabinoid | CB2 | human | CHO-K1 | C1230-1 | DC1230-1 | MC1230-1 |
| Cannabinoid | CB2 | human | CHO-K1 | C1230-1a | DC1230-1a | MC1230-1a |
| Cannabinoid | CB2 | human | CHO-K1 β-Arrestin2 | CA1230BA2-1 | DCA1230BA2-1 | MCA1230BA2-1 |
| Cannabinoid | CB2 | rat | CHO-K1 | Cr1230-1 | DCr1230-1 | MCr1230-1 |
| Cannabinoid | CB2 | rat | CHO-K1 | Cr1230-1a | DCr1230-1a | MCr1230-1a |
| Cannabinoid | CB2 | mouse | CHO-K1 β-Arrestin2 | CAm1230BA2-1 | DCAm1230BA2-1 | MCAm1230BA2-1 |
| Cannabinoid | CB2 | mouse | CHO-K1 | Cm1230-1 | DCm1230-1 | MCm1230-1 |
| Cannabinoid | CB2 | mouse | CHO-K1 | Cm1230-1a | DCm1230-1a | MCm1230-1a |
| Cannabinoid | CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1 | DCAr1230BA2-1 | MCAr1230BA2-1 |
| Cannabinoid | CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1a | DCAr1230BA2-1a | MCAr1230BA2-1a |
| Cannabinoid | GPR55 | human | HEK293T | H1113 | H1113 | H1113 |
| Cannabinoid | GPR55 | human | HEK293T | C1113b | DC1113b | MC1113b |
| Cannabinoid | GPR55 | human | HEK293T | C1113d | DC1113d | MC1113d |
| Chemokine | CCR1 | human | HEK293T | C1009 | DC1009 | MC1009 |
| Chemokine | CCR1 | human | HEK293T Gαqi5 | CG1009 | DCG1009 | MCG1009 |
| Chemokine | CCR2 | human | HEK293T | C1010 | DC1010 | MC1010 |
| Chemokine | CCR3 | human | HEK293T | C1011 | DC1011 | MC1011 |
| Chemokine | CCR3 | human | HEK293T Gαqi5 | CG1011 | DCG1011 | MCG1011 |
| Chemokine | CCR4 | human | HEK293T | C1012 | DC1012 | MC1012 |
| Chemokine | CCR4 | human | HEK293T Gαqi5 | CG1012 | DCG1012 | MCG1012 |
| Chemokine | CCR5 | human | HEK293T | C1013a | DC1013a | MC1013a |
| Chemokine | CCR5 | human | HEK293T | C1013b | DC1013b | MC1013b |
| Chemokine | CCR5 | human | HEK293T Gαqi5 | CG1013 | DCG1013 | MCG1013 |
| Chemokine | CCR6 | human | HEK293T | C1014a | DC1014a | MC1014a |
| Chemokine | CCR6 | human | HEK293T | C1014b | DC1014b | MC1014b |
| Chemokine | CCR6 | mouse | HEK293T | Cm1014 | DCm1014 | MCm1014 |
| Chemokine | CCR7 | human | HEK293T | C1015 | DC1015 | MC1015 |
| Chemokine | CCR7 | human | HEK293T Gαqi5 | CG1015 | DCG1015 | MCG1015 |
| Chemokine | CCR8 | human | HEK293T | C1016 | DC1016 | MC1016 |
| Chemokine | CCR8 | human | HEK293T | C1016a | DC1016a | MC1016a |
| Chemokine | CCR8 | human | HEK293T Gαqi5 | CG1016 | DCG1016 | MCG1016 |
| Chemokine | CCR9 | dog | HEK293T Gαqi5 | CGd1017 | DCGd1017 | MCGd1017 |
| Chemokine | CCR9 | human | HEK293T | C1017 | DC1017 | MC1017 |
| Chemokine | CCR9 | human | HEK293T | C1017a | DC1017a | MC1017a |
| Chemokine | CCR9 | human | HEK293T Gαqi5 | CG1017 | DCG1017 | MCG1017 |
| Chemokine | CCR9 | human | HEK293T Gαqi5 | CG1017A | DCG1017A | MCG1017A |
| Chemokine | CCR9 | mouse | HEK293T | Cm1017 | DCm1017 | MCm1017 |
| Chemokine | CCR9 | mouse | HEK293T Gαqi5 | CGm1017 | DCGm1017 | MCGm1017 |
| Chemokine | CCR9 | rat | HEK293T Gαqi5 | CGr1017 | DCGr1017 | MCGr1017 |
| Chemokine | CCR10 | human | HEK293T | C1018 | DC1018 | MC1018 |
| Chemokine | CCR10 | human | CHO-K1 Gαqi5 | CG1018-1 | DCG1018-1 | MCG1018-1 |
| Chemokine | CMKLR1 | human | HEK293T | C1147 | DC1147 | MC1147 |
| Chemokine | CMKLR1 | human | HEK293T Gαqi5 | CG1147 | DCG1147 | MCG1147 |
| Chemokine | CX3CR1 | human | HEK293T | C1008 | DC1008 | MC1008 |
| Chemokine | CX3CR1 | human | HEK293T Gαqi5 | CG1008a | DCG1008a | MCG1008a |
| Chemokine | CX3CR1 | human | HEK293T Gαqi5 | CG1008b | DCG1008b | MCG1008b |
| Chemokine | CXCR1 | human | HEK293T | C1001a | DC1001a | MC1001a |
| Chemokine | CXCR1 | human | HEK293T Gαqi5 | CG1001 | DCG1001 | MCG1001 |
| Chemokine | CXCR2 | human | HEK293T | C1002 | DC1002 | MC1002 |
| Chemokine | CXCR2 | human | HEK293T Gαqi5 | CG1002 | DCG1002 | MCG1002 |
| Chemokine | CXCR3 | human | HEK293T | C1003 | DC1003 | MC1003 |
| Chemokine | CXCR3 | human | HEK293T | C1003a | DC1003a | MC1003a |
| Chemokine | CXCR3 | human | HEK293T Gαqi5 | CG1003 | DCG1003 | MCG1003 |
| Chemokine | CXCR4 | human | HEK293T | C1004-1 | DC1004-1 | MC1004-1 |
| Chemokine | CXCR4 | human | HEK293T Gαqi5 | CG1004 | DCG1004 | MCG1004 |
| Chemokine | CXCR5 | human | HEK293T | C1005 | DC1005 | MC1005 |
| Chemokine | CXCR5 | human | HEK293T | C1005a | DC1005a | MC1005a |
| Chemokine | CXCR5 | human | CHO-K1 | C1005-1 | DC1005-1 | MC1005-1 |
| Chemokine | CXCR5 | human | CHO-K1 | C1005-1a | DC1005-1a | MC1005-1a |
| Chemokine | CXCR6 | human | HEK293T | C1006 | DC1006 | MC1006 |
| Chemokine | CXCR6 | human | CHO-K1 | C1006-1 | DC1006-1 | MC1006-1 |
| Chemokine | CXCR6 | human | HEK293T Gαqi5 | CG1006 | DCG1006 | MCG1006 |
| Chemokine | CXCR7 | human | HEK293T | C1150 | DC1150 | MC1150 |
| Chemokine | CXCR7 | human | HEK293T | CA1150BA2a | DCA1150BA2a | MCA1150BA2a |
| Chemokine | XCR1 | human | HEK293T | C1007 | DC1007 | MC1007 |
| Chemokine | XCR1 | human | HEK293T Gαqi5 | CG1007 | DCG1007 | MCG1007 |
| Cholecystokinin | CCK1 | human | CHO-K1 | C1038-1a | DC1038-1a | MC1038-1a |
| Cholecystokinin | CCK1 | human | HEK293T | C1038 | DC1038 | MC1038 |
| Cholecystokinin | CCK2 | human | HEK293T | H1039 | DH1039 | MH1039 |
| Citric Acid Cycle Intermediates | GPR91 | human | CHO-K1 | C1144-1 | DC1144-1 | MC1144-1 |
| Citric Acid Cycle Intermediates | GPR91 | mouse | CHO-K1 | Cm1144-1 | DCm1144-1 | MCm1144-1 |
| Citric Acid Cycle Intermediates | GPR91 | rat | CHO-K1 | Cr1144-1 | DCr1144-1 | MCr1144-1 |
| Citric Acid Cycle Intermediates | GPR91 | human | CHO-K1 B-Arrestin2 | CA1141BA2-1 | DCA1141BA2-1 | MCA1141BA2-1 |
| Citric Acid Cycle Intermediates | GPR99 | human | CHO-K1 | C1132-1 | DC1132-1 | MC1132-1 |
| Corticotrophin-Releasing Factor | CRF1 | human | HEK293T | C1040 | DC1040 | MC1040 |
| Corticotrophin-Releasing Factor | CRF1 | human | HEK293T Gαqi5 | CG1040 | DCG1040 | MCG1040 |
| Corticotrophin-Releasing Factor | CRF2 | human | HEK293T | C1041 | DC1041 | MC1041 |
| Corticotrophin-Releasing Factor | CRF2 | human | HEK293TGα16 | CG1041 | DCG1041 | MCG1041 |
