| Receptor Family | Receptor | Species | Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Adenosine | A1 | human | HEK293T | C1427B | DC1427B | MC1427B |
| A1 | human | CHO-K1 | C1427-1 | DC1427-1 | MC1427-1 | |
| A1 | rat | HEK293T | Cr1427 | DCr1427 | MCr1427 | |
| A2A | human | HEK293T | C1428 | DC1428 | MC1428 | |
| A2A | human | CHO-K1 | C1428-1 | DC1428-1 | MC1428-1 | |
| A2A | mouse | HEK293T | Cm1428A | DCm1428A | MCm1428A | |
| A2A | mouse | HEK293T | Cm1428B | DCm1428B | MCm1428B | |
| A2A | mouse | CHO-K1 | Cm1428-1 | DCm1428-1 | MCm1428-1 | |
| A2A | rat | HEK293T | Cr1428 | DCr1428 | MCr1428 | |
| A2B | human | HEK293T | C1429 | DC1429 | MC1429 | |
| A2B | human | CHO-K1 | C1429-1 | DC1429-1 | MC1429-1 | |
| A2B | human | HEK293T | C1429a | DC1429a | MC1429a | |
| A2B | rat | HEK293T | Cr1429 | DCr1429 | MCr1429 | |
| A3 | human | HEK293T | C1430 | DC1430 | MC1430 | |
| A3 | human | CHO-K1 | C1430-1 | DC1430-1 | MC1430-1 | |
| A3 | rat | HEK293T | Cr1430 | DCr1430 | MCr1430 | |
| Adhesion Class GPCRs | GPR97 | human | HEK293T | C1396 | DC1396 | MC1396 |
| GPR110 | human | HEK293T | C1378 | DC1378 | MC1378 | |
| Adrenergic | alpha1A | human | CHO-K1 | C1431-1 | DC1431-1 | MC1431-1 |
| alpha1B | human | CHO-K1 | C1432-1 | DC1432-1 | MC1432-1 | |
| alpha1D | human | CHO-K1 | C1433-1 | DC1433-1 | MC1433-1 | |
| alpha2A | human | CHO-K1 | C1434-1 | DC1434-1 | MC1434-1 | |
| alpha2A | human | CHO-K1 | C1434-1a | DC1434-1a | MC1434-1a | |
| alpha2A | human | CHO-K1 Gqi5 | CG1434-1 | DCG1434-1 | MCG1434-1 | |
| alpha2B | human | CHO-K1 | C1435-1 | DC1435-1 | MC1435-1 | |
| alpha2B | human | CHO-K1 Gqi5 | CG1435-1 | DCG1435-1 | MCG1435-1 | |
| alpha2C | human | CHO-K1 | C1436-1 | DC1436-1 | MC1436-1 | |
| alpha2C | human | CHO-K1 Gqi5 | CG1436-1 | DCG1436-1 | MCG1436-1 | |
| beta1 | human | HEK293T | H1437 | H1437 | H1437 | |
| beta1 | human | CHO-K1 | C1437-1 | DC1437-1 | MC1437-1 | |
| beta2 | human | CHO-K1 | C1438-1a | DC1438-1a | MC1438-1a | |
| beta2 | human | HEK293T β-Arrestin1 | CA1438BA1 | DCA1438BA1 | MCA1438BA1 | |
| beta2 | human | HEK293T β-Arrestin2 | CA1438BA2 | DCA1438BA2 | MCA1438BA2 | |
| beta3 | human | HEK293T | C1439a | DC1439a | MC1439a | |
| Anaphylatoxin | C3AR1 | human | HEK293T | C1222 | DC1222 | MC1222 |
| C5R1 | human | HEK293T | C1221 | DC1221 | MC1221 | |
| Angiotensin | AT1 | mouse | CHO-K1 | Cm1417-1 | DCm1417-1 | MCm1417-1 |
| AT1 | mouse | CHO-K1 | Cm1417-1a | DCm1417-1a | MCm1417-1a | |
| AT1 | human | HEK293T | H1417 | DH1417 | MH1417 | |
| AT1 | human | HEK293T | HA1417- BA1 | DHA1417- BA1 | MHA1417- BA1 | |
| AT1 | human | HEK293T | HA1417-BA2 | DHA1417-BA2 | MHA1417-BA2 | |
| Apelin | APJ | human | HEK293T | C1196a | DC1196a | MC1196a |
| APJ | human | CHO-K1 | C1196-1 | DC1196-1 | MC1196-1 | |
| APJ | human | HEK293T Gαqi5 | CG1196a | DCG1196a | MCG1196a | |
| Bile Acid | GPBA | human | CHO-K1 | C1361-1 | DC1361-1 | MC1361-1 |
| GPBA | human | CHO-K1 | C1361-1a | DC1361-1a | MC1361-1a | |
| GPBA | rat | CHO-K1 | Cr1361-1 | DCr1361-1 | MCr1361-1 | |
| GPBA | mouse | CHO-K1 | Cm1361-1 | DCm1361-1 | MCm1361-1 | |
| GPBA Mutant W83G | human | CHO-K1 | C1361-1MT1 | DC1361-1MT1 | MC1361-1MT1 | |
| GPBA Mutant W83A | human | CHO-K1 | C1361-1MT2 | DC1361-1MT2 | MC1361-1MT2 | |
| GPBA Mutant V88L | human | CHO-K1 | C1361-1MT3 | DC1361-1MT3 | MC1361-1MT3 | |
| GPBA Mutant Y89A | human | CHO-K1 | C1361-1MT4 | DC1361-1MT4 | MC1361-1MT4 | |
| GPBA Mutant Y89H | human | CHO-K1 | C1361-1MT5 | DC1361-1MT5 | MC1361-1MT5 | |
| GPBA Mutant F96A | human | CHO-K1 | C1361-1MT6 | DC1361-1MT6 | MC1361-1MT6 | |
| GPBA Mutant W237A | human | CHO-K1 | C1361-1MT7 | DC1361-1MT7 | MC1361-1MT7 | |
| GPBA Mutant W240A | human | CHO-K1 | C1361-1MT8 | DC1361-1MT8 | MC1361-1MT8 | |
| Bombesin | BB1 | human | HEK293T | C1211 | DC1211 | MC1211 |
| BB1 | rat | C6 | C1211-1 | DC1211-1 | MC1211-1 | |
| BB2 | human | HEK293T | C1215 | DC1215 | MC1215 | |
| BB3 | human | HEK293T | C1214 | DC1214 | MC1214 | |
| BB3 | human | HEK293T | H1214 | DH1214 | MH1214 | |
| Bradykinin | B1 | human | HEK293T | C1198a | DC1198a | MC1198a |
| B1 | mouse | HEK293T | Cm1198 | DCm1198 | MCm1198 | |
| B2 | human | HEK293T | H1199 | DH1199 | MH1199 | |
| B2 | mouse | HEK293T | Cm1199 | DCm1199 | MCm1199 | |
| B2 | rat | HEK293T | Cr1199 | DCr1199 | MCr1199 | |
| B2 | dog | HEK293T | cd1199 | DCd1199 | MCd1199 | |
| B2 | rhesus monkey | HEK293T | Cpr1199 | DCpr1199 | MCpr1199 | |
| B2 | guinea pig | HEK293T | Cc1199 | DCc1199 | MCc1199 | |
| B2 | rabbit | HEK293T | Cb1199 | DCb1199 | MCb1199 | |
| Calcitonin | CALCRL | human | HEK293T | C1232 | DC1232 | MC1232 |
| CALCRL | human | CHO-K1 | C1232-1 | DC1232-1 | MC1232-1 | |
| CGRP | human | CHO-K1 | C1515-1 | DC1515-1 | MC1515-1 | |
| AM1 | human | CHO-K1 | C1516-1 | DC1516-1 | MC1516-1 | |
| AM2 | human | CHO-K1 | C1517-1 | DC1517-1 | MC1517-1 | |
| CT | human | HEK293T | H1231 | DH1231 | MH1231 | |
| CT | human | CHO-K1 | C1231-1A | DC1231-1A | MC1231-1A | |
| CT | human | CHO-K1 | C1231-1B | DC1231-1B | MC1231-1B | |
| AMY1 | human | CHO-K1 | C1509-1a | DC1509-1a | MC1509-1a | |
| AMY2 | human | CHO-K1 | C1510-1a | DC1510-1a | MC1510-1a | |
| AMY2 | human | CHO-K1 | C1510-1b | DC1510-1b | MC1510-1b | |
| AMY3 | human | CHO-K1 | C1511-1a | DC1511-1a | MC1511-1a | |
| Calcium-Sensing | CaSR | human | HEK293T | C1233 | DC1233 | MC1233 |
| CaSR | rat | HEK293T | Hr1233 | DHr1233 | MHr1233 | |
| Cannabinoid | CB1 | human | HEK293T | C1229 | DC1229 | MC1229 |
| CB1 | human | CHO-K1 | C1229-1a | DC1229-1a | MC1229-1a | |
| CB1 | human | CHO-K1 | C1229-1 | DC1229-1 | MC1229-1 | |
| CB1a | human | CHO-K1 | C1512-1 | DC1512-1 | MC1512-1 | |
| CB1b | human | CHO-K1 | C1513-1 | DC1513-1 | MC1513-1 | |
| CB1 | mouse | CHO-K1 | Cm1229-1A | DCm1229-1A | MCm1229-1A | |
| CB1 | mouse | CHO-K1 | Cm1229-1B | DCm1229-1B | MCm1229-1B | |
| CB1 | dog | HEK293T | Cd1229 | DCd1229 | MCd1229 | |
| CB1 | dog | HEK293T | Cd1229a | DCd1229a | MCd1229a | |
| CB1 | dog | HEK293T | Cd1229b | DCd1229b | MCd1229b | |
| CB1 MUTANT B | human | CHO-K1 β-Arrestin2 | CA1513BA2-1 | DCA1513BA2-1 | MCA1513BA2-1 | |
| CB2 | human | CHO-K1 | C1230-1 | DC1230-1 | MC1230-1 | |
| CB2 | human | CHO-K1 | C1230-1a | DC1230-1a | MC1230-1a | |
| CB2 | human | CHO-K1 β-Arrestin2 | CA1230BA2-1 | DCA1230BA2-1 | MCA1230BA2-1 | |
| CB2 | rat | CHO-K1 | Cr1230-1 | DCr1230-1 | MCr1230-1 | |
| CB2 | rat | CHO-K1 | Cr1230-1a | DCr1230-1a | MCr1230-1a | |
| CB2 | mouse | CHO-K1 β-Arrestin2 | CAm1230BA2-1 | DCAm1230BA2-1 | MCAm1230BA2-1 | |
| CB2 | mouse | CHO-K1 | Cm1230-1 | DCm1230-1 | MCm1230-1 | |
| CB2 | mouse | CHO-K1 | Cm1230-1a | DCm1230-1a | MCm1230-1a | |
| CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1 | DCAr1230BA2-1 | MCAr1230BA2-1 | |
| CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1a | DCAr1230BA2-1a | MCAr1230BA2-1a | |
| GPR55 | human | HEK293T | H1113 | H1113 | H1113 | |
| GPR55 | human | HEK293T | C1113b | DC1113b | MC1113b | |
| GPR55 | human | HEK293T | C1113d | DC1113d | MC1113d | |
| Chemokine | CCR1 | human | HEK293T | C1009 | DC1009 | MC1009 |
| CCR1 | human | HEK293T Gαqi5 | CG1009 | DCG1009 | MCG1009 | |
| CCR2 | human | HEK293T | C1010 | DC1010 | MC1010 | |
| CCR3 | human | HEK293T | C1011 | DC1011 | MC1011 | |
| CCR3 | human | HEK293T Gαqi5 | CG1011 | DCG1011 | MCG1011 | |
| CCR4 | human | HEK293T | C1012 | DC1012 | MC1012 | |
| CCR4 | human | HEK293T Gαqi5 | CG1012 | DCG1012 | MCG1012 | |
| CCR5 | human | HEK293T | C1013a | DC1013a | MC1013a | |