| Dopamine | D1 | human | HEK293T | C1335 | DC1335 | MC1335 |
| Dopamine | D1 | human | HEK293T | H1335 | DH1335 | MH1335 |
| Dopamine | D2 | human | HEK293T | C1336 | DC1336 | MC1336 |
| Dopamine | D2 | human | HEK293T | C1336a | DC1336a | MC1336a |
| Dopamine | D2 Ghrelin | human | HEK293T | C1514 | DC1514 | MC1514 |
| Dopamine | D3 | human | HEK293T Gqi5 | CG1337 | DCG1337 | MCG1337 |
| Dopamine | D4 | human | HEK293T | C1338 | DC1338 | MC1338 |
| Dopamine | D4 | human | HEK293T Gαqi5 | CG1338 | DCG1338 | MCG1338 |
| Dopamine | D5 | human | HEK293T | C1339 | DC1339 | MC1339 |
| Endothelin | ETA | human | CHO-K1 | C1216-1 | DC1216-1 | MC1216-1 |
| Endothelin | ETA | rat | CHO-K1 | Cr1216-1 | DCr1216-1 | MCr1216-1 |
| Endothelin | ETB | human | CHO-K1 | C1217-1 | DC1217-1 | MC1217-1 |
| Free Fatty Acid | GPR119 | human | CHO-K1 | C1298-1a | DC1298-1a | MC1298-1a |
| Free Fatty Acid | GPR119 | human | HEK293T | C1298 | DC1298 | MC1298 |
| Free Fatty Acid | GPR119 | mouse | CHO-K1 | Cm1298-1 | DCm1298-1 | MCm1298-1 |
| Free Fatty Acid | GPR120 | human | HEK293T | C1294 | DC1294 | MC1294 |
| Free Fatty Acid | GPR120 | human | HEK293T Gαqi5 | CG1294 | DCG1294 | MCG1294 |
| Free Fatty Acid | GPR120 | human | CHO-K1 | C1294-1 | DC1294-1 | MC1294-1 |
| Free Fatty Acid | GPR120L | human | HEK293T | C1522 | DC1522 | MC1522 |
| Free Fatty Acid | GPR120L | human | HEK293T β-Arrestin2 | CA1522 | DCA1522 | MCA1522 |
| Free Fatty Acid | GPR120 | mouse | HEK293T Gαqi5 | CGm1294 | DCGm1294 | MCGm1294 |
| Free Fatty Acid | GPR120 | rat | HEK293T | Cr1294 | DCr1294 | MCr1294 |
| Free Fatty Acid | GPR40 | cynomolgus monkey | CHO-K1 | Cpc1101-1 | DCpc1101-1 | MCpc1101-1 |
| Free Fatty Acid | GPR40 | cynomolgus monkey | CHO-K1 | CApr1101-1 | DCApr1101-1 | MCApr1101-1 |
| Free Fatty Acid | GPR40 | cynomolgus monkey | CHO-K1 β-Arrestin2 | CApc1101-1 | DCApc1101-1 | MCApc1101-1 |
| Free Fatty Acid | GPR40 | dog | CHO-K1 | Cd1101-1 | DCd1101-1 | MCd1101-1 |
| Free Fatty Acid | GPR40 | human | HEK293T | C1101 | DC1101 | MC1101 |
| Free Fatty Acid | GPR40 | human | CHO-K1 | C1101-1 | DC1101-1 | MC1101-1 |
| Free Fatty Acid | GPR40 | human | CHO-K1 | C1101-1A | DC1101-1A | MC1101-1A |
| Free Fatty Acid | GPR40 | human | CHO-K1 β-Arrestin2 | CA1101-1 | DCA1101-1 | MCA1101-1 |
| Free Fatty Acid | GPR40 | mouse | HEK293T | Cm1101 | DCm1101 | MCm1101 |
| Free Fatty Acid | GPR40 | rat | HEK293T | Cr1101 | DCr1101 | MCr1101 |
| Free Fatty Acid | GPR40 | rat | CHO-K1 | Cr1101-1 | DCr1101-1 | MCr1101-1 |
| Free Fatty Acid | GPR40 | rhesus monkey | CHO-K1 | Cpr1101-1 | DCpr1101-1 | MCpr1101-1 |
| Free Fatty Acid | GPR40 | rat | CHO-K1 β-Arrestin2 | CAr1101-1 | DCAr1101-1 | MCAr1101-1 |
| Free Fatty Acid | GPR41 | human | HEK293T | C1102 | DC1102 | MC1102 |
| Free Fatty Acid | GPR41 | human | CHO-K1 Gα16 | C1102-1 | DCG1102-1 | MC1102-1 |
| Free Fatty Acid | GPR41 | human | HEK293T Gαqi5 | CG1102 | DCG1102 | MCG1102 |
| Free Fatty Acid | GPR41 | mouse | CHO-K1 Gα16 | CGm1102-1 | DCGm1102-1 | MCGm1102-1 |
| Free Fatty Acid | GPR41 | rat | HEK293T | Cr1102 | DCr1102 | MCr1102 |
| Free Fatty Acid | GPR43 | human | HEK293T | C1104 | DC1104 | MC1104 |
| Free Fatty Acid | GPR43 | human | CHO-K1 | C1104-1 | DC1104-1 | MC1104-1 |
| Free Fatty Acid | GPR43 | human | CHO-K1 Gα16 | HG1104-1 | DHG1104-1 | MHG1104-1 |
| Free Fatty Acid | GPR43 | mouse | HEK293T | Cm1104 | DCm1104 | MCm1104 |
| Free Fatty Acid | GPR43 | rat | HEK293T | Cr1104 | DCr1104 | MCr1104 |
| Free Fatty Acid | GPR43 | dog | CHO-K1 | Cd1104-1A | DCd1104-1A | MCd1104-1A |
| Free Fatty Acid | GPR43 | dog | CHO-K1 | Cd1104-1B | DCd1104-1B | MCd1104-1B |
| Free Fatty Acid | GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1A | DCpc1104-1A | MCpc1104-1A |
| Free Fatty Acid | GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1B | DCpc1104-1B | MCpc1104-1B |
| Free Fatty Acid | GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1A | DCpr1104-1A | MCpr1104-1A |
| Free Fatty Acid | GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1B | DCpr1104-1B | MCpr1104-1B |
| Free Fatty Acid | GPR84 | human | CHO-K1 | C1137-1 | DC1137-1 | MC1137-1 |
| Free Fatty Acid | GPR84 | human | CHO-K1 Gαqi5 | CG1137-1 | DCG1137-1 | MCG1137-1 |
| Frizzled | SMO | human | HEK293T | C1442 | DC1442 | MC1442 |
| Frizzled | SMO | human | HEK293T | H1442 | DH1442 | MH1442 |
| Galanin | GAL1 | human | CHO-K1 Gαqi5 | CG1178-1 | DCG1178-1 | MCG1178-1 |
| Galanin | GAL1 | human | HEK293T | C1178 | DC1178 | MC1178 |
| Galanin | GAL2 | human | CHO-K1 | C1179-1 | DC1179-1 | MC1179-1 |
| Ghrelin | Ghrelin | human | HEK293T | C1197b | DC1197b | MC1197b |
| Ghrelin | Ghrelin | human | CHO-K1 | C1197-1 | DC1197-1 | MC1197-1 |
| Ghrelin | Ghrelin | mouse | HEK293T | Cm1197 | DCm1197 | MCm1197 |
| Glucagon | GHRH | human | HEK293T | C1291 | DC1291 | MC1291 |
| Glucagon | GIP | human | HEK293T | C1290 | DC1290 | MC1290 |
| Glucagon | GIP | human | HEK293T β-Arrestin2 | CA1290 | DCA1290 | MCA1290 |
| Glucagon | GIP | human | HEK293T β-Arrestin2 | CA1290BA1 | DCA1290BA1 | MCA1290BA1 |
| Glucagon | GIP | mouse | HEK293T | Cm1290 | DCm1290 | MCm1290 |
| Glucagon | GIP | rat | HEK293T | Cr1290 | DCr1290 | MCr1290 |
| Glucagon | GIP | dog | HEK293T | Cd1290 | DCd1290 | MCd1290 |
| Glucagon | GIP | dog | HEK293T | Cd1290a | DCd1290a | MCd1290a |
| Glucagon | GIP | rabbit | HEK293T | Cb1290 | DCb1290 | MCb1290 |
| Glucagon | GIP | pig | HEK293T | Cp1290 | DCp1290 | MCp1290 |
| Glucagon | GIP | rhesus monkey | HEK293T | Cpr1290 | DCpr1290 | MCpr1290 |
| Glucagon | GIP | rhesus monkey | HEK293T | Cpr1290a | DCpr1290a | MCpr1290a |
| Glucagon | GIP | ferret | HEK293T | Cf1290 | DCf1290 | MCf1290 |
| Glucagon | GIP | ferret | HEK293T | Cf1290a | DCf1290a | MCf1290a |
| Glucagon | GLP-1 | human | HEK293T | C1267 | DC1267 | MC1267 |
| Glucagon | GLP-1 | human | CHO-K1 | C1267-1 | DC1267-1 | MC1267-1 |
| Glucagon | GLP-1 | human | CHO-K1 | C1267-1a | DC1267-1a | MC1267-1a |
| Glucagon | GLP-1 | human | CHO-K1 β-Arrestin2 | CA1267-1 | DCA1267-1 | MCA1267-1 |
| Glucagon | GLP-1 | human | HEK293T β-Arrestin2 | CA1267BA2 | DCA1267BA2 | MCA1267BA2 |
| Glucagon | GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1 | DCpc1267-1 | MCpc1267-1 |
| Glucagon | GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1a | DCpc1267-1a | MCpc1267-1a |
| Glucagon | GLP-1 | rat | CHO-K1 | Cr1267-1 | DCr1267-1 | MCr1267-1 |
| Glucagon | GLP-1 | dog | CHO-K1 | Cd1267-1 | DCd1267-1 | MCd1267-1 |
| Glucagon | GLP-1 | dog | HEK293T | Cd1267-1a | DCd1267-1a | MCd1267-1a |
| Glucagon | GLP-1 | mouse | CHO-K1 | Cm1267-1 | DCm1267-1 | MCm1267-1 |
| Glucagon | GLP-1 | mouse | CHO-K1 | Cm1267-1a | DCm1267-1a | MCm1267-1a |
| Glucagon | GLP-1 | pig | CHO-K1 | Cp1267-1 | DCp1267-1 | MCp1267-1 |
| Glucagon | GLP-2 | human | HEK293T | C1268 | DC1268 | MC1268 |
| Glucagon | GLP-2 | rat | HEK293T | Cr1268 | DCr1268 | MCr1268 |
| Glucagon | Glucagon | human | HEK293T | C1266 | DC1266 | MC1266 |
| Glucagon | Glucagon | dog | HEK293T | Cd1266 | DCd1266 | MCd1266 |
| Glucagon | Glucagon | pig | HEK293T | Cp1266 | DCp1266 | MCp1266 |
| Glucagon | Glucagon | rat | HEK293T | Cr1266 | DCr1266 | MCr1266 |
| Glucagon | Glucagon | human | HEK293T | C1266A | DC1266A | MC1266A |
| Glucagon | Glucagon | human | CHO-K1 | C1266-1 | DC1266-1 | MC1266-1 |
| Glucagon | Glucagon | human | CHO-K1 | C1266-1a | DC1266-1a | MC1266-1a |
| Glucagon | Glucagon | human | CHO-K1 β-Arrestin2 | CA1266-1 | DCA1266-1 | MCA1266-1 |
| Glucagon | Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1 | DCpc1266-1 | MCpc1266-1 |
| Glucagon | Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1a | DCpc1266-1a | MCpc1266-1a |
| Glucagon | Glucagon | cynomolgus monkey | HEK293T | Cpc1266 | DCpc1266 | MCpc1266 |
| Glucagon | Glucagon | cynomolgus monkey | HEK293T | Cpc1266a | DCpc1266a | MCpc1266a |
| Glucagon | Secretin | human | CHO-K1 | C1228-1 | DC1228-1 | MC1228-1 |
| Glycoprotein Hormone | TSH | human | HEK293T | H1177 | DH1177 | MH1177 |
| Glycoprotein Hormone | TSH | rat | HEK293T | C1177-1 | DC1177-1 | MC1177-1 |
| Gonadotrophin-Releasing Hormone | GnRH | human | HEK293T | C1283 | DC1283 | MC1283 |
| Gonadotrophin-Releasing Hormone | GnRH | dog | HEK293T | Cd1283 | DCd1283 | MCd1283 |
| Gonadotrophin-Releasing Hormone | FSHR | human | HEK293T | C1175 | DC1175 | MC1175 |
| Histamine | H1 | human | HEK293T | C1027 | DC1027 | MC1027 |
| Histamine | H1 | mouse | HEK293T | Cm1027 | DCm1027 | MCm1027 |
| Histamine | H2 | human | HEK293T | C1028 | DC1028 | MC1028 |
| Histamine | H3 | human | HEK293T | C1029 | DC1029 | MC1029 |
| Histamine | H3 | human | HEK293T Gαqi5 | CG1029 | DCG1029 | MCG1029 |
| Histamine | H3 | mouse | HEK293T | Cm1029 | DCm1029 | MCm1029 |
| Histamine | H3 | mouse | CHO-K1 | Cm1029-1 | DCm1029-1 | MCm1029-1 |
| Histamine | H4 | human | HEK293T | C1030 | DC1030 | MC1030 |
| Histamine | H4 | human | HEK293T Gαqi5 | CG1030 | DCG1030 | MCG1030 |
| Histamine | H4 | human | HEK293T β-Arrestin2 | CA1030BA2 | DCA1030BA2 | MCA1030BA2 |
| Histamine | H4 | mouse | HEK293T | Cm1030 | DCm1030 | MCm1030 |
| Histamine | H4 | mouse | HEK293T Gαqi5 | CGm1030 | DCGm1030 | MCGm1030 |
| Hydroxycarboxylic acid | GPR81 | human | HEK293T | |||
| KiSS1-Derived Peptide | KiSS1 | human | CHO dhfr- | C1036 | DC1036 | MC1036 |
| KiSS1-Derived Peptide | KiSS1 | rat | CHO dhfr- | C1036-1 | DC1036-1 | MC1036-1 |
| Leukotriene/Lipoxin | BLT1 | human | HEK293T | H1165a | DH1165a | H1165a |
| Leukotriene/Lipoxin | BLT2 | human | HEK293T | C1272 | DC1272 | MC1272 |
| Leukotriene/Lipoxin | BLT2 | human | HEK293T | C1272A | DC1272A | MC1272A |
| Leukotriene/Lipoxin | BLT2 | human | HEK293T | C1272b | DC1272b | MC1272b |
| Leukotriene/Lipoxin | BLT2 | human | HEK293T | C1272c | DC1272c | MC1272c |
| Leukotriene/Lipoxin | BLT2 | monkey | HEK293T | Cp1272a | DCp1272a | MCp1272a |
| Leukotriene/Lipoxin | BLT2 | monkey | HEK293T | Cp1272 | DCp1272 | MCp1272 |
| Leukotriene/Lipoxin | BLT2 | mouse | HEK293T | Cm1272a | DCm1272a | MCm1272a |
| Leukotriene/Lipoxin | BLT2 | mouse | HEK293T | Cm1272 | DCm1272 | MCm1272 |
| Leukotriene/Lipoxin | CysLT1 | human | HEK293T | C1308 | DC1308 | MC1308 |
| Leukotriene/Lipoxin | CysLT2 | human | HEK293T | C1307 | DC1307 | MC1307 |
| Leukotriene/Lipoxin | OXE | human | HEK293T | |||
| Lysophospholipid | GPR87 | human | RH7777 | C1140-6 | DC1140-6 | MC1140-6 |
| Lysophospholipid | LPA1 | human | RH7777 | C1048-6 | DC1048-6 | MC1048-6 |
| Lysophospholipid | LPA1 | mouse | RH7777 | Cm1048-6A | DCm1048-6A | MCm1048-6A |
| Lysophospholipid | LPA1 | mouse | RH7777 | Cm1048-6B | DCm1048-6B | MCm1048-6B |
| Lysophospholipid | LPA1 | rat | RH7777 | Cr1048-6B | DCr1048-6B | MCr1048-6B |
| Lysophospholipid | LPA2 | human | RH7777 | C1050-6 | DC1050-6 | MC1050-6 |
| Lysophospholipid | LPA3 | human | RH7777 | C1053-6 | DC1053-6 | MC1053-6 |
| Lysophospholipid | LPA3 | human | RH7777 | C1053-6a | DC1053-6a | MC1053-6a |
| Lysophospholipid | LPA4 | human | CHO-K1 | C1087-1a | DC1087-1a | MC1087-1a |
| Lysophospholipid | LPA4 | human | CHO-K1 | C1087-1b | DC1087-1b | MC1087-1b |
| Lysophospholipid | LPA5 | human | RH7777 | C1145-6 | DC1145-6 | MC1145-6 |
| Lysophospholipid | LPA5 | mouse | RH7777 | Cm1145-6 | DCm1145-6 | MCm1145-6 |
| Lysophospholipid | S1P1 | human | CHO-K1 | C1047-1 | DC1047-1 | MC1047-1 |
| Lysophospholipid | S1P1 | human | CHO-K1 Gαqi5 | CG1047-1 | DCG1047-1 | MCG1047-1 |
| Lysophospholipid | S1P2 | human | CHO-K1 | C1051-1 | DC1051-1 | MC1051-1 |
| Lysophospholipid | S1P2 | human | CHO-K1 Gαqi5 | CG1051-1 | DCG1051-1 | MCG1051-1 |
| Lysophospholipid | S1P2 | mouse | CHO-K1 | Cm1051-1 | DCm1051-1 | MCm1051-1 |
| Lysophospholipid | S1P2 | rat | CHO-K1 | Cr1051-1 | DCr1051-1 | MCr1051-1 |