| CCR5 | human | HEK293T | C1013b | DC1013b | MC1013b | |
| CCR5 | human | HEK293T Gαqi5 | CG1013 | DCG1013 | MCG1013 | |
| CCR6 | human | HEK293T | C1014a | DC1014a | MC1014a | |
| CCR6 | human | HEK293T | C1014b | DC1014b | MC1014b | |
| CCR6 | mouse | HEK293T | Cm1014 | DCm1014 | MCm1014 | |
| CCR7 | human | HEK293T | C1015 | DC1015 | MC1015 | |
| CCR7 | human | HEK293T Gαqi5 | CG1015 | DCG1015 | MCG1015 | |
| CCR8 | human | HEK293T | C1016 | DC1016 | MC1016 | |
| CCR8 | human | HEK293T | C1016a | DC1016a | MC1016a | |
| CCR8 | human | HEK293T Gαqi5 | CG1016 | DCG1016 | MCG1016 | |
| CCR9 | dog | HEK293T Gαqi5 | CGd1017 | DCGd1017 | MCGd1017 | |
| CCR9 | human | HEK293T | C1017 | DC1017 | MC1017 | |
| CCR9 | human | HEK293T | C1017a | DC1017a | MC1017a | |
| CCR9 | human | HEK293T Gαqi5 | CG1017 | DCG1017 | MCG1017 | |
| CCR9 | human | HEK293T Gαqi5 | CG1017A | DCG1017A | MCG1017A | |
| CCR9 | mouse | HEK293T | Cm1017 | DCm1017 | MCm1017 | |
| CCR9 | mouse | HEK293T Gαqi5 | CGm1017 | DCGm1017 | MCGm1017 | |
| CCR9 | rat | HEK293T Gαqi5 | CGr1017 | DCGr1017 | MCGr1017 | |
| CCR10 | human | HEK293T | C1018 | DC1018 | MC1018 | |
| CCR10 | human | CHO-K1 Gαqi5 | CG1018-1 | DCG1018-1 | MCG1018-1 | |
| CMKLR1 | human | HEK293T | C1147 | DC1147 | MC1147 | |
| CMKLR1 | human | HEK293T Gαqi5 | CG1147 | DCG1147 | MCG1147 | |
| CX3CR1 | human | HEK293T | C1008 | DC1008 | MC1008 | |
| CX3CR1 | human | HEK293T Gαqi5 | CG1008a | DCG1008a | MCG1008a | |
| CX3CR1 | human | HEK293T Gαqi5 | CG1008b | DCG1008b | MCG1008b | |
| CXCR1 | human | HEK293T | C1001a | DC1001a | MC1001a | |
| CXCR1 | human | HEK293T Gαqi5 | CG1001 | DCG1001 | MCG1001 | |
| CXCR2 | human | HEK293T | C1002 | DC1002 | MC1002 | |
| CXCR2 | human | HEK293T Gαqi5 | CG1002 | DCG1002 | MCG1002 | |
| CXCR3 | human | HEK293T | C1003 | DC1003 | MC1003 | |
| CXCR3 | human | HEK293T | C1003a | DC1003a | MC1003a | |
| CXCR3 | human | HEK293T Gαqi5 | CG1003 | DCG1003 | MCG1003 | |
| CXCR4 | human | HEK293T | C1004-1 | DC1004-1 | MC1004-1 | |
| CXCR4 | human | HEK293T Gαqi5 | CG1004 | DCG1004 | MCG1004 | |
| CXCR5 | human | HEK293T | C1005 | DC1005 | MC1005 | |
| CXCR5 | human | HEK293T | C1005a | DC1005a | MC1005a | |
| CXCR5 | human | CHO-K1 | C1005-1 | DC1005-1 | MC1005-1 | |
| CXCR5 | human | CHO-K1 | C1005-1a | DC1005-1a | MC1005-1a | |
| CXCR6 | human | HEK293T | C1006 | DC1006 | MC1006 | |
| CXCR6 | human | CHO-K1 | C1006-1 | DC1006-1 | MC1006-1 | |
| CXCR6 | human | HEK293T Gαqi5 | CG1006 | DCG1006 | MCG1006 | |
| CXCR7 | human | HEK293T | C1150 | DC1150 | MC1150 | |
| CXCR7 | human | HEK293T | CA1150BA2a | DCA1150BA2a | MCA1150BA2a | |
| XCR1 | human | HEK293T | C1007 | DC1007 | MC1007 | |
| XCR1 | human | HEK293T Gαqi5 | CG1007 | DCG1007 | MCG1007 | |
| Cholecystokinin | CCK1 | human | CHO-K1 | C1038-1a | DC1038-1a | MC1038-1a |
| CCK1 | human | HEK293T | C1038 | DC1038 | MC1038 | |
| CCK2 | human | HEK293T | H1039 | DH1039 | MH1039 | |
| Citric Acid Cycle Intermediates | GPR91 | human | CHO-K1 | C1144-1 | DC1144-1 | MC1144-1 |
| GPR91 | mouse | CHO-K1 | Cm1144-1 | DCm1144-1 | MCm1144-1 | |
| GPR91 | rat | CHO-K1 | Cr1144-1 | DCr1144-1 | MCr1144-1 | |
| GPR91 | human | CHO-K1 B-Arrestin2 | CA1141BA2-1 | DCA1141BA2-1 | MCA1141BA2-1 | |
| GPR91 | human | CHO-K1 B-Arrestin2 | CA1144BA2-1 | DCA1144BA2-1 | MCA1144BA2-1 | |
| GPR99 | human | CHO-K1 | C1132-1 | DC1132-1 | MC1132-1 | |
| Corticotrophin-Releasing Factor | CRF1 | human | HEK293T | C1040 | DC1040 | MC1040 |
| CRF1 | human | HEK293T Gαqi5 | CG1040 | DCG1040 | MCG1040 | |
| CRF2 | human | HEK293T | C1041 | DC1041 | MC1041 | |
| CRF2 | human | HEK293TGα16 | CG1041 | DCG1041 | MCG1041 | |
| Dopamine | D1 | human | HEK293T | C1335 | DC1335 | MC1335 |
| D1 | human | HEK293T | H1335 | DH1335 | MH1335 | |
| D2 | human | HEK293T | C1336 | DC1336 | MC1336 | |
| D2 | human | HEK293T | C1336a | DC1336a | MC1336a | |
| D2 | human | HEK293T | C1336b | DC1336b | MC1336b | |
| D2 Ghrelin | human | HEK293T | C1514 | DC1514 | MC1514 | |
| D3 | human | HEK293T Gqi5 | CG1337 | DCG1337 | MCG1337 | |
| D4 | human | HEK293T | C1338 | DC1338 | MC1338 | |
| D4 | human | HEK293T Gαqi5 | CG1338 | DCG1338 | MCG1338 | |
| D5 | human | HEK293T | C1339 | DC1339 | MC1339 | |
| Endothelin | ETA | human | CHO-K1 | C1216-1 | DC1216-1 | MC1216-1 |
| ETA | rat | CHO-K1 | Cr1216-1 | DCr1216-1 | MCr1216-1 | |
| ETB | human | CHO-K1 | C1217-1 | DC1217-1 | MC1217-1 | |
| Free Fatty Acid | GPR119 | human | CHO-K1 | C1298-1a | DC1298-1a | MC1298-1a |
| GPR119 | human | HEK293T | C1298 | DC1298 | MC1298 | |
| GPR119 | mouse | CHO-K1 | Cm1298-1 | DCm1298-1 | MCm1298-1 | |
| GPR120 | human | HEK293T | C1294 | DC1294 | MC1294 | |
| GPR120 | human | HEK293T Gαqi5 | CG1294 | DCG1294 | MCG1294 | |
| GPR120 | human | CHO-K1 | C1294-1 | DC1294-1 | MC1294-1 | |
| GPR120L | human | HEK293T | C1522 | DC1522 | MC1522 | |
| GPR120L | human | HEK293T β-Arrestin2 | CA1522 | DCA1522 | MCA1522 | |
| GPR120 | mouse | HEK293T Gαqi5 | CGm1294 | DCGm1294 | MCGm1294 | |
| GPR120 | rat | HEK293T | Cr1294 | DCr1294 | MCr1294 | |
| GPR40 | cynomolgus monkey | CHO-K1 | Cpc1101-1 | DCpc1101-1 | MCpc1101-1 | |
| GPR40 | cynomolgus monkey | CHO-K1 | CApr1101-1 | DCApr1101-1 | MCApr1101-1 | |
| GPR40 | cynomolgus monkey | CHO-K1 β-Arrestin2 | CApc1101-1 | DCApc1101-1 | MCApc1101-1 | |
| GPR40 | dog | CHO-K1 | Cd1101-1 | DCd1101-1 | MCd1101-1 | |
| GPR40 | human | HEK293T | C1101 | DC1101 | MC1101 | |
| GPR40 | human | CHO-K1 | C1101-1 | DC1101-1 | MC1101-1 | |
| GPR40 | human | CHO-K1 | C1101-1A | DC1101-1A | MC1101-1A | |
| GPR40 | human | CHO-K1 β-Arrestin2 | CA1101-1 | DCA1101-1 | MCA1101-1 | |
| GPR40 | mouse | HEK293T | Cm1101 | DCm1101 | MCm1101 | |
| GPR40 | rat | HEK293T | Cr1101 | DCr1101 | MCr1101 | |
| GPR40 | rat | CHO-K1 | Cr1101-1 | DCr1101-1 | MCr1101-1 | |
| GPR40 | rhesus monkey | CHO-K1 | Cpr1101-1 | DCpr1101-1 | MCpr1101-1 | |
| GPR40 | rat | CHO-K1 β-Arrestin2 | CAr1101-1 | DCAr1101-1 | MCAr1101-1 | |
| GPR41 | human | HEK293T | C1102 | DC1102 | MC1102 | |
| GPR41 | human | CHO-K1 Gα16 | C1102-1 | DCG1102-1 | MC1102-1 | |
| GPR41 | human | HEK293T Gαqi5 | CG1102 | DCG1102 | MCG1102 | |
| GPR41 | mouse | CHO-K1 Gα16 | CGm1102-1 | DCGm1102-1 | MCGm1102-1 | |
| GPR41 | rat | HEK293T | Cr1102 | DCr1102 | MCr1102 | |
| GPR43 | human | HEK293T | C1104 | DC1104 | MC1104 | |
| GPR43 | human | CHO-K1 | C1104-1 | DC1104-1 | MC1104-1 | |
| GPR43 | human | CHO-K1 Gα16 | HG1104-1 | DHG1104-1 | MHG1104-1 | |
| GPR43 | mouse | HEK293T | Cm1104 | DCm1104 | MCm1104 | |
| GPR43 | rat | HEK293T | Cr1104 | DCr1104 | MCr1104 | |
| GPR43 | dog | CHO-K1 | Cd1104-1A | DCd1104-1A | MCd1104-1A | |
| GPR43 | dog | CHO-K1 | Cd1104-1B | DCd1104-1B | MCd1104-1B | |
| GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1A | DCpc1104-1A | MCpc1104-1A | |
| GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1B | DCpc1104-1B | MCpc1104-1B | |
| GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1A | DCpr1104-1A | MCpr1104-1A | |
| GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1B | DCpr1104-1B | MCpr1104-1B | |
| GPR84 | human | CHO-K1 | C1137-1 | DC1137-1 | MC1137-1 | |
| GPR84 | human | CHO-K1 Gαqi5 | CG1137-1 | DCG1137-1 | MCG1137-1 | |
| Frizzled | SMO | human | HEK293T | C1442 | DC1442 | MC1442 |
| SMO | human | HEK293T | H1442 | DH1442 | MH1442 | |
| Galanin | GAL1 | human | CHO-K1 Gαqi5 | CG1178-1 | DCG1178-1 | MCG1178-1 |
| GAL1 | human | HEK293T | C1178 | DC1178 | MC1178 | |