| Lysophospholipid | S1P3 | human | RH7777 | C1049-6 | DC1049-6 | MC1049-6 |
| Lysophospholipid | S1P3 | human | CHO-K1 | C1049-1 | DC1049-1 | MC1049-1 |
| Lysophospholipid | S1P3 | human | CHO-K1 Gαqi5 | CG1049-1 | DCG1049-1 | MCG1049-1 |
| Lysophospholipid | S1P3 | mouse | CHO-K1 Gαqi5 | CGm1049-1 | DCGm1049-1 | MCGm1049-1 |
| Lysophospholipid | S1P3 | rat | CHO-K1 Gαqi5 | CGr1049-1 | DCGr1049-1 | MCGr1049-1 |
| Lysophospholipid | S1P4 | human | CHO-K1 Gαqi5 | CG1052-1 | DCG1052-1 | MCG1052-1 |
| Lysophospholipid | S1P4 | mouse | CHO-K1 Gαqi5 | CGm1052-1 | DCGm1052-1 | MCGm1052-1 |
| Lysophospholipid | S1P4 | rat | CHO-K1 Gαqi5 | CGr1052-1 | DCGr1052-1 | MCGr1052-1 |
| Lysophospholipid | S1P5 | human | CHO-K1 | C1054-1 | DC1054-1 | MC1054-1 |
| Lysophospholipid | S1P5 | human | CHO-K1 Gαqi5 | CG1054-1 | DCG1054-1 | MCG1054-1 |
| Melanin-Concentrating Hormone | MCH1 | human | HEK293T Gαqi5 | C1031-3 | DC1031-3 | MC1031-3 |
| Melanin-Concentrating Hormone | MCH1 | rat | HEK293T Gαqi5 | C1031-4 | DC1031-4 | MC1031-4 |
| Melanin-Concentrating Hormone | MCH2 | human | CHO dhfr- | C1032 | DC1032 | MC1032 |
| Melanocortin | MC1 | human | HEK293T | C1340 | DC1340 | MC1340 |
| Melanocortin | MC4 | human | HEK293T | H1343 | H1343 | H1343 |
| Melatonin | MT1 | human | CHO-K1 | C1223-1 | DC1223-1 | MC1223-1 |
| Melatonin | MT2 | human | HEK293T Gαqi5 | C1224 | DC1224 | MC1224 |
| Melatonin | MT2 | mouse | HEK293T | Cm1224 | DCm1224 | MCm1224 |
| Melatonin | MT2 | rat | HEK293T | Cr1224 | DCr1224 | MCr1224 |
| Metabotropic Glutamate | mGlu1 | human | CHO-K1 | C1188-1 | DC1188-1 | MC1188-1 |
| Metabotropic Glutamate | mGlu2 | human | HEK293T | C1189a | DC1189a | MC1189a |
| Metabotropic Glutamate | mGlu2 | human | HEK293T Gqi5 | HG1189Gi | DHG1189Gi | MHG1189Gi |
| Metabotropic Glutamate | mGlu2 | human | HEK293T Gαqi5 | HG1189 | HG1189 | HG1189 |
| Metabotropic Glutamate | mGlu2 | human | HEK293T Gαqi5 | HG1189a | HG1189a | HG1189a |
| Metabotropic Glutamate | mGlu2 | rat | HEK293T Gαqi5 | HGr1189b | DHGr1189b | MHGr1189b |
| Metabotropic Glutamate | mGlu3 | human | HEK293T Gαqi5 | CG1190 | DCG1190 | MCG1190 |
| Metabotropic Glutamate | mGlu4 | dog | CHO-K1 Gαqi5 | HGd1191-1 | DHGd1191-1 | MHGd1191-1 |
| Metabotropic Glutamate | mGlu4 | human | HEK293T | C1191a | DC1191a | MC1191a |
| Metabotropic Glutamate | mGlu4 | human | HEK293T Gαqi5 | CG1191 | DCG1191 | MCG1191 |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1a | DHGm1191-1a | MHGm1191-1a |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1b | DHGm1191-1b | MHGm1191-1b |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1c | DHGm1191-1c | MHGm1191-1c |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1d | DHGm1191-1d | MHGm1191-1d |
| Metabotropic Glutamate | mGlu4 | rat | HEK293T | Cr1191 | DCr1191 | MCr1191 |
| Metabotropic Glutamate | mGlu4 | human | HEK293T Gαqi5 | CG1191a | DCG1191a | MCG1191a |
| Metabotropic Glutamate | mGlu5 | human | HEK293T | C1192 | DC1192 | MC1192 |
| Metabotropic Glutamate | mGlu5 | human | HEK293T B-ARRESTIN2 | CA1192BA2 | DCA1192BA2 | MCA1192BA2 |
| Metabotropic Glutamate | mGlu6 | human | HEK293T | C1193 | DC1193 | MC1193 |
| Metabotropic Glutamate | mGlu6 | human | HEK293T Gαqi5 | CG1193 | DCG1193 | MCG1193 |
| Metabotropic Glutamate | mGlu7 | human | HEK293T | C1194 | DC1194 | MC1194 |
| Metabotropic Glutamate | mGlu7 | human | HEK293T Gαqi5 | CG1194 | DCG1194 | MCG1194 |
| Metabotropic Glutamate | mGlu8 | human | HEK293T | C1195 | DC1195 | MC1195 |
| Metabotropic Glutamate | mGlu8 | human | HEK293T | C1195a | DC1195a | MC1195a |
| Metabotropic Glutamate | mGlu8 | human | HEK293T Gαqi5 | CG1195 | DCG1195 | MCG1195 |
| Metabotropic Glutamate | mGlu8 | human | CHO-K1 | C1195-1a | DC1195-1a | MC1195-1a |
| Motilin | motilin | human | HEK293T | H1297 | H1297 | H1297 |
| Muscarinic | M1 | human | CHO-K1 | C1022-1 | DC1022-1 | MC1022-1 |
| Muscarinic | M1 | human | CHO-K1 | C1022-1a | DC1022-1a | MC1022-1a |
| Muscarinic | M2 | human | CHO-K1 | C1023-1 | DC1023-1 | MC1023-1 |
| Muscarinic | M3 | human | CHO-K1 | C1024-1 | DC1024-1 | MC1024-1 |
| Muscarinic | M3 | mouse | CHO-K1 | Cm1024-1 | DCm1024-1 | MCm1024-1 |
| Muscarinic | M4 | human | CHO-K1 | C1025-1 | DC1025-1 | MC1025-1 |
| Muscarinic | M4 | human | CHO-K1 Gαqi5 | CG1025-1 | DCG1025-1 | MCG1025-1 |
| Muscarinic | M4 | mouse | CHO-K1 | Cm1025-1 | DCm1025-1 | MCm1025-1 |
| Muscarinic | M5 | human | CHO-K1 | C1026-1 | DC1026-1 | MC1026-1 |
| N-formylpeptide | FPR1 | human | HEK293T | C1243 | DC1243 | MC1243 |
| N-formylpeptide | FPR1 | human | HEK293T | C1243a | DC1243a | MC1243a |
| N-formylpeptide | FPR1 | human | HEK293T Gαqi5 | CG1243 | DCG1243 | MCG1243 |
| N-formylpeptide | FPR2 | human | HEK293T | C1244 | DC1244 | MC1244 |
| N-formylpeptide | FPR2 | human | HEK293T | C1244a | DC1244a | MC1244a |
| N-formylpeptide | FPR3 | human | HEK293T | C1245 | DC1245 | MC1245 |
| Neuromedin U | NMU1 | human | HEK293T | C1122 | DC1122 | MC1122 |
| Neuromedin U | NMU2 | human | HEK293T | C1213 | DC1213 | MC1213 |
| Neuropeptide FF/AF | NPFF1 | human | HEK293T | C1363 | DC1363 | MC1363 |
| Neuropeptide FF/AF | NPFF2 | human | HEK293T Gαqi5 | CG1364 | DCG1364 | MCG1364 |
| Neuropeptide S | NPS | mouse | HEK293T | C1355-1 | DC1355-1 | MC1355-1 |
| Neuropeptide S | NPS | human | HEK293T | C1355a | DC1355a | MC1355a |
| Neuropeptide S | NPS(2) | human | HEK293T | C1356 | DC1356 | MC1356 |
| Neuropeptide S | NPSIle107 | human | HEK293T | C1355-2 | DC1355-2 | MC1355-2 |
| Neuropeptide W/B | NPBW1 | rat | HEK293T Gαqi5 | C1124-1 | DC1124-1 | MC1124-1 |
| Neuropeptide W/B | NPBW1 | human | HEK293T Gαqi5 | C1124 | DC1124 | MC1124 |
| Neuropeptide W/B | NPBW2 | human | HEK293T Gαqi5 | C1133 | DC1133 | MC1133 |
| Neuropeptide Y | Y1 | human | CHO-K1 Gαqi5 | CG1273-1 | DCG1273-1 | MCG1273-1 |