| GAL2 | human | CHO-K1 | C1179-1 | DC1179-1 | MC1179-1 | |
| Ghrelin | Ghrelin | human | HEK293T | C1197b | DC1197b | MC1197b |
| Ghrelin | human | CHO-K1 | C1197-1 | DC1197-1 | MC1197-1 | |
| Ghrelin | mouse | HEK293T | Cm1197 | DCm1197 | MCm1197 | |
| Glucagon | GHRH | human | HEK293T | C1291 | DC1291 | MC1291 |
| GIP | human | HEK293T | C1290 | DC1290 | MC1290 | |
| GIP | human | HEK293T β-Arrestin2 | CA1290 | DCA1290 | MCA1290 | |
| GIP | mouse | HEK293T | Cm1290 | DCm1290 | MCm1290 | |
| GIP | rat | HEK293T | Cr1290 | DCr1290 | MCr1290 | |
| GIP | dog | HEK293T | Cd1290 | DCd1290 | MCd1290 | |
| GIP | dog | HEK293T | Cd1290a | DCd1290a | MCd1290a | |
| GIP | rabbit | HEK293T | Cb1290 | DCb1290 | MCb1290 | |
| GIP | pig | HEK293T | Cp1290 | DCp1290 | MCp1290 | |
| GIP | rhesus monkey | HEK293T | Cpr1290 | DCpr1290 | MCpr1290 | |
| GIP | rhesus monkey | HEK293T | Cpr1290a | DCpr1290a | MCpr1290a | |
| GIP | ferret | HEK293T | Cf1290 | DCf1290 | MCf1290 | |
| GIP | ferret | HEK293T | Cf1290a | DCf1290a | MCf1290a | |
| GLP-1 | human | HEK293T | C1267 | DC1267 | MC1267 | |
| GLP-1 | human | CHO-K1 | C1267-1 | DC1267-1 | MC1267-1 | |
| GLP-1 | human | CHO-K1 | C1267-1a | DC1267-1a | MC1267-1a | |
| GLP-1 | human | CHO-K1 β-Arrestin2 | CA1267-1 | DCA1267-1 | MCA1267-1 | |
| GLP-1 | human | HEK293T β-Arrestin2 | CA1267BA2 | DCA1267BA2 | MCA1267BA2 | |
| GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1 | DCpc1267-1 | MCpc1267-1 | |
| GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1a | DCpc1267-1a | MCpc1267-1a | |
| GLP-1 | rat | CHO-K1 | Cr1267-1 | DCr1267-1 | MCr1267-1 | |
| GLP-1 | dog | CHO-K1 | Cd1267-1 | DCd1267-1 | MCd1267-1 | |
| GLP-1 | dog | HEK293T | Cd1267-1a | DCd1267-1a | MCd1267-1a | |
| GLP-1 | dog | HEK293T | Cd1267-1b | DCd1267-1b | MCd1267-1b | |
| GLP-1 | mouse | CHO-K1 | Cm1267-1 | DCm1267-1 | MCm1267-1 | |
| GLP-1 | mouse | CHO-K1 | Cm1267-1a | DCm1267-1a | MCm1267-1a | |
| GLP-1 | pig | CHO-K1 | Cp1267-1 | DCp1267-1 | MCp1267-1 | |
| GLP-1 | rabbit | CHO-K1 | Cb1267-1 | DCb1267-1 | MCb1267-1 | |
| GLP-1 | rabbit | CHO-K1 | Cb1267-1a | DCb1267-1a | MCb1267-1a | |
| GLP-2 | human | HEK293T | C1268 | DC1268 | MC1268 | |
| GLP-2 | rat | HEK293T | Cr1268 | DCr1268 | MCr1268 | |
| Glucagon | human | HEK293T | C1266 | DC1266 | MC1266 | |
| Glucagon | dog | HEK293T | Cd1266 | DCd1266 | MCd1266 | |
| Glucagon | pig | HEK293T | Cp1266 | DCp1266 | MCp1266 | |
| Glucagon | rat | HEK293T | Cr1266 | DCr1266 | MCr1266 | |
| Glucagon | human | HEK293T | C1266A | DC1266A | MC1266A | |
| Glucagon | human | CHO-K1 | C1266-1 | DC1266-1 | MC1266-1 | |
| Glucagon | human | CHO-K1 | C1266-1a | DC1266-1a | MC1266-1a | |
| Glucagon | human | CHO-K1 β-Arrestin2 | CA1266-1 | DCA1266-1 | MCA1266-1 | |
| Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1 | DCpc1266-1 | MCpc1266-1 | |
| Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1a | DCpc1266-1a | MCpc1266-1a | |
| Glucagon | cynomolgus monkey | HEK293T | Cpc1266 | DCpc1266 | MCpc1266 | |
| Glucagon | cynomolgus monkey | HEK293T | Cpc1266a | DCpc1266a | MCpc1266a | |
| Secretin | human | CHO-K1 | C1228-1 | DC1228-1 | MC1228-1 | |
| Glycoprotein Hormone | TSH | human | HEK293T | H1177 | DH1177 | MH1177 |
| TSH | rat | HEK293T | C1177-1 | DC1177-1 | MC1177-1 | |
| Gonadotrophin-Releasing Hormone | GnRH | human | HEK293T | C1283 | DC1283 | MC1283 |
| GnRH | dog | HEK293T | Cd1283 | DCd1283 | MCd1283 | |
| FSHR | human | HEK293T | C1175 | DC1175 | MC1175 | |
| Histamine | H1 | human | HEK293T | C1027 | DC1027 | MC1027 |
| H1 | mouse | HEK293T | Cm1027 | DCm1027 | MCm1027 | |
| H2 | human | HEK293T | C1028 | DC1028 | MC1028 | |
| H3 | human | HEK293T | C1029 | DC1029 | MC1029 | |
| H3 | human | HEK293T Gαqi5 | CG1029 | DCG1029 | MCG1029 | |
| H3 | mouse | HEK293T | Cm1029 | DCm1029 | MCm1029 | |
| H3 | mouse | CHO-K1 | Cm1029-1 | DCm1029-1 | MCm1029-1 | |
| H4 | human | HEK293T | C1030 | DC1030 | MC1030 | |
| H4 | human | HEK293T Gαqi5 | CG1030 | DCG1030 | MCG1030 | |
| H4 | human | HEK293T β-Arrestin2 | CA1030BA2 | DCA1030BA2 | MCA1030BA2 | |
| H4 | mouse | HEK293T | Cm1030 | DCm1030 | MCm1030 | |
| H4 | mouse | HEK293T Gαqi5 | CGm1030 | DCGm1030 | MCGm1030 | |
| Hydroxycarboxylic acid | GPR81 | human | HEK293T | |||
| KiSS1-Derived Peptide | KiSS1 | human | CHO dhfr- | C1036 | DC1036 | MC1036 |
| KiSS1 | rat | CHO dhfr- | C1036-1 | DC1036-1 | MC1036-1 | |
| Leukotriene/Lipoxin | BLT1 | human | HEK293T | H1165a | DH1165a | H1165a |
| BLT2 | human | HEK293T | C1272 | DC1272 | MC1272 | |
| BLT2 | human | HEK293T | C1272A | DC1272A | MC1272A | |
| BLT2 | human | HEK293T | C1272b | DC1272b | MC1272b | |
| BLT2 | human | HEK293T | C1272c | DC1272c | MC1272c | |
| BLT2 | monkey | HEK293T | Cp1272a | DCp1272a | MCp1272a | |
| BLT2 | monkey | HEK293T | Cp1272 | DCp1272 | MCp1272 | |
| BLT2 | mouse | HEK293T | Cm1272a | DCm1272a | MCm1272a | |
| BLT2 | mouse | HEK293T | Cm1272 | DCm1272 | MCm1272 | |
| CysLT1 | human | HEK293T | C1308 | DC1308 | MC1308 | |
| CysLT2 | human | HEK293T | C1307 | DC1307 | MC1307 | |
| OXE | human | HEK293T | ||||
| Lysophospholipid | GPR87 | human | RH7777 | C1140-6 | DC1140-6 | MC1140-6 |
| LPA1 | human | RH7777 | C1048-6 | DC1048-6 | MC1048-6 | |
| LPA1 | mouse | RH7777 | Cm1048-6A | DCm1048-6A | MCm1048-6A | |
| LPA1 | mouse | RH7777 | Cm1048-6B | DCm1048-6B | MCm1048-6B | |
| LPA1 | rat | RH7777 | Cr1048-6B | DCr1048-6B | MCr1048-6B | |
| LPA2 | human | RH7777 | C1050-6 | DC1050-6 | MC1050-6 | |
| LPA3 | human | RH7777 | C1053-6 | DC1053-6 | MC1053-6 | |
| LPA3 | human | RH7777 | C1053-6a | DC1053-6a | MC1053-6a | |
| LPA4 | human | CHO-K1 | C1087-1a | DC1087-1a | MC1087-1a | |
| LPA4 | human | CHO-K1 | C1087-1b | DC1087-1b | MC1087-1b | |
| LPA5 | human | RH7777 | C1145-6 | DC1145-6 | MC1145-6 | |
| LPA5 | mouse | RH7777 | Cm1145-6 | DCm1145-6 | MCm1145-6 | |
| S1P1 | human | CHO-K1 | C1047-1 | DC1047-1 | MC1047-1 | |
| S1P1 | human | CHO-K1 Gαqi5 | CG1047-1 | DCG1047-1 | MCG1047-1 | |
| S1P2 | human | CHO-K1 | C1051-1 | DC1051-1 | MC1051-1 | |
| S1P2 | human | CHO-K1 Gαqi5 | CG1051-1 | DCG1051-1 | MCG1051-1 | |
| S1P2 | mouse | CHO-K1 | Cm1051-1 | DCm1051-1 | MCm1051-1 | |
| S1P2 | rat | CHO-K1 | Cr1051-1 | DCr1051-1 | MCr1051-1 | |
| S1P3 | human | RH7777 | C1049-6 | DC1049-6 | MC1049-6 | |
| S1P3 | human | CHO-K1 | C1049-1 | DC1049-1 | MC1049-1 | |
| S1P3 | human | CHO-K1 Gαqi5 | CG1049-1 | DCG1049-1 | MCG1049-1 | |
| S1P3 | mouse | CHO-K1 Gαqi5 | CGm1049-1 | DCGm1049-1 | MCGm1049-1 | |
| S1P3 | rat | CHO-K1 Gαqi5 | CGr1049-1 | DCGr1049-1 | MCGr1049-1 | |
| S1P4 | human | CHO-K1 Gαqi5 | CG1052-1 | DCG1052-1 | MCG1052-1 | |
| S1P4 | mouse | CHO-K1 Gαqi5 | CGm1052-1 | DCGm1052-1 | MCGm1052-1 | |
| S1P4 | rat | CHO-K1 Gαqi5 | CGr1052-1 | DCGr1052-1 | MCGr1052-1 | |
| S1P5 | human | CHO-K1 | C1054-1 | DC1054-1 | MC1054-1 | |
| S1P5 | human | CHO-K1 Gαqi5 | CG1054-1 | DCG1054-1 | MCG1054-1 | |
| Melanin-Concentrating Hormone | MCH1 | human | HEK293T Gαqi5 | C1031-3 | DC1031-3 | MC1031-3 |
| MCH1 | rat | HEK293T Gαqi5 | C1031-4 | DC1031-4 | MC1031-4 | |
| MCH2 | human | CHO dhfr- | C1032 | DC1032 | MC1032 | |
| Melanocortin | MC1 | human | HEK293T | C1340 | DC1340 | MC1340 |
| MC4 | human | HEK293T | H1343 | H1343 | H1343 | |
| Melatonin | MT1 | human | CHO-K1 | C1223-1 | DC1223-1 | MC1223-1 |
| MT2 | human | HEK293T Gαqi5 | C1224 | DC1224 | MC1224 | |
| MT2 | mouse | HEK293T | Cm1224 | DCm1224 | MCm1224 | |
| MT2 | rat | HEK293T | Cr1224 | DCr1224 | MCr1224 | |