| Neuropeptide Y | Y2 | human | CHO-K1 Gαqi5 | CG1274-1 | DCG1274-1 | MCG1274-1 |
| Neuropeptide Y | Y2 | rat | CHO-K1 | Cr1274-1 | DCr1274-1 | MCr1274-1 |
| Neuropeptide Y | Y4 | human | CHO-K1 | C1300-1 | DC1300-1 | MC1300-1 |
| Neuropeptide Y | Y4 | human | CHO-K1 Gαqi5 | CG1300-1 | DCG1300-1 | MCG1300-1 |
| Neuropeptide Y | Y5 | human | HEK293T | C1275a | DC1275a | MC1275a |
| Neuropeptide Y | Y5 | human | HEK293T Gαqi5 | CG1275 | DCG1275 | MCG1275 |
| Neurotensin | NTS1 | human | CHO-K1 | C1276-1 | DC1276-1 | MC1276-1 |
| Neurotensin | NTS2 | human | CHO-K1 | C1277-1 | DC1277-1 | MC1277-1 |
| Neurotensin | NTS2 | human | HEK293T | C1277 | DC1277 | MC1277 |
| Neurotensin | NTS2 | human | HEK293T | C1277a | DC1277a | MC1277a |
| Nicotinic Acid | GPR109A | human | CHO-K1 | C1370-1 | DC1370-1 | MC1370-1 |
| Nicotinic Acid | GPR109B | human | CHO-K1 | C1059-1 | DC1059-1 | MC1059-1 |
| Nicotinic Acid | GPR81 | human | HEK293T | C1134 | DC1134 | MC1134 |
| Opioid | delta | human | CHO-K1 | C1351-1 | DC1351-1 | MC1351-1 |
| Opioid | delta | human | CHO-K1 Gαqi5 | CG1351-1 | DCG1351-1 | MCG1351-1 |
| Opioid | delta | human | CHO-K1 | CA1351-1 | DCA1351-1 | MCA1351-1 |
| Opioid | delta | rat | CHO dhfr- | C1351 | DC1351 | MC1351 |
| Opioid | kappa | human | CHO-K1 | C1352-1a | DC1352-1a | MC1352-1a |
| Opioid | kappa | human | CHO-K1 Gαqi5 | CG1352-1 | DCG1352-1 | MCG1352-1 |
| Opioid | kappa | human | CHO-K1 | CA1352-1a | DCA1352-1a | MCA1352-1a |
| Opioid | kappa | human | CHO-K1 β-Arrestin2 | CA1352BA2-1 | DCA1352BA2-1 | MCA1352BA2-1 |
| Opioid | kappa | human | HEK293T | C1352 | DC1352 | MC1352 |
| Opioid | kappa | rat | CHO dhfr- | C1352-1 | DC1352-1 | MC1352-1 |
| Opioid | kappa | rat | CHO dhfr- | Cr1352-8 | DCr1352-8 | MCr1352-8 |
| Opioid | mu | human | CHO-K1 | C1350-1a | DC1350-1a | MC1350-1a |
| Opioid | mu | human | CHO-K1 Gαqi5 | CG1350-1a | DCG1350-1a | MCG1350-1a |
| Opioid | mu | human | CHO-K1 | CA1350-1a | DCA1350-1a | MCA1350-1a |
| Opioid | mu | rat | CHO dhfr- | Cr1350-1a | DCr1350-1a | MCr1350-1a |
| Opioid | mu Mutant Y150F | human | CHO-K1 | C1350-1MT1 | DC1350-1MT1 | MC1350-1MT1 |
| Opioid | mu Mutant Y150A | human | CHO-K1 | C1350-1MT2 | DC1350-1MT2 | MC1350-1MT2 |
| Opioid | mu Mutant M153A | human | CHO-K1 | C1350-1MT3 | DC1350-1MT3 | MC1350-1MT3 |
| Opioid | mu Mutant H299N | human | CHO-K1 | C1350-1MT4 | DC1350-1MT4 | MC1350-1MT4 |
| Opioid | mu Mutant H299A | human | CHO-K1 | C1350-1MT5 | DC1350-1MT5 | MC1350-1MT5 |
| Opioid | NOP | human | CHO-K1 | C1354-1 | DC1354-1 | MC1354-1 |
| Opioid | NOP | human | CHO-K1 Gαqi5 | CG1354-1 | DCG1354-1 | MCG1354-1 |
| Opioid | NOP | human | CHO-K1 β-Arrestin2 | CA1354-1 | DCA1354-1 | MCA1354-1 |
| Opioid | NOP | human | HEK293T | C1354a | DC1354a | MC1354a |
| Opioid | NOP | rat | CHO dhfr- | Cr1354 | DCr1354 | MCr1354 |
| Orexin | OX1 | human | CHO-K1 | C1033-1 | DC1033-1 | MC1033-1 |
| Orexin | OX2 | human | CHO-K1 | C1034-1 | DC1034-1 | MC1034-1 |
| Orphan | GPR3 | human | HEK293T | C1091 | DC1091 | MC1091 |
| Orphan | GPR6 | human | HEK293T | C1116 | DC1116 | MC1116 |
| Orphan | GPR6 | human | HEK293T | C1116a | DC1116a | MC1116a |
| Orphan | GPR15 | human | HEK293T | C1069 | DC1069 | MC1069 |
| Orphan | GPR34 | human | HEK293T Gαqi5 | CG1095 | DCG1095 | MCG1095 |
| Orphan | GPR35 | dog | HEK293T Gα16 | CGd1096 | DCGd1096 | MCGd1096 |
| Orphan | GPR35 | dog | CHO-K1 Gα16 | CGd1096-1 | DCGd1096-1 | MCGd1096-1 |
| Orphan | GPR35 | mouse | CHO-K1 | Cm1096-1 | DCm1096-1 | MCm1096-1 |
| Orphan | GPR35 | mouse | CHO-K1 Gα16 | CGm1096-1 | DCGm1096-1 | MCGm1096-1 |
| Orphan | GPR35 (short form) | human | CHO-K1 | C1096-1 | DC1096-1 | MC1096-1 |
| Orphan | GPR35 (short form) | human | CHO-K1 β-Arrestin2 | CA1096-1 | DCA1096-1 | MCA1096-1 |
| Orphan | GPR35 (short form) | human | CHO-K1 Gα16 | CG1096-1 | DCG1096-1 | MCG1096-1 |
| Orphan | GPR35 (short form) | human | HEK293T Gα16 | CG1096 | DCG1096 | MCG1096 |
| Orphan | GPR35 (long form) | human | CHO-K1 β-Arrestin2 | CA1523-1 | DCA1523-1 | MCA1523-1 |
| Orphan | GPR35 (long form) T108M Mutant | human | CHO-K1 β-Arrestin2 | CA1524-1 | DCA1524-1 | MCA1524-1 |
| Orphan | GPR37L1 | human | HEK293T | C1098 | DC1098 | MC1098 |
| Orphan | GPR45 | human | CHO-K1 | CG1106-1 | DCG1106-1 | MCG1106-1 |
| Orphan | GPR45 | human | CHO-K1 | CG1106-1a | DCG1106-1a | MCG1106-1a |
| Orphan | GPR50 | human | HEK293T | C1110 | DC1110 | MC1110 |
| Orphan | GPR52 | human | HEK293T | C1112 | DC1112 | MC1112 |
| Orphan | GPR52 | human | HEK293T | C1112a | DC1112a | MC1112a |
| Orphan | GPR52 | human | HEK293T β-Arrestin2 | CA1112BA2 | DCA1112BA2 | MCA1112BA2 |
| Orphan | GPR85 | human | HEK293T | C1138 | DC1138 | MC1138 |
| Orphan | GPR85 | human | CHO-K1 | C1138-1 | DC1138-1 | MC1138-1 |
| Orphan | GPR88 | human | CHO-K1 | C1141-1 | DC1141-1 | MC1141-1 |
| Orphan | GPR88 | rat | CHO-K1 | Cr1141-1 | DCr1141-1 | MCr1141-1 |
| Orphan | GPR142 | human | HEK293T | C1286 | DC1286 | MC1286 |
| Orphan | GPR142 | human | HEK293T | C1286a | DC1286a | MC1286a |
| Orphan | GPR151 | human | CHO-K1 Gα16 Gαqi5 | CG1181-1 | DCG1181-1 | MCG1181-1 |
| Orphan | GPRC5A | human | HEK293T | CA1525 | DCA1525 | MCA1525 |
| Orphan | MRGX1 | human | CHO dhfr-Gαqi5 | C1256 | DC1256 | MC1256 |
| Orphan | MRGX2 | human | HEK293T Gαqi5 | C1257 | DC1257 | MC1257 |
| Orphan | MRGX2 | human | HEK293T | C1257a | DC1257a | MC1257a |
| Orphan | MRGX2 | rhesus monkey | CHO-K1 | Cpr1257-1 | DCpr1257-1 | MCpr1257-1 |
| Orphan | MRGX2 | human | HEK293T β-Arrestin2 | CA1257aBA2 | DCA1257aBA2 | MCA1257aBA2 |
| Orphan | MRGX2 | human | HEK293T β-Arrestin2 | CA1257bBA2 | DCA1257bBA2 | MCA1257bBA2 |
| Orphan | MRGX4 | human | HEK293T | C1259 | DC1259 | MC1259 |
| Orphan | MAS1 | human | HEK293T | C1225 | DC1225 | MC1225 |
| Oxysterol | EBI2 | human | CHO-K1 Gαqi5 | CG1242-1 | DCG1242-1 | MCG1242-1 |