| Metabotropic Glutamate | mGlu1 | human | CHO-K1 | C1188-1 | DC1188-1 | MC1188-1 |
| mGlu2 | human | HEK293T | C1189a | DC1189a | MC1189a | |
| mGlu2 | human | HEK293T Gqi5 | HG1189Gi | DHG1189Gi | MHG1189Gi | |
| mGlu2 | human | HEK293T Gαqi5 | HG1189 | HG1189 | HG1189 | |
| mGlu2 | human | HEK293T Gαqi5 | HG1189a | HG1189a | HG1189a | |
| mGlu2 | rat | HEK293T Gαqi5 | HGr1189b | DHGr1189b | MHGr1189b | |
| mGlu3 | human | HEK293T Gαqi5 | CG1190 | DCG1190 | MCG1190 | |
| mGlu4 | dog | CHO-K1 Gαqi5 | HGd1191-1 | DHGd1191-1 | MHGd1191-1 | |
| mGlu4 | human | HEK293T | C1191a | DC1191a | MC1191a | |
| mGlu4 | human | HEK293T Gαqi5 | CG1191 | DCG1191 | MCG1191 | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1a | DHGm1191-1a | MHGm1191-1a | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1b | DHGm1191-1b | MHGm1191-1b | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1c | DHGm1191-1c | MHGm1191-1c | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1d | DHGm1191-1d | MHGm1191-1d | |
| mGlu4 | rat | HEK293T | Cr1191 | DCr1191 | MCr1191 | |
| mGlu4 | human | HEK293T Gαqi5 | CG1191a | DCG1191a | MCG1191a | |
| mGlu5 | human | HEK293T | C1192 | DC1192 | MC1192 | |
| mGlu5 | human | HEK293T B-ARRESTIN2 | CA1192BA2 | DCA1192BA2 | MCA1192BA2 | |
| mGlu6 | human | HEK293T | C1193 | DC1193 | MC1193 | |
| mGlu6 | human | HEK293T Gαqi5 | CG1193 | DCG1193 | MCG1193 | |
| mGlu7 | human | HEK293T | C1194 | DC1194 | MC1194 | |
| mGlu7 | human | HEK293T Gαqi5 | CG1194 | DCG1194 | MCG1194 | |
| mGlu8 | human | HEK293T | C1195 | DC1195 | MC1195 | |
| mGlu8 | human | HEK293T | C1195a | DC1195a | MC1195a | |
| mGlu8 | human | HEK293T Gαqi5 | CG1195 | DCG1195 | MCG1195 | |
| mGlu8 | human | CHO-K1 | C1195-1a | DC1195-1a | MC1195-1a | |
| Motilin | motilin | human | HEK293T | H1297 | H1297 | H1297 |
| Muscarinic | M1 | human | CHO-K1 | C1022-1 | DC1022-1 | MC1022-1 |
| M1 | human | CHO-K1 | C1022-1a | DC1022-1a | MC1022-1a | |
| M2 | human | CHO-K1 | C1023-1 | DC1023-1 | MC1023-1 | |
| M3 | human | CHO-K1 | C1024-1 | DC1024-1 | MC1024-1 | |
| M3 | mouse | CHO-K1 | Cm1024-1 | DCm1024-1 | MCm1024-1 | |
| M4 | human | CHO-K1 | C1025-1 | DC1025-1 | MC1025-1 | |
| M4 | human | CHO-K1 Gαqi5 | CG1025-1 | DCG1025-1 | MCG1025-1 | |
| M4 | mouse | CHO-K1 | Cm1025-1 | DCm1025-1 | MCm1025-1 | |
| M5 | human | CHO-K1 | C1026-1 | DC1026-1 | MC1026-1 | |
| N-formylpeptide | FPR1 | human | HEK293T | C1243 | DC1243 | MC1243 |
| FPR1 | human | HEK293T | C1243a | DC1243a | MC1243a | |
| FPR1 | human | HEK293T Gαqi5 | CG1243 | DCG1243 | MCG1243 | |
| FPR2 | human | HEK293T | C1244 | DC1244 | MC1244 | |
| FPR2 | human | HEK293T | C1244a | DC1244a | MC1244a | |
| FPR3 | human | HEK293T | C1245 | DC1245 | MC1245 | |
| Neuromedin U | NMU1 | human | HEK293T | C1122 | DC1122 | MC1122 |
| NMU2 | human | HEK293T | C1213 | DC1213 | MC1213 | |
| Neuropeptide FF/AF | NPFF1 | human | HEK293T | C1363 | DC1363 | MC1363 |
| NPFF2 | human | HEK293T Gαqi5 | CG1364 | DCG1364 | MCG1364 | |
| Neuropeptide S | NPS | mouse | HEK293T | C1355-1 | DC1355-1 | MC1355-1 |
| NPS | human | HEK293T | C1355a | DC1355a | MC1355a | |
| NPS(2) | human | HEK293T | C1356 | DC1356 | MC1356 | |
| NPSIle107 | human | HEK293T | C1355-2 | DC1355-2 | MC1355-2 | |
| Neuropeptide W/B | NPBW1 | rat | HEK293T Gαqi5 | C1124-1 | DC1124-1 | MC1124-1 |
| NPBW1 | human | HEK293T Gαqi5 | C1124 | DC1124 | MC1124 | |
| NPBW2 | human | HEK293T Gαqi5 | C1133 | DC1133 | MC1133 | |
| Neuropeptide Y | Y1 | human | CHO-K1 Gαqi5 | CG1273-1 | DCG1273-1 | MCG1273-1 |
| Y2 | human | CHO-K1 Gαqi5 | CG1274-1 | DCG1274-1 | MCG1274-1 | |
| Y2 | rat | CHO-K1 | Cr1274-1 | DCr1274-1 | MCr1274-1 | |
| Y4 | human | CHO-K1 | C1300-1 | DC1300-1 | MC1300-1 | |
| Y4 | human | CHO-K1 Gαqi5 | CG1300-1 | DCG1300-1 | MCG1300-1 | |
| Y5 | human | HEK293T | C1275a | DC1275a | MC1275a | |
| Y5 | human | HEK293T Gαqi5 | CG1275 | DCG1275 | MCG1275 | |
| Neurotensin | NTS1 | human | CHO-K1 | C1276-1 | DC1276-1 | MC1276-1 |
| NTS2 | human | CHO-K1 | C1277-1 | DC1277-1 | MC1277-1 | |
| NTS2 | human | HEK293T | C1277 | DC1277 | MC1277 | |
| NTS2 | human | HEK293T | C1277a | DC1277a | MC1277a | |
| Nicotinic Acid | GPR109A | human | CHO-K1 | C1370-1 | DC1370-1 | MC1370-1 |
| GPR109B | human | CHO-K1 | C1059-1 | DC1059-1 | MC1059-1 | |
| GPR81 | human | HEK293T | C1134 | DC1134 | MC1134 | |
| Opioid | delta | human | CHO-K1 | C1351-1 | DC1351-1 | MC1351-1 |
| delta | human | CHO-K1 Gαqi5 | CG1351-1 | DCG1351-1 | MCG1351-1 | |
| delta | human | CHO-K1 | CA1351-1 | DCA1351-1 | MCA1351-1 | |
| delta | rat | CHO dhfr- | C1351 | DC1351 | MC1351 | |
| kappa | human | CHO-K1 | C1352-1a | DC1352-1a | MC1352-1a | |
| kappa | human | CHO-K1 Gαqi5 | CG1352-1 | DCG1352-1 | MCG1352-1 | |
| kappa | human | CHO-K1 | CA1352-1a | DCA1352-1a | MCA1352-1a | |
| kappa | human | CHO-K1 β-Arrestin2 | CA1352BA2-1 | DCA1352BA2-1 | MCA1352BA2-1 | |
| kappa | human | HEK293T | C1352 | DC1352 | MC1352 | |
| kappa | rat | CHO dhfr- | C1352-1 | DC1352-1 | MC1352-1 | |
| kappa | rat | CHO dhfr- | Cr1352-8 | DCr1352-8 | MCr1352-8 | |
| mu | human | CHO-K1 | C1350-1a | DC1350-1a | MC1350-1a | |
| mu | human | CHO-K1 Gαqi5 | CG1350-1a | DCG1350-1a | MCG1350-1a | |
| mu | human | CHO-K1 | CA1350-1a | DCA1350-1a | MCA1350-1a | |
| mu | rat | CHO dhfr- | Cr1350-1a | DCr1350-1a | MCr1350-1a | |
| mu Mutant Y150F | human | CHO-K1 | C1350-1MT1 | DC1350-1MT1 | MC1350-1MT1 | |
| mu Mutant Y150A | human | CHO-K1 | C1350-1MT2 | DC1350-1MT2 | MC1350-1MT2 | |
| mu Mutant M153A | human | CHO-K1 | C1350-1MT3 | DC1350-1MT3 | MC1350-1MT3 | |
| mu Mutant H299N | human | CHO-K1 | C1350-1MT4 | DC1350-1MT4 | MC1350-1MT4 | |
| mu Mutant H299A | human | CHO-K1 | C1350-1MT5 | DC1350-1MT5 | MC1350-1MT5 | |
| NOP | human | CHO-K1 | C1354-1 | DC1354-1 | MC1354-1 | |
| NOP | human | CHO-K1 Gαqi5 | CG1354-1 | DCG1354-1 | MCG1354-1 | |
| NOP | human | CHO-K1 β-Arrestin2 | CA1354-1 | DCA1354-1 | MCA1354-1 | |
| NOP | human | HEK293T | C1354a | DC1354a | MC1354a | |
| NOP | rat | CHO dhfr- | Cr1354 | DCr1354 | MCr1354 | |
| Orexin | OX1 | human | CHO-K1 | C1033-1 | DC1033-1 | MC1033-1 |
| OX2 | human | CHO-K1 | C1034-1 | DC1034-1 | MC1034-1 | |
| Orphan | GPR3 | human | HEK293T | C1091 | DC1091 | MC1091 |
| GPR6 | human | HEK293T | C1116 | DC1116 | MC1116 | |
| GPR6 | human | HEK293T | C1116a | DC1116a | MC1116a | |
| GPR15 | human | HEK293T | C1069 | DC1069 | MC1069 | |
| GPR34 | human | HEK293T Gαqi5 | CG1095 | DCG1095 | MCG1095 | |
| GPR35 | dog | HEK293T Gα16 | CGd1096 | DCGd1096 | MCGd1096 | |
| GPR35 | dog | CHO-K1 Gα16 | CGd1096-1 | DCGd1096-1 | MCGd1096-1 | |
| GPR35 | mouse | CHO-K1 | Cm1096-1 | DCm1096-1 | MCm1096-1 | |
| GPR35 | mouse | CHO-K1 Gα16 | CGm1096-1 | DCGm1096-1 | MCGm1096-1 | |
| GPR35 (short form) | human | CHO-K1 | C1096-1 | DC1096-1 | MC1096-1 | |
| GPR35 (short form) | human | CHO-K1 β-Arrestin2 | CA1096-1 | DCA1096-1 | MCA1096-1 | |
| GPR35 (short form) | human | CHO-K1 Gα16 | CG1096-1 | DCG1096-1 | MCG1096-1 | |
| GPR35 (short form) | human | HEK293T Gα16 | CG1096 | DCG1096 | MCG1096 | |
| GPR35 (long form) | human | CHO-K1 β-Arrestin2 | CA1523-1 | DCA1523-1 | MCA1523-1 | |
| GPR35 (long form) T108M Mutant | human | CHO-K1 β-Arrestin2 | CA1524-1 | DCA1524-1 | MCA1524-1 | |
| GPR37L1 | human | HEK293T | C1098 | DC1098 | MC1098 | |
| GPR45 | human | CHO-K1 | CG1106-1 | DCG1106-1 | MCG1106-1 | |
| GPR45 | human | CHO-K1 | CG1106-1a | DCG1106-1a | MCG1106-1a | |
| GPR50 | human | HEK293T | C1110 | DC1110 | MC1110 | |
| GPR52 | human | HEK293T | C1112 | DC1112 | MC1112 | |
| GPR52 | human | HEK293T | C1112a | DC1112a | MC1112a | |
| GPR52 | human | HEK293T β-Arrestin2 | CA1112BA2 | DCA1112BA2 | MCA1112BA2 | |
| GPR61 | human | HEK293T | C1117 | DC1117 | MC1117 | |
| GPR61 | human | HEK293T | C1117a | DC1117a | MC1117a | |
| GPR61 | human | HEK293T | C1117b | DC1117b | MC1117b | |
| GPR75 | human | HEK293T | C1129 | DC1129 | MC1129 | |
| GPR85 | human | HEK293T | C1138 | DC1138 | MC1138 | |
| GPR85 | human | CHO-K1 | C1138-1 | DC1138-1 | MC1138-1 | |
| GPR88 | human | CHO-K1 | C1141-1 | DC1141-1 | MC1141-1 | |
| GPR88 | rat | CHO-K1 | Cr1141-1 | DCr1141-1 | MCr1141-1 | |
| GPR142 | human | HEK293T | C1286 | DC1286 | MC1286 | |
| GPR142 | human | HEK293T | C1286a | DC1286a | MC1286a | |
| GPR151 | human | CHO-K1 Gα16 Gαqi5 | CG1181-1 | DCG1181-1 | MCG1181-1 | |
| GPRC5A | human | HEK293T | CA1525 | DCA1525 | MCA1525 | |
| MRGX1 | human | CHO dhfr-Gαqi5 | C1256 | DC1256 | MC1256 | |
| MRGX1 | human | HEK293T | C1256a | DC1256a | MC1256a | |
| MRGX2 | human | HEK293T Gαqi5 | C1257 | DC1257 | MC1257 | |
| MRGX2 | human | HEK293T | C1257a | DC1257a | MC1257a | |
| MRGX2 | human | HEK293T | C1257b | DC1257b | MC1257b | |
| MRGX2 | rhesus monkey | CHO-K1 | Cpr1257-1 | DCpr1257-1 | MCpr1257-1 | |
| MRGX2 | human | HEK293T β-Arrestin2 | CA1257aBA2 | DCA1257aBA2 | MCA1257aBA2 | |
| MRGX2 | human | HEK293T β-Arrestin2 | CA1257bBA2 | DCA1257bBA2 | MCA1257bBA2 | |
| MRGX4 | human | HEK293T | C1259 | DC1259 | MC1259 | |
| MAS1 | human | HEK293T | C1225 | DC1225 | MC1225 | |
| Oxysterol | EBI2 | human | CHO-K1 Gαqi5 | CG1242-1 | DCG1242-1 | MCG1242-1 |
| EBI2 | mouse | CHO-K1 Gαqi5 | CGm1242-1 | DCGm1242-1 | MCGm1242-1 | |
| EBI2 | mouse | CHO-K1 | Cm1242-1 | DCm1242-1 | MCm1242-1 | |
| Parathyroid Hormone | PTH1 | human | HEK293T | C1301 | DC1301 | MC1301 |
| PTH1 | human | HEK293T | C1301-1 | DC1301-1 | MC1301-1 | |
| PTH2 | human | HEK293T | H1302 | DH1302 | H1302 | |
| Platelet-Activating Factor | PAF | human | HEK293T | C1218 | DC1218 | MC1218 |
| Prokineticin | PK1 | human | CHO-K1 | C1128-1 | DC1128-1 | MC1128-1 |
| PK2 | human | CHO-K1 | C1127-1 | DC1127-1 | MC1127-1 | |
| PK2 | human | CHO-K1 | C1127-1a | DC1127-1a | MC1127-1a | |
| PK2 mutant | human | CHO-K1 | C1127CT-1 | DC1127DCT-1 | MC1127MCT-1 | |
| Prolactin-Releasing Peptide | PrRP | human | CHO dhfr- | C1037 | DC1037 | MC1037 |
| Prostanoid | DP1 | human | HEK293T | C1200 | DC1200 | MC1200 |
| DP2 | human | HEK293T | H1105 | DH1105 | MH1105 | |
| DP2 | human | HEK293T | H1105a | DH1105a | MH1105a | |
| EP1 | human | HEK293T | C1201a | DC1201a | MC1201a | |
| EP2 | human | HEK293T | C1202 | DC1202 | MC1202 | |
| EP2 | mouse | HEK293T | Cm1202 | DCm1202 | MCm1202 | |
| EP2 | mouse | HEK293T | Cm1202-3 | DCm1202-3 | MCm1202-3 | |
| EP2 | rat | HEK293T | Cr1202 | DCr1202 | MCr1202 | |
| EP2 | rat | HEK293T | Cr1202-134 | DCr1202-134 | MCr1202-134 | |
| EP3 | human | CHO-K1 | C1203-1 | DC1203-1 | MC1203-1 | |
| EP3 | human | CHO-K1 | C1203-1a | DC1203-1a | MC1203-1a | |
| EP3 | human | CHO-K1 | C1203-1b | DC1203-1b | MC1203-1b | |
| EP3 | human | CHO-K1 | C1203-1c | DC1203-1DC | MC1203-1MC | |
| EP3 | human | CHO-K1 | C1203-1d | DC1203-1d | MC1203-1d | |
| EP4 | human | HEK293T | C1204 | DC1204 | MC1204 | |
| FP | human | HEK293T | C1205 | DC1205 | MC1205 | |
| IP1 | human | CHO-K1 | C1206-1 | DC1206-1 | MC1206-1 | |
| TP | human | HEK293T | C1365 | DC1365 | MC1365 | |
| TP | human | HEK293T | H1365 | H1365 | H1365 | |
| Protease-Activated | PAR1 | human | CHO-K1 | C1207-1 | DC1207-1 | MC1207-1 |
| PAR1 | human | HeLa | C1207-7 | DC1207-7 | MC1207-7 | |
| PAR2 | human | HeLa | C1208-7 | DC1208-7 | MC1208-7 | |
| PAR4 | human | HeLa | C1210-7 | DC1210-7 | MC1210-7 | |
| Proton-Sensing Receptors | GPR4 | human | HEK293T | C1100 | DC1100 | MC1100 |
| GPR4 | human | HEK293T | CA1100 | DCA1100 | MCA1100 | |
| GPR65 | human | HEK293T | C1121 | DC1121 | MC1121 | |
| GPR65 | human | HEK293T | CA1121 | DCA1121 | MCA1121 | |
| GPR65 | human | HEK293T | C1121a | DC1121a | MC1121a | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP20 | DC1121-CSP20 | MC1121-CSP20 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP23 | DC1121-CSP23 | MC1121-CSP23 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP30 | DC1121-CSP30 | MC1121-CSP30 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP36 | DC1121-CSP36 | MC1121-CSP36 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP38 | DC1121-CSP38 | MC1121-CSP38 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP44 | DC1121-CSP44 | MC1121-CSP44 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP75 | DC1121-CSP75 | MC1121-CSP75 | |
| GPR68 | human | HEK293T | C1123 | DC1123 | MC1123 | |
| GPR68 | human | HEK293T | CA1123 | DCA1123 | MCA1123 | |
| GPR132 | human | HEK293T | CA1066 | DCA1066 | MCA1066 | |
| Purinergic | GPR17 (short form) | human | 1321N1 | C1526-3 | DC1526-3 | MC1526-3 |
| GPR17 | mouse | 1321N1 | Cm1526-3 | DCm1526-3 | MCm1526-3 | |
| GPR17 | rat | 1321N1 | Cr1526-3 | DCr1526-3 | MCr1526-3 | |
| GPR17 | rat | 1321N1 | Cr1525-3 | DCr1525-3 | MCr1525-3 | |
| P2Y1 | human | 1321N1 | C1160-3 | DC1160-3 | MC1160-3 | |
| P2Y2 | human | 1321N1 | C1161-3 | DC1161-3 | MC1161-3 | |
| P2Y2 | human | HEK293T | C1161 | DC1161 | MC1161 | |
| P2Y2 | rat | 1321N1 | Cr1161-3 | DCr1161-3 | MCr1161-3 | |
| P2Y4 | human | 1321N1 | C1162-3 | DC1162-3 | MC1162-3 | |
| P2Y6 | human | 1321N1 | C1164-3 | DC1164-3 | MC1164-3 | |
| P2Y11 | human | 1321N1 | C1169-3 | DC1169-3 | MC1169-3 | |
| P2Y12 | human | 1321N1 | C1170-3 | DC1170-3 | MC1170-3 | |
| P2Y12 | human | 1321N1 | C1170-3a | DC1170-3a | MC1170-3a | |
| P2Y12 | rat | CHO dhfr- | C1170-1 | DC1170-1 | MC1170-1 | |
| P2Y13 | human | 1321N1 | C1139-3 | DC1139-3 | MC1139-3 | |
| P2Y14 | human | HEK293T | C1057 | DC1057 | MC1057 | |
| P2Y14 | human | HEK293T Gαqi5 | CG1057 | DCG1057 | MCG1057 | |
| P2Y14 | rat | HEK293T Gαqi5 | CGr1057 | DCGr1057 | MCGr1057 | |
| P2Y14 | monkey | HEK293T Gαqi5 | CGp1057 | DCGp1057 | MCGp1057 | |
| Relaxin | RXFP1 | human | HEK293T | C1287 | DC1287 | MC1287 |
| RXFP1 | human | HEK293T | C1287NTa | DC1287NTa | MC1287NTa | |
| RXFP1 | human | HEK293T | C1287NTb | DC1287NTb | MC1287NTb | |
| RXFP2 | human | HEK293T | C1289NTa | DC1289NTa | MC1289NTa | |
| RXFP2 | human | HEK293T | C1289NTb | DC1289NTb | MC1289NTb | |
| RXFP3 | human | HEK293T | C1306 | DC1306 | MC1306 | |
| SARS-CoV-2 | ACE2 | human | HEK293T | C2006 | DC2006 | MC2006 |
| TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 | |
| Serotonin | 5-HT1A | human | HEK293T | C1319 | DC1319 | MC1319 |
| 5-HT1A | human | HEK293T | C1319a | DC1319a | MC1319a | |
| 5-HT1B | human | HEK293T | C1320 | DC1320 | MC1320 | |
| 5-HT1B | human | HEK293T | C1320a | DC1320a | MC1320a | |
| 5-HT1B | human | HEK293T Gαqi5 | CG1320 | DCG1320 | MCG1320 | |
| 5-HT2A | human | HEK293T | C1324 | DC1324 | MC1324 | |
| 5-HT2A | human | CHO-K1 | C1324-1 | DC1324-1 | MC1324-1 | |
| 5-HT2A | mouse | HEK293T | Cm1324 | DCm1324 | MCm1324 | |
| 5-HT2A | mouse | CHO-K1 | Cm1324-1 | DCm1324-1 | MCm1324-1 | |
| 5-HT2A | dog | HEK293T | Cd1324 | DCd1324 | MCd1324 | |
| 5-HT2B | human | CHO-K1 | C1325-1 | DC1325-1 | MC1325-1 | |
| 5-HT2B | human | HEK293T | C1325 | DC1325 | MC1325 | |
| 5-HT2B | mouse | HEK293T | Cm1325 | DCm1325 | MCm1325 | |
| 5-HT2C | human | CHO-K1 | C1326-1 | DC1326-1 | MC1326-1 | |
| 5-HT4A | human | CHO-K1 | C1518-1 | DC1518-1 | MC1518-1 | |