| Oxysterol | EBI2 | mouse | CHO-K1 Gαqi5 | CGm1242-1 | DCGm1242-1 | MCGm1242-1 |
| Oxysterol | EBI2 | mouse | CHO-K1 | Cm1242-1 | DCm1242-1 | MCm1242-1 |
| Parathyroid Hormone | PTH1 | human | HEK293T | C1301 | DC1301 | MC1301 |
| Parathyroid Hormone | PTH1 | human | HEK293T | C1301-1 | DC1301-1 | MC1301-1 |
| Parathyroid Hormone | PTH2 | human | HEK293T | H1302 | DH1302 | H1302 |
| Platelet-Activating Factor | PAF | human | HEK293T | C1218 | DC1218 | MC1218 |
| Prokineticin | PK1 | human | CHO-K1 | C1128-1 | DC1128-1 | MC1128-1 |
| Prokineticin | PK2 | human | CHO-K1 | C1127-1 | DC1127-1 | MC1127-1 |
| Prokineticin | PK2 | human | CHO-K1 | C1127-1a | DC1127-1a | MC1127-1a |
| Prokineticin | PK2 mutant | human | CHO-K1 | C1127CT-1 | DC1127DCT-1 | MC1127MCT-1 |
| Prolactin-Releasing Peptide | PrRP | human | CHO dhfr- | C1037 | DC1037 | MC1037 |
| Prostanoid | DP1 | human | HEK293T | C1200 | DC1200 | MC1200 |
| Prostanoid | DP2 | human | HEK293T | H1105 | DH1105 | MH1105 |
| Prostanoid | DP2 | human | HEK293T | H1105a | DH1105a | MH1105a |
| Prostanoid | EP1 | human | HEK293T | C1201a | DC1201a | MC1201a |
| Prostanoid | EP2 | human | HEK293T | C1202 | DC1202 | MC1202 |
| Prostanoid | EP2 | mouse | HEK293T | Cm1202 | DCm1202 | MCm1202 |
| Prostanoid | EP2 | mouse | HEK293T | Cm1202-3 | DCm1202-3 | MCm1202-3 |
| Prostanoid | EP2 | rat | HEK293T | Cr1202 | DCr1202 | MCr1202 |
| Prostanoid | EP2 | rat | HEK293T | Cr1202-134 | DCr1202-134 | MCr1202-134 |
| Prostanoid | EP3 | human | CHO-K1 | C1203-1 | DC1203-1 | MC1203-1 |
| Prostanoid | EP3 | human | CHO-K1 | C1203-1a | DC1203-1a | MC1203-1a |
| Prostanoid | EP3 | human | CHO-K1 | C1203-1b | DC1203-1b | MC1203-1b |
| Prostanoid | EP3 | human | CHO-K1 | C1203-1c | DC1203-1DC | MC1203-1MC |
| Prostanoid | EP3 | human | CHO-K1 | C1203-1d | DC1203-1d | MC1203-1d |
| Prostanoid | EP4 | human | HEK293T | C1204 | DC1204 | MC1204 |
| Prostanoid | FP | human | HEK293T | C1205 | DC1205 | MC1205 |
| Prostanoid | IP1 | human | CHO-K1 | C1206-1 | DC1206-1 | MC1206-1 |
| Prostanoid | TP | human | HEK293T | C1365 | DC1365 | MC1365 |
| Prostanoid | TP | human | HEK293T | H1365 | H1365 | H1365 |
| Protease-Activated | PAR1 | human | CHO-K1 | C1207-1 | DC1207-1 | MC1207-1 |
| Protease-Activated | PAR1 | human | HeLa | C1207-7 | DC1207-7 | MC1207-7 |
| Protease-Activated | PAR2 | human | HeLa | C1208-7 | DC1208-7 | MC1208-7 |
| Protease-Activated | PAR4 | human | HeLa | C1210-7 | DC1210-7 | MC1210-7 |
| Proton-Sensing Receptors | GPR4 | human | HEK293T | C1100 | DC1100 | MC1100 |
| Proton-Sensing Receptors | GPR4 | human | HEK293T | CA1100 | DCA1100 | MCA1100 |
| Proton-Sensing Receptors | GPR65 | human | HEK293T | C1121 | DC1121 | MC1121 |
| Proton-Sensing Receptors | GPR65 | human | HEK293T | CA1121 | DCA1121 | MCA1121 |
| Proton-Sensing Receptors | GPR65 | human | HEK293T | C1121a | DC1121a | MC1121a |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP20 | DC1121-CSP20 | MC1121-CSP20 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP23 | DC1121-CSP23 | MC1121-CSP23 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP30 | DC1121-CSP30 | MC1121-CSP30 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP36 | DC1121-CSP36 | MC1121-CSP36 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP38 | DC1121-CSP38 | MC1121-CSP38 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP44 | DC1121-CSP44 | MC1121-CSP44 |
| Proton-Sensing Receptors | GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP75 | DC1121-CSP75 | MC1121-CSP75 |
| Proton-Sensing Receptors | GPR68 | human | HEK293T | C1123 | DC1123 | MC1123 |
| Proton-Sensing Receptors | GPR68 | human | HEK293T | CA1123 | DCA1123 | MCA1123 |
| Proton-Sensing Receptors | GPR132 | human | HEK293T | CA1066 | DCA1066 | MCA1066 |
| Purinergic | GPR17 (long form) | human | 1321N1 | C1076-3 | DC1076-3 | MC1076-3 |
| Purinergic | GPR17 (long form) | human | 1321N1 | C1076-3a | DC1076-3a | MC1076-3a |
| Purinergic | GPR17 (short form) | human | 1321N1 | C1526-3 | DC1526-3 | MC1526-3 |
| Purinergic | GPR17 | mouse | 1321N1 | Cm1526-3 | DCm1526-3 | MCm1526-3 |
| Purinergic | GPR17 | rat | 1321N1 | Cr1526-3 | DCr1526-3 | MCr1526-3 |
| Purinergic | GPR17 | rat | 1321N1 | Cr1525-3 | DCr1525-3 | MCr1525-3 |
| Purinergic | P2Y1 | human | 1321N1 | C1160-3 | DC1160-3 | MC1160-3 |
| Purinergic | P2Y2 | human | 1321N1 | C1161-3 | DC1161-3 | MC1161-3 |
| Purinergic | P2Y2 | human | HEK293T | C1161 | DC1161 | MC1161 |
| Purinergic | P2Y2 | rat | 1321N1 | Cr1161-3 | DCr1161-3 | MCr1161-3 |
| Purinergic | P2Y4 | human | 1321N1 | C1162-3 | DC1162-3 | MC1162-3 |
| Purinergic | P2Y6 | human | 1321N1 | C1164-3 | DC1164-3 | MC1164-3 |
| Purinergic | P2Y11 | human | 1321N1 | C1169-3 | DC1169-3 | MC1169-3 |
| Purinergic | P2Y12 | human | 1321N1 | C1170-3 | DC1170-3 | MC1170-3 |
| Purinergic | P2Y12 | human | 1321N1 | C1170-3a | DC1170-3a | MC1170-3a |
| Purinergic | P2Y12 | rat | CHO dhfr- | C1170-1 | DC1170-1 | MC1170-1 |
| Purinergic | P2Y13 | human | 1321N1 | C1139-3 | DC1139-3 | MC1139-3 |
| Purinergic | P2Y14 | human | HEK293T | C1057 | DC1057 | MC1057 |
| Purinergic | P2Y14 | human | HEK293T Gαqi5 | CG1057 | DCG1057 | MCG1057 |
| Purinergic | P2Y14 | rat | HEK293T Gαqi5 | CGr1057 | DCGr1057 | MCGr1057 |
| Purinergic | P2Y14 | monkey | HEK293T Gαqi5 | CGp1057 | DCGp1057 | MCGp1057 |
| Relaxin | RXFP1 | human | HEK293T | C1287 | DC1287 | MC1287 |
| Relaxin | RXFP1 | human | HEK293T | C1287NTa | DC1287NTa | MC1287NTa |
| Relaxin | RXFP1 | human | HEK293T | C1287NTb | DC1287NTb | MC1287NTb |
| Relaxin | RXFP2 | human | HEK293T | C1289NTa | DC1289NTa | MC1289NTa |
| Relaxin | RXFP2 | human | HEK293T | C1289NTb | DC1289NTb | MC1289NTb |
| Relaxin | RXFP3 | human | HEK293T | C1306 | DC1306 | MC1306 |
| SARS-CoV-2 | ACE2 | human | HEK293T | C2006 | DC2006 | MC2006 |
| SARS-CoV-2 | TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 |