| 5-HT4A | mouse | CHO-K1 | Cm1518-1 | DCm1518-1 | MCm1518-1 | |
| 5-HT4B | human | CHO-K1 | C1330-1 | DC1330-1 | MC1330-1 | |
| 5-HT4B | human | HEK293T | C1330 | DC1330 | MC1330 | |
| 5-HT4D | human | CHO-K1 | C1520-1 | DC1520-1 | MC1520-1 | |
| 5-HT6 | human | CHO-K1 | C1331-1 | DC1331-1 | MC1331-1 | |
| 5-HT7 | human | HEK293T | C1334 | DC1334 | MC1334 | |
| Somatostatin | sst1 | human | CHO-K1 | C1345-1a | DC1345-1a | MC1345-1a |
| sst1 | human | CHO-K1 Gα16 | CG1345-1 | DCG1345-1 | MCG1345-1 | |
| sst2 | human | CHO-K1 | C1346-1 | DC1346-1 | MC1346-1 | |
| sst2 | human | CHO-K1 Gα16 | CG1346-1 | DCG1346-1 | MCG1346-1 | |
| sst3 | human | CHO-K1 | C1347-1 | DC1347-1 | MC1347-1 | |
| sst3 | human | CHO-K1 Gα16 | CG1347-1 | DCG1347-1 | MCG1347-1 | |
| sst4 | human | CHO-K1 | C1348-1a | DC1348-1a | MC1348-1a | |
| sst4 | human | CHO-K1 Gα16 | CG1348-1 | DCG1348-1 | MCG1348-1 | |
| sst5 | human | CHO-K1 | C1349-1 | DC1349-1 | MC1349-1 | |
| sst5 | human | CHO-K1 Gα16 | CG1349-1 | DCG1349-1 | MCG1349-1 | |
| Tachykinin | NK1 | human | HEK293T | C1303 | DC1303 | MC1303 |
| NK2 | human | HEK293T | C1304 | DC1304 | MC1304 | |
| NK3 | human | HEK293T | C1305 | DC1305 | MC1305 | |
| NK3 | rat | HEK293T | Cr1305 | DCr1305 | MCr1305 | |
| NK3 | mouse | HEK293T | Cm1305 | DCm1305 | MCm1305 | |
| Thyrotropin-Releasing Hormone | TRH | human | HEK293T | |||
| Trace Amine | TA1 | rat | HEK293T | C1357 | DC1357 | MC1357 |
| TA1 | human | HEK293T | C1357a | DC1357a | MC1357a | |
| TA1 | rat | HEK293T Gαqi5 | Cr1357 | DCr1357 | MCr1357 | |
| Urotensin | UT | rat | CHO dhfr- | C1035-1 | DC1035-1 | MC1035-1 |
| UT | human | CHO-K1 | C1035-1a | DC1035-1a | MC1035-1a | |
| Vasoactive Intestinal Peptide | PAC1 | human | HEK293T | C1415 | DC1415 | MC1415 |
| VPAC1 | human | CHO-K1 | C1292-1 | DC1292-1 | MC1292-1 | |
| VPAC2 | human | HEK293T | H1293 | DH1293 | MH1293 | |
| Vasopressin/Oxytocin | OT | human | CHO-K1 | C1299-1 | DC1299-1 | MC1299-1 |
| OT | rabbit | HEK293T | Cb1299 | DCb1299 | MCb1299 | |
| OT | rabbit | HEK293T | Cb1299L | DCb1299L | MCb1299L | |
| V1A | human | CHO-K1 | C1042-1 | DC1042-1 | MC1042-1 | |
| V1A | rabbit | HEK293T | Cb1042 | DCb1042 | MCb1042 | |
| V1B | human | CHO-K1 | C1043-1 | DC1043-1 | MC1043-1 | |
| V1B | rabbit | HEK293T | Cb1043 | DCb1043 | MCb1043 | |
| V1B | rabbit | HEK293T | Cb1043L | DCb1043L | MCb1043L | |
| V2 | human | CHO-K1 | C1044-1 | DC1044-1 | MC1044-1 | |
| V2 | rabbit | HEK293T | Cb1044 | DCb1044 | MCb1044 | |
| V2 | rabbit | HEK293T | Cb1044L | DCb1044L | MCb1044L | |
| V2 | dog | CHO-K1 | Cd1044-1 | DCd1044-1 | MCd1044-1 | |
| Zinc | GPR39 | human | HEK293T | H1099 | DH1099 | MH1099 |
| Target Family | Target | Species | Cells |
|---|---|---|---|
| Kinase | AMPK | human | C2C12 |
| DNA-PK | human | Hela | |
| Aryl Hydrocarbon Receptor (Nuclear Hormone Receptor) | AHR | human | Hep G2 |
| AHR | mouse | Hepa1-6 | |
| AHR | human | HG2L6.1c1 CALUX | |
| AHR | mouse | H1L6.c3 CALUX | |
| Chemokine | CCR4 | human | H9 |
| CCR6 | human | H9 | |
| Calcitonin | CGRP | human | SK-N-MC |
| Free Fatty Acid | GPR40 | mouse | MIN6 |
| Lysophospholipid | LPA | human | Human Fibroblast-Like Synoviocytes-Rheumatoid |
| Melanin-Concentrating Hormone | MCH1 | human | YS35 |
| Opioid | mu | human | SK-N-SH |
| Serotonin | 5-HT | human | Human Heart Valvular Interstitial Cells |
| Receptor Family | Target | Species | Parental | Stable Cell Line | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Integrin | a V b 1 | human | CHOB2 | C3001-1 | DC3001-1 | MC3001-1 |
| Potassium Channel | TMEM175 | human | HEK293T | C1527 | DC1527 | MC1527 |
| TMEM175 | human | HEK293T | C1527a | DC1527a | MC1527a | |
| Receptor Tyrosine Kinases | TrKA | human | CHO-K1 | CK1001-1 | DCK1001-1 | MCK1001-1 |
| TrKA | human | CHO-K1 | CK1001-1b | DCK1001-1b | MCK1001-1b | |
| TrKA | rat | CHO-K1 | CKr1001-1 | DCKr1001-1 | MCKr1001-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1 | DCK1002-1 | MCK1002-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1a | DCK1002-1a | MCK1002-1a | |
| SARS-CoV-2 | TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 |
| Zinc Transporter | ZnT3 | human | Hela | C2001-7 | DC2001-7 | MC2001-7 |
| ZnT8 | human | CHO-K1 | C2002-1 | DC2002-1 | MC2002-1 |
| Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|
| HEK293T | DC0001 | MC0001 | |
| HEK293T Gαqi5 | CG0001 | DCG0001 | MCG0001 |
| CHO-K1 | DC0001-1 | MC0001-1 | |
| CHO-K1 Gαqi5 | CG0001-1 | DCG0001-1 | MCG0001-1 |
| CHO-K1 Gα16 | CG0002-1 | DCG0002-1 | MCG0002-1 |
| CHO-K1 Gα16 Gαqi5 | CG0003-1 | DCG0003-1 | MCG0003-1 |
| CHO dhfr- | DCD0001-1 | MCD0001-1 | |
| CHO-K1 NFAT | CK0001-1 | DCK0001-1 | MCK0001-1 |
| 1321N1 | DC0001-3 | MC0001-3 | |
| RH7777 | DC0001-6 | MC0001-6 | |
| Hela | DC0001-7 | MC0001-7 |
| Assay Kit | Unit Size (384-well) | Catalog | Description | Data |
|---|---|---|---|---|
| MULTISCREEN™ β-Arrestin Assay Kit | 1 plate 96- well/384-well | MSBAK01-1 | The kits contain the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Validated by MULTISCREEN™ stable cell lines co-expressing target GPCRs and MULTISCREEN™ β-Arrestin sensors. Suitable for any cell line or primary cells co-expressing endogenous or untagged GPCR target and MULTISCREEN™ β-Arrestin sensor. |  β-Arrestin Recruitment Dose Response in MULTISCREEN™ MOR β-Arrestin2 CHO-K1 stable cell line (CA1350-1a) measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in assay buffer in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | MSBAK01-10 | |||
| 100 plates 96-well/384-well | MSBAK01-100 | |||
| MULTISCREEN™ β-Arrestin BacMam Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKBM01-1 Or β-Arrestin2 MSBAKBM02-1 | The kits contain BacMam viral particles of MULTISCREEN™ β-Arrestin sensor cDNA, control GFP BacMam viral particle, the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. |  β-Arrestin Recruitment Dose Response in MULTISCREEN™ MOR CHO-K1 stable cell line (C1350-1a) infected with β-Arrestin sensor BacMam virus for 48 hours before being measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-10 Or β-Arrestin2 MSBAKBM02-10 |
|||
| 100 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-100 Or β-Arrestin2 MSBAKBM02-100 |
|||
| MULTISCREEN™ β-Arrestin HSV Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKHSV01-1 Or β-Arrestin2 MSBAKHSV02-1 | The kits contain HSV viral particles of MULTISCREEN™ β-Arrestin sensor cDNA, control GFP HSV viral particle, the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. |  β-Arrestin Recruitment Dose Response in MULTISCREEN™ KOR HEK293T stable cell line (C1352) infected with β-Arrestin HSV sensor for 48 hours before being measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist Dynorphin B and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-10 Or β-Arrestin2 MSBAKHSV02-10 |
|||
| 100 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-100 Or β-Arrestin2 MSBAKHSV02-100 |
|||
| MULTISCREEN™ Calcium 1.0 No Wash Assay Kit | 1000 tests | MSCA01-1 | MULTISCREEN™ Calcium 1.0 No Wash Assay Kits provide homogeneous fluorescence-based assays for intracellular calcium mobilization detection in 96-well, 384-well and higher multiplexity. Pre-loaded with Calcium 1.0 is taken up by the cells where the lipophilic blocking groups of Calcium 1.0 are cleaved by esterases, resulting in a negatively charged fluorescent dye that stays inside cells. The fluorescence signal is greatly enhanced after binding to intracellular calcium released by cell-stimulation. Long wavelength, high sensitivity, and >100 times fluorescence enhancement make Calcium 1.0 an ideal indicator for intracellular calcium release assays measuring GPCRs, calcium channels and receptor tyrosine kinase signaling. MULTISCREEN™ Calcium 1.0 No Wash Assay Kits are validated by MULTISCREEN™ stable cell lines. |  Calcium Dose Response in MULTISCREEN™ A2B-HEK293T stable cell line (C1429) measured with MULTISCREEN™ Calcium 1.0 No Wash Assay Kit. Cells were seeded in assay buffer in a 384-well black wall clear bottom PDL-coated plate, incubated with the MULTISCREEN™ Calcium 1.0 No Wash Assay Kit before being treated with control agonist NECA and measured by FLIPR. |
| 10000 tests | MSCA01-10 | |||
| 100000 tests | MSCA01-100 | |||
| MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kit | 500 tests | MSCM01-1 | MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kits provide a homogenous TR-FRET assay method for adenylyl cyclase activity detection in 96-well, 384-well and higher multiplexity. α-cAMP antibody (Ab) is labeled with MULTISCREEN™Eu while cAMP is labeled with MULTISCREEN™650. In the absence of cAMP, MULTISCREEN™650-cAMP is bound to MULTISCREEN™Eu-α-cAMP-Ab to give a strong TR-FRET Emission at 655 nm. Free cAMP in the test sample competes for binding to the MULTISCREEN™ Eu-α-cAMP-Ab, reducing TR-FRET signal from MULTISCREEN™650-cAMP binding. The MULTISCREEN™650-cAMP only has fluorescence lifetime of nanosecond while MULTISCREEN™Eu-α-cAMP-Ab has much longer fluorescence lifetime value due to TR-FRET. The magnitude of TR-FRET is proportional to the concentration of cAMP in a sample. MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kits are validated by MULTISCREEN™ stable cell lines. |  cAMP Dose-Response in MULTISCREEN™ β1-HEK293T stable cell line (C1437-1) measured with MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kit. Cells were seeded in a 384-well solid white plate, incubated with Isoproterenol and 1mM IBMX before being treated with MULTISCREEN™Eu-α-cAMP-Ab and MULTISCREEN™650-cAMP, and measured by FlexStation 3. |
| 5000 tests | MSCM01-5 | |||
| 25000 tests | MSCM01-25 | |||
| MULTISCREEN™ Cell Viability Assay Kit | 400 tests | MSCV01-1 | The MULTISCREEN™ Cell Viability Assay Kit (DTT free) delivers a fast, simple, and highly sensitive luminescence assay for monitoring cell proliferation, viability, and toxicity in mammalian cells. Using firefly luciferase to detect endogenous ATP, it provides bright, stable signals with sensitivity to detect as low as 50 cells per well. Ready-to-use and compatible with 96- and 384-well plates, the kit ensures reliable, reproducible results and has been validated with MULTISCREEN™ stable cell lines, making it an ideal choice for accurate, efficient cell viability testing. |  ATP Dose-Response in MULTISCREEN™ MDA-MB-231 parental cells measured with MULTISCREEN™ Cell Viability Assay Kit. Cells were seeded in a 384-well solid white plate, incubated with compound before addition of MULTISCREEN™ ATP assay reagent, and measured by FlexStation 3. |
| 4000 tests | MSCV01-10 | |||
| 40000 tests | MSCV01-100 |
| Receptor Family | Receptor | Species | Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Adenosine | A1 | human | HEK293T | C1427B | DC1427B | MC1427B |
| A1 | human | CHO-K1 | C1427-1 | DC1427-1 | MC1427-1 | |
| A1 | rat | HEK293T | Cr1427 | DCr1427 | MCr1427 | |
| A2A | human | HEK293T | C1428 | DC1428 | MC1428 | |
| A2A | human | CHO-K1 | C1428-1 | DC1428-1 | MC1428-1 | |
| A2A | mouse | HEK293T | Cm1428A | DCm1428A | MCm1428A | |
| A2A | mouse | HEK293T | Cm1428B | DCm1428B | MCm1428B | |
| A2A | mouse | CHO-K1 | Cm1428-1 | DCm1428-1 | MCm1428-1 | |
| A2A | rat | HEK293T | Cr1428 | DCr1428 | MCr1428 | |
| A2B | human | HEK293T | C1429 | DC1429 | MC1429 | |
| A2B | human | CHO-K1 | C1429-1 | DC1429-1 | MC1429-1 | |
| A2B | human | HEK293T | C1429a | DC1429a | MC1429a | |
| A2B | rat | HEK293T | Cr1429 | DCr1429 | MCr1429 | |
| A3 | human | HEK293T | C1430 | DC1430 | MC1430 | |
| A3 | human | CHO-K1 | C1430-1 | DC1430-1 | MC1430-1 | |
| A3 | rat | HEK293T | Cr1430 | DCr1430 | MCr1430 | |
| Adhesion Class GPCRs | GPR97 | human | HEK293T | C1396 | DC1396 | MC1396 |
| GPR110 | human | HEK293T | C1378 | DC1378 | MC1378 | |
| Adrenergic | alpha1A | human | CHO-K1 | C1431-1 | DC1431-1 | MC1431-1 |
| alpha1B | human | CHO-K1 | C1432-1 | DC1432-1 | MC1432-1 | |
| alpha1D | human | CHO-K1 | C1433-1 | DC1433-1 | MC1433-1 | |
| alpha2A | human | CHO-K1 | C1434-1 | DC1434-1 | MC1434-1 | |
| alpha2A | human | CHO-K1 | C1434-1a | DC1434-1a | MC1434-1a | |
| alpha2A | human | CHO-K1 Gqi5 | CG1434-1 | DCG1434-1 | MCG1434-1 | |
| alpha2B | human | CHO-K1 | C1435-1 | DC1435-1 | MC1435-1 | |
| alpha2B | human | CHO-K1 Gqi5 | CG1435-1 | DCG1435-1 | MCG1435-1 | |
| alpha2C | human | CHO-K1 | C1436-1 | DC1436-1 | MC1436-1 | |
| alpha2C | human | CHO-K1 Gqi5 | CG1436-1 | DCG1436-1 | MCG1436-1 | |
| beta1 | human | HEK293T | H1437 | H1437 | H1437 | |
| beta1 | human | CHO-K1 | C1437-1 | DC1437-1 | MC1437-1 | |
| beta2 | human | CHO-K1 | C1438-1a | DC1438-1a | MC1438-1a | |
| beta2 | human | HEK293T β-Arrestin1 | CA1438BA1 | DCA1438BA1 | MCA1438BA1 | |
| beta2 | human | HEK293T β-Arrestin2 | CA1438BA2 | DCA1438BA2 | MCA1438BA2 | |
| beta3 | human | HEK293T | C1439a | DC1439a | MC1439a | |
| Anaphylatoxin | C3AR1 | human | HEK293T | C1222 | DC1222 | MC1222 |
| C5R1 | human | HEK293T | C1221 | DC1221 | MC1221 | |
| Angiotensin | AT1 | mouse | CHO-K1 | Cm1417-1 | DCm1417-1 | MCm1417-1 |
| AT1 | mouse | CHO-K1 | Cm1417-1a | DCm1417-1a | MCm1417-1a | |
| AT1 | human | HEK293T | H1417 | DH1417 | MH1417 | |
| AT1 | human | HEK293T | HA1417- BA1 | DHA1417- BA1 | MHA1417- BA1 | |
| AT1 | human | HEK293T | HA1417-BA2 | DHA1417-BA2 | MHA1417-BA2 | |
| Apelin | APJ | human | HEK293T | C1196a | DC1196a | MC1196a |
| APJ | human | CHO-K1 | C1196-1 | DC1196-1 | MC1196-1 | |
| APJ | human | HEK293T Gαqi5 | CG1196a | DCG1196a | MCG1196a | |
| Bile Acid | GPBA | human | CHO-K1 | C1361-1 | DC1361-1 | MC1361-1 |
| GPBA | human | CHO-K1 | C1361-1a | DC1361-1a | MC1361-1a | |
| GPBA | rat | CHO-K1 | Cr1361-1 | DCr1361-1 | MCr1361-1 | |
| GPBA | mouse | CHO-K1 | Cm1361-1 | DCm1361-1 | MCm1361-1 | |
| GPBA Mutant W83G | human | CHO-K1 | C1361-1MT1 | DC1361-1MT1 | MC1361-1MT1 | |
| GPBA Mutant W83A | human | CHO-K1 | C1361-1MT2 | DC1361-1MT2 | MC1361-1MT2 | |
| GPBA Mutant V88L | human | CHO-K1 | C1361-1MT3 | DC1361-1MT3 | MC1361-1MT3 | |
| GPBA Mutant Y89A | human | CHO-K1 | C1361-1MT4 | DC1361-1MT4 | MC1361-1MT4 | |
| GPBA Mutant Y89H | human | CHO-K1 | C1361-1MT5 | DC1361-1MT5 | MC1361-1MT5 | |
| GPBA Mutant F96A | human | CHO-K1 | C1361-1MT6 | DC1361-1MT6 | MC1361-1MT6 | |
| GPBA Mutant W237A | human | CHO-K1 | C1361-1MT7 | DC1361-1MT7 | MC1361-1MT7 | |
| GPBA Mutant W240A | human | CHO-K1 | C1361-1MT8 | DC1361-1MT8 | MC1361-1MT8 | |
| Bombesin | BB1 | human | HEK293T | C1211 | DC1211 | MC1211 |
| BB1 | rat | C6 | C1211-1 | DC1211-1 | MC1211-1 | |
| BB2 | human | HEK293T | C1215 | DC1215 | MC1215 | |
| BB3 | human | HEK293T | C1214 | DC1214 | MC1214 | |
| BB3 | human | HEK293T | H1214 | DH1214 | MH1214 | |
| Bradykinin | B1 | human | HEK293T | C1198a | DC1198a | MC1198a |
| B1 | mouse | HEK293T | Cm1198 | DCm1198 | MCm1198 | |
| B2 | human | HEK293T | H1199 | DH1199 | MH1199 | |
| B2 | mouse | HEK293T | Cm1199 | DCm1199 | MCm1199 | |
| B2 | rat | HEK293T | Cr1199 | DCr1199 | MCr1199 | |
| B2 | dog | HEK293T | cd1199 | DCd1199 | MCd1199 | |