| Serotonin | 5-HT1A | human | HEK293T | C1319 | DC1319 | MC1319 |
| Serotonin | 5-HT1A | human | HEK293T | C1319a | DC1319a | MC1319a |
| Serotonin | 5-HT1B | human | HEK293T | C1320 | DC1320 | MC1320 |
| Serotonin | 5-HT1B | human | HEK293T | C1320a | DC1320a | MC1320a |
| Serotonin | 5-HT1B | human | HEK293T Gαqi5 | CG1320 | DCG1320 | MCG1320 |
| Serotonin | 5-HT2A | human | CHO-K1 | C1324-1 | DC1324-1 | MC1324-1 |
| Serotonin | 5-HT2A | mouse | HEK293T | Cm1324 | DCm1324 | MCm1324 |
| Serotonin | 5-HT2A | mouse | CHO-K1 | Cm1324-1 | DCm1324-1 | MCm1324-1 |
| Serotonin | 5-HT2A | dog | HEK293T | Cd1324 | DCd1324 | MCd1324 |
| Serotonin | 5-HT2B | human | CHO-K1 | C1325-1 | DC1325-1 | MC1325-1 |
| Serotonin | 5-HT2B | human | HEK293T | C1325 | DC1325 | MC1325 |
| Serotonin | 5-HT2B | mouse | HEK293T | Cm1325 | DCm1325 | MCm1325 |
| Serotonin | 5-HT2C | human | CHO-K1 | C1326-1 | DC1326-1 | MC1326-1 |
| Serotonin | 5-HT4A | human | CHO-K1 | C1518-1 | DC1518-1 | MC1518-1 |
| Serotonin | 5-HT4A | mouse | CHO-K1 | Cm1518-1 | DCm1518-1 | MCm1518-1 |
| Serotonin | 5-HT4B | human | CHO-K1 | C1330-1 | DC1330-1 | MC1330-1 |
| Serotonin | 5-HT4B | human | HEK293T | C1330 | DC1330 | MC1330 |
| Serotonin | 5-HT4D | human | CHO-K1 | C1520-1 | DC1520-1 | MC1520-1 |
| Serotonin | 5-HT6 | human | CHO-K1 | C1331-1 | DC1331-1 | MC1331-1 |
| Serotonin | 5-HT7 | human | HEK293T | C1334 | DC1334 | MC1334 |
| Somatostatin | sst1 | human | CHO-K1 | C1345-1a | DC1345-1a | MC1345-1a |
| Somatostatin | sst1 | human | CHO-K1 Gα16 | CG1345-1 | DCG1345-1 | MCG1345-1 |
| Somatostatin | sst2 | human | CHO-K1 | C1346-1 | DC1346-1 | MC1346-1 |
| Somatostatin | sst2 | human | CHO-K1 Gα16 | CG1346-1 | DCG1346-1 | MCG1346-1 |
| Somatostatin | sst3 | human | CHO-K1 | C1347-1 | DC1347-1 | MC1347-1 |
| Somatostatin | sst3 | human | CHO-K1 Gα16 | CG1347-1 | DCG1347-1 | MCG1347-1 |
| Somatostatin | sst4 | human | CHO-K1 | C1348-1a | DC1348-1a | MC1348-1a |
| Somatostatin | sst4 | human | CHO-K1 Gα16 | CG1348-1 | DCG1348-1 | MCG1348-1 |
| Somatostatin | sst5 | human | CHO-K1 | C1349-1 | DC1349-1 | MC1349-1 |
| Somatostatin | sst5 | human | CHO-K1 Gα16 | CG1349-1 | DCG1349-1 | MCG1349-1 |
| Tachykinin | NK1 | human | HEK293T | C1303 | DC1303 | MC1303 |
| Tachykinin | NK2 | human | HEK293T | C1304 | DC1304 | MC1304 |
| Tachykinin | NK3 | human | HEK293T | C1305 | DC1305 | MC1305 |
| Tachykinin | NK3 | rat | HEK293T | Cr1305 | DCr1305 | MCr1305 |
| Tachykinin | NK3 | mouse | HEK293T | Cm1305 | DCm1305 | MCm1305 |
| Thyrotropin-Releasing Hormone | TRH | human | HEK293T | |||
| Trace Amine | TA1 | rat | HEK293T | C1357 | DC1357 | MC1357 |
| Trace Amine | TA1 | human | HEK293T | C1357a | DC1357a | MC1357a |
| Trace Amine | TA1 | rat | HEK293T Gαqi5 | Cr1357 | DCr1357 | MCr1357 |
| Urotensin | UT | rat | CHO dhfr- | C1035-1 | DC1035-1 | MC1035-1 |
| Urotensin | UT | human | CHO-K1 | C1035-1a | DC1035-1a | MC1035-1a |
| Vasoactive Intestinal Peptide | PAC1 | human | HEK293T | C1415 | DC1415 | MC1415 |
| Vasoactive Intestinal Peptide | VPAC1 | human | CHO-K1 | C1292-1 | DC1292-1 | MC1292-1 |
| Vasoactive Intestinal Peptide | VPAC2 | human | HEK293T | H1293 | DH1293 | MH1293 |
| Vasopressin/Oxytocin | OT | human | CHO-K1 | C1299-1 | DC1299-1 | MC1299-1 |
| Vasopressin/Oxytocin | OT | rabbit | HEK293T | Cb1299 | DCb1299 | MCb1299 |
| Vasopressin/Oxytocin | OT | rabbit | HEK293T | Cb1299L | DCb1299L | MCb1299L |
| Vasopressin/Oxytocin | V1A | human | CHO-K1 | C1042-1 | DC1042-1 | MC1042-1 |
| Vasopressin/Oxytocin | V1A | rabbit | HEK293T | Cb1042 | DCb1042 | MCb1042 |
| Vasopressin/Oxytocin | V1B | human | CHO-K1 | C1043-1 | DC1043-1 | MC1043-1 |
| Vasopressin/Oxytocin | V1B | rabbit | HEK293T | Cb1043 | DCb1043 | MCb1043 |
| Vasopressin/Oxytocin | V1B | rabbit | HEK293T | Cb1043L | DCb1043L | MCb1043L |
| Vasopressin/Oxytocin | V2 | human | CHO-K1 | C1044-1 | DC1044-1 | MC1044-1 |
| Vasopressin/Oxytocin | V2 | rabbit | HEK293T | Cb1044 | DCb1044 | MCb1044 |
| Vasopressin/Oxytocin | V2 | rabbit | HEK293T | Cb1044L | DCb1044L | MCb1044L |
| Vasopressin/Oxytocin | V2 | dog | CHO-K1 | Cd1044-1 | DCd1044-1 | MCd1044-1 |
| Zinc | GPR39 | human | HEK293T | H1099 | DH1099 | MH1099 |
Endogenous Targets
| Target Family | Target | Species | Cells |
|---|---|---|---|
| Kinase | AMPK | human | C2C12 |
| DNA-PK | human | Hela | |
| Aryl Hydrocarbon Receptor (Nuclear Hormone Receptor) | AHR | human | Hep G2 |
| AHR | mouse | Hepa1-6 | |
| AHR | human | HG2L6.1c1 CALUX | |
| AHR | mouse | H1L6.c3 CALUX | |
| Chemokine | CCR4 | human | H9 |
| CCR6 | human | H9 | |
| Calcitonin | CGRP | human | SK-N-MC |
| Free Fatty Acid | GPR40 | mouse | MIN6 |
| Lysophospholipid | LPA | human | Human Fibroblast-Like Synoviocytes-Rheumatoid |
| Melanin-Concentrating Hormone | MCH1 | human | YS35 |
| Opioid | mu | human | SK-N-SH |
| Serotonin | 5-HT | human | Human Heart Valvular Interstitial Cells |
Other Targets
| Receptor Family | Target | Species | Parental | Stable Cell Line | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Integrin | a V b 1 | human | CHOB2 | C3001 | DC3001 | MC3001 |
| Potassium Channel | TMEM175 | human | HEK293T | C1527 | DC1527 | MC1527 |
| TMEM175 | human | HEK293T | C1527a | DC1527a | MC1527a | |
| Receptor Tyrosine Kinases | TrKA | human | CHO-K1 | CK1001-1 | DCK1001-1 | MCK1001-1 |
| TrKA | human | CHO-K1 | CK1001-1b | DCK1001-1b | MCK1001-1b | |
| TrKA | rat | CHO-K1 | CKr1001-1 | DCKr1001-1 | MCKr1001-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1 | DCK1002-1 | MCK1002-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1a | DCK1002-1a | MCK1002-1a | |
| SARS-CoV-2 | TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 |
| Zinc Transporter | ZnT3 | human | Hela | C2001-7 | DC2001-7 | MC2001-7 |
| ZnT8 | human | CHO-K1 | C2002-1 | DC2002-1 | MC2002-1 |
Parental Lines
| Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|
| HEK293T | DC0001 | MC0001 | |
| HEK293T Gαqi5 | CG0001 | DCG0001 | MCG0001 |
| CHO-K1 | DC0001-1 | MC0001-1 | |
| CHO-K1 Gαqi5 | CG0001-1 | DCG0001-1 | MCG0001-1 |
| CHO-K1 Gα16 | CG0002-1 | DCG0002-1 | MCG0002-1 |
| CHO-K1 Gα16 Gαqi5 | CG0003-1 | DCG0003-1 | MCG0003-1 |
| CHO dhfr- | DCD0001-1 | MCD0001-1 | |
| CHO-K1 NFAT | CK0001-1 | DCK0001-1 | MCK0001-1 |
| 1321N1 | DC0001-3 | MC0001-3 | |
| RH7777 | DC0001-6 | MC0001-6 | |
| Hela | DC0001-7 | MC0001-7 |
Assay Kits
| Assay Kit | Unit Size (384-well) | Catalog | Description | Data |
|---|---|---|---|---|
| MultiScreen™ β-Arrestin Assay Kit | 1 plate 96- well/384-well | MSBAK01-1 | The kits contain the substrate for Multiscreen™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Validated by Multiscreen™ stable cell lines co-expressing target GPCRs and Multiscreen™ β-Arrestin sensors. Suitable for any cell line or primary cells co-expressing endogenous or untagged GPCR target and Multiscreen™ β-Arrestin sensor. |  β-Arrestin Recruitment Dose Response in MultiScreen™ MOR β-Arrestin2 CHO-K1 stable cell line (CA1350-1a) measured with MultiScreen™ β-Arrestin Assay Kit. Cells were seeded in assay buffer in a 384-well plate, incubated with the MultiScreen™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | MSBAK01-10 | |||
| 100 plates 96-well/384-well | MSBAK01-100 | |||
| MultiScreen™ β-Arrestin BacMam Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKBM01-1 Or β-Arrestin2 MSBAKBM02-1 | The kits contain BacMam viral particles of Multiscreen™ β-Arrestin sensor cDNA, control GFP BacMam viral particle, the substrate for Multiscreen™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. |  β-Arrestin Recruitment Dose Response in MultiScreen™ MOR CHO-K1 stable cell line (C1350-1a) infected with β-Arrestin sensor BacMam virus for 48 hours before being measured with MultiScreen™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MultiScreen™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-10 Or β-Arrestin2 MSBAKBM02-10 |
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| 100 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-100 Or β-Arrestin2 MSBAKBM02-100 |
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| MultiScreen™ β-Arrestin HSV Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKHSV01-1 Or β-Arrestin2 MSBAKHSV02-1 | The kits contain HSV viral particles of Multiscreen™ β-Arrestin sensor cDNA, control GFP HSV viral particle, the substrate for Multiscreen™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. |  β-Arrestin Recruitment Dose Response in MultiScreen™ KOR HEK293T stable cell line (C1352) infected with β-Arrestin HSV sensor for 48 hours before being measured with MultiScreen™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MultiScreen™ Substrate before being treated with control agonist Dynorphin B and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-10 Or β-Arrestin2 MSBAKHSV02-10 |
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| 100 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-100 Or β-Arrestin2 MSBAKHSV02-100 |
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| MultiScreen™ Calcium 1.0 No Wash Assay Kit | 1000 tests | MSCA01-1 | Multiscreen™ Calcium 1.0 No Wash Assay Kits provide homogeneous fluorescence-based assays for intracellular calcium mobilization detection in 96-well, 384-well and higher multiplexity. Pre-loaded with Calcium 1.0 is taken up by the cells where the lipophilic blocking groups of Calcium 1.0 are cleaved by esterases, resulting in a negatively charged fluorescent dye that stays inside cells. The fluorescence signal is greatly enhanced after binding to intracellular calcium released by cell-stimulation. Long wavelength, high sensitivity, and >100 times fluorescence enhancement make Calcium 1.0 an ideal indicator for intracellular calcium release assays measuring GPCRs, calcium channels and receptor tyrosine kinase signaling. Multiscreen™ Calcium 1.0 No Wash Assay Kits are validated by Multiscreen™ stable cell lines. |  Calcium Dose Response in MultiScreen™ A2B-HEK293T stable cell line (C1429) measured with MultiScreen™ Calcium 1.0 No Wash Assay Kit. Cells were seeded in assay buffer in a 384-well black wall clear bottom PDL-coated plate, incubated with the MultiScreen™ Calcium 1.0 No Wash Assay Kit before being treated with control agonist NECA and measured by FLIPR. |
| 10000 tests | MSCA01-10 | |||
| 100000 tests | MSCA01-100 | |||
| MultiScreen™ TR-FRET cAMP 1.0 No Wash Assay Kit | 500 tests | MSCM01-1 | Multiscreen™ TR-FRET cAMP 1.0 No Wash Assay Kits provide a homogenous TR-FRET assay method for adenylyl cyclase activity detection in 96-well, 384-well and higher multiplexity. α-cAMP antibody (Ab) is labeled with MultiScreen™Eu while cAMP is labeled with MultiScreen™650. In the absence of cAMP, MultiScreen™650-cAMP is bound to MultiScreen™Eu-α-cAMP-Ab to give a strong TR-FRET Emission at 655 nm. Free cAMP in the test sample competes for binding to the MultiScreen™ Eu-α-cAMP-Ab, reducing TR-FRET signal from MultiScreen™650-cAMP binding. The MultiScreen™650-cAMP only has fluorescence lifetime of nanosecond while MultiScreen™Eu-α-cAMP-Ab has much longer fluorescence lifetime value due to TR-FRET. The magnitude of TR-FRET is proportional to the concentration of cAMP in a sample. Multiscreen™ TR-FRET cAMP 1.0 No Wash Assay Kits are validated by Multiscreen™ stable cell lines. |  cAMP Dose-Response in MultiScreen™ β1-HEK293T stable cell line (C1437-1) measured with MultiScreen™ TR-FRET cAMP 1.0 No Wash Assay Kit. Cells were seeded in a 384-well solid white plate, incubated with Isoproterenol and 1mM IBMX before being treated with MultiScreen™Eu-α-cAMP-Ab and MultiScreen™650-cAMP, and measured by FlexStation 3. |
| 5000 tests | MSCM01-5 | |||
| 25000 tests | MSCM01-25 |