| B2 | rhesus monkey | HEK293T | Cpr1199 | DCpr1199 | MCpr1199 | |
| B2 | guinea pig | HEK293T | Cc1199 | DCc1199 | MCc1199 | |
| B2 | rabbit | HEK293T | Cb1199 | DCb1199 | MCb1199 | |
| Calcitonin | CALCRL | human | HEK293T | C1232 | DC1232 | MC1232 |
| CALCRL | human | CHO-K1 | C1232-1 | DC1232-1 | MC1232-1 | |
| CGRP | human | CHO-K1 | C1515-1 | DC1515-1 | MC1515-1 | |
| AM1 | human | CHO-K1 | C1516-1 | DC1516-1 | MC1516-1 | |
| AM2 | human | CHO-K1 | C1517-1 | DC1517-1 | MC1517-1 | |
| CT | human | HEK293T | H1231 | DH1231 | MH1231 | |
| CT | human | CHO-K1 | C1231-1A | DC1231-1A | MC1231-1A | |
| CT | human | CHO-K1 | C1231-1B | DC1231-1B | MC1231-1B | |
| AMY1 | human | CHO-K1 | C1509-1a | DC1509-1a | MC1509-1a | |
| AMY2 | human | CHO-K1 | C1510-1a | DC1510-1a | MC1510-1a | |
| AMY2 | human | CHO-K1 | C1510-1b | DC1510-1b | MC1510-1b | |
| AMY3 | human | CHO-K1 | C1511-1a | DC1511-1a | MC1511-1a | |
| Calcium-Sensing | CaSR | human | HEK293T | C1233 | DC1233 | MC1233 |
| CaSR | rat | HEK293T | Hr1233 | DHr1233 | MHr1233 | |
| Cannabinoid | CB1 | human | HEK293T | C1229 | DC1229 | MC1229 |
| CB1 | human | CHO-K1 | C1229-1a | DC1229-1a | MC1229-1a | |
| CB1 | human | CHO-K1 | C1229-1 | DC1229-1 | MC1229-1 | |
| CB1a | human | CHO-K1 | C1512-1 | DC1512-1 | MC1512-1 | |
| CB1b | human | CHO-K1 | C1513-1 | DC1513-1 | MC1513-1 | |
| CB1 | mouse | CHO-K1 | Cm1229-1A | DCm1229-1A | MCm1229-1A | |
| CB1 | mouse | CHO-K1 | Cm1229-1B | DCm1229-1B | MCm1229-1B | |
| CB1 | dog | HEK293T | Cd1229 | DCd1229 | MCd1229 | |
| CB1 | dog | HEK293T | Cd1229a | DCd1229a | MCd1229a | |
| CB1 | dog | HEK293T | Cd1229b | DCd1229b | MCd1229b | |
| CB1 MUTANT B | human | CHO-K1 β-Arrestin2 | CA1513BA2-1 | DCA1513BA2-1 | MCA1513BA2-1 | |
| CB2 | human | CHO-K1 | C1230-1 | DC1230-1 | MC1230-1 | |
| CB2 | human | CHO-K1 | C1230-1a | DC1230-1a | MC1230-1a | |
| CB2 | human | CHO-K1 β-Arrestin2 | CA1230BA2-1 | DCA1230BA2-1 | MCA1230BA2-1 | |
| CB2 | rat | CHO-K1 | Cr1230-1 | DCr1230-1 | MCr1230-1 | |
| CB2 | rat | CHO-K1 | Cr1230-1a | DCr1230-1a | MCr1230-1a | |
| CB2 | mouse | CHO-K1 β-Arrestin2 | CAm1230BA2-1 | DCAm1230BA2-1 | MCAm1230BA2-1 | |
| CB2 | mouse | CHO-K1 | Cm1230-1 | DCm1230-1 | MCm1230-1 | |
| CB2 | mouse | CHO-K1 | Cm1230-1a | DCm1230-1a | MCm1230-1a | |
| CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1 | DCAr1230BA2-1 | MCAr1230BA2-1 | |
| CB2 | rat | CHO-K1 β-Arrestin2 | CAr1230BA2-1a | DCAr1230BA2-1a | MCAr1230BA2-1a | |
| GPR55 | human | HEK293T | H1113 | H1113 | H1113 | |
| GPR55 | human | HEK293T | C1113b | DC1113b | MC1113b | |
| GPR55 | human | HEK293T | C1113d | DC1113d | MC1113d | |
| Chemokine | CCR1 | human | HEK293T | C1009 | DC1009 | MC1009 |
| CCR1 | human | HEK293T Gαqi5 | CG1009 | DCG1009 | MCG1009 | |
| CCR2 | human | HEK293T | C1010 | DC1010 | MC1010 | |
| CCR3 | human | HEK293T | C1011 | DC1011 | MC1011 | |
| CCR3 | human | HEK293T Gαqi5 | CG1011 | DCG1011 | MCG1011 | |
| CCR4 | human | HEK293T | C1012 | DC1012 | MC1012 | |
| CCR4 | human | HEK293T Gαqi5 | CG1012 | DCG1012 | MCG1012 | |
| CCR5 | human | HEK293T | C1013a | DC1013a | MC1013a | |
| CCR5 | human | HEK293T | C1013b | DC1013b | MC1013b | |
| CCR5 | human | HEK293T Gαqi5 | CG1013 | DCG1013 | MCG1013 | |
| CCR6 | human | HEK293T | C1014a | DC1014a | MC1014a | |
| CCR6 | human | HEK293T | C1014b | DC1014b | MC1014b | |
| CCR6 | mouse | HEK293T | Cm1014 | DCm1014 | MCm1014 | |
| CCR7 | human | HEK293T | C1015 | DC1015 | MC1015 | |
| CCR7 | human | HEK293T Gαqi5 | CG1015 | DCG1015 | MCG1015 | |
| CCR8 | human | HEK293T | C1016 | DC1016 | MC1016 | |
| CCR8 | human | HEK293T | C1016a | DC1016a | MC1016a | |
| CCR8 | human | HEK293T Gαqi5 | CG1016 | DCG1016 | MCG1016 | |
| CCR9 | dog | HEK293T Gαqi5 | CGd1017 | DCGd1017 | MCGd1017 | |
| CCR9 | human | HEK293T | C1017 | DC1017 | MC1017 | |
| CCR9 | human | HEK293T | C1017a | DC1017a | MC1017a | |
| CCR9 | human | HEK293T Gαqi5 | CG1017 | DCG1017 | MCG1017 | |
| CCR9 | human | HEK293T Gαqi5 | CG1017A | DCG1017A | MCG1017A | |
| CCR9 | mouse | HEK293T | Cm1017 | DCm1017 | MCm1017 | |
| CCR9 | mouse | HEK293T Gαqi5 | CGm1017 | DCGm1017 | MCGm1017 | |
| CCR9 | rat | HEK293T Gαqi5 | CGr1017 | DCGr1017 | MCGr1017 | |
| CCR10 | human | HEK293T | C1018 | DC1018 | MC1018 | |
| CCR10 | human | CHO-K1 Gαqi5 | CG1018-1 | DCG1018-1 | MCG1018-1 | |
| CMKLR1 | human | HEK293T | C1147 | DC1147 | MC1147 | |
| CMKLR1 | human | HEK293T Gαqi5 | CG1147 | DCG1147 | MCG1147 | |
| CX3CR1 | human | HEK293T | C1008 | DC1008 | MC1008 | |
| CX3CR1 | human | HEK293T Gαqi5 | CG1008a | DCG1008a | MCG1008a | |
| CX3CR1 | human | HEK293T Gαqi5 | CG1008b | DCG1008b | MCG1008b | |
| CXCR1 | human | HEK293T | C1001a | DC1001a | MC1001a | |
| CXCR1 | human | HEK293T Gαqi5 | CG1001 | DCG1001 | MCG1001 | |
| CXCR2 | human | HEK293T | C1002 | DC1002 | MC1002 | |
| CXCR2 | human | HEK293T Gαqi5 | CG1002 | DCG1002 | MCG1002 | |
| CXCR3 | human | HEK293T | C1003 | DC1003 | MC1003 | |
| CXCR3 | human | HEK293T | C1003a | DC1003a | MC1003a | |
| CXCR3 | human | HEK293T Gαqi5 | CG1003 | DCG1003 | MCG1003 | |
| CXCR4 | human | HEK293T | C1004-1 | DC1004-1 | MC1004-1 | |
| CXCR4 | human | HEK293T Gαqi5 | CG1004 | DCG1004 | MCG1004 | |
| CXCR5 | human | HEK293T | C1005 | DC1005 | MC1005 | |
| CXCR5 | human | HEK293T | C1005a | DC1005a | MC1005a | |
| CXCR5 | human | CHO-K1 | C1005-1 | DC1005-1 | MC1005-1 | |
| CXCR5 | human | CHO-K1 | C1005-1a | DC1005-1a | MC1005-1a | |
| CXCR6 | human | HEK293T | C1006 | DC1006 | MC1006 | |
| CXCR6 | human | CHO-K1 | C1006-1 | DC1006-1 | MC1006-1 | |
| CXCR6 | human | HEK293T Gαqi5 | CG1006 | DCG1006 | MCG1006 | |
| CXCR7 | human | HEK293T | C1150 | DC1150 | MC1150 | |
| CXCR7 | human | HEK293T | CA1150BA2a | DCA1150BA2a | MCA1150BA2a | |
| XCR1 | human | HEK293T | C1007 | DC1007 | MC1007 | |
| XCR1 | human | HEK293T Gαqi5 | CG1007 | DCG1007 | MCG1007 | |
| Cholecystokinin | CCK1 | human | CHO-K1 | C1038-1a | DC1038-1a | MC1038-1a |
| CCK1 | human | HEK293T | C1038 | DC1038 | MC1038 | |
| CCK2 | human | HEK293T | H1039 | DH1039 | MH1039 | |
| Citric Acid Cycle Intermediates | GPR91 | human | CHO-K1 | C1144-1 | DC1144-1 | MC1144-1 |
| GPR91 | mouse | CHO-K1 | Cm1144-1 | DCm1144-1 | MCm1144-1 | |
| GPR91 | rat | CHO-K1 | Cr1144-1 | DCr1144-1 | MCr1144-1 | |
| GPR91 | human | CHO-K1 B-Arrestin2 | CA1141BA2-1 | DCA1141BA2-1 | MCA1141BA2-1 | |
| GPR91 | human | CHO-K1 B-Arrestin2 | CA1144BA2-1 | DCA1144BA2-1 | MCA1144BA2-1 | |
| GPR99 | human | CHO-K1 | C1132-1 | DC1132-1 | MC1132-1 | |
| Corticotrophin-Releasing Factor | CRF1 | human | HEK293T | C1040 | DC1040 | MC1040 |
| CRF1 | human | HEK293T Gαqi5 | CG1040 | DCG1040 | MCG1040 | |
| CRF2 | human | HEK293T | C1041 | DC1041 | MC1041 | |
| CRF2 | human | HEK293TGα16 | CG1041 | DCG1041 | MCG1041 | |
| Dopamine | D1 | human | HEK293T | C1335 | DC1335 | MC1335 |
| D1 | human | HEK293T | H1335 | DH1335 | MH1335 | |
| D2 | human | HEK293T | C1336 | DC1336 | MC1336 | |
| D2 | human | HEK293T | C1336a | DC1336a | MC1336a | |
| D2 | human | HEK293T | C1336b | DC1336b | MC1336b | |
| D2 Ghrelin | human | HEK293T | C1514 | DC1514 | MC1514 | |
| D3 | human | HEK293T Gqi5 | CG1337 | DCG1337 | MCG1337 | |
| D4 | human | HEK293T | C1338 | DC1338 | MC1338 | |
| D4 | human | HEK293T Gαqi5 | CG1338 | DCG1338 | MCG1338 | |
| D5 | human | HEK293T | C1339 | DC1339 | MC1339 | |
| Endothelin | ETA | human | CHO-K1 | C1216-1 | DC1216-1 | MC1216-1 |
| ETA | rat | CHO-K1 | Cr1216-1 | DCr1216-1 | MCr1216-1 | |
| ETB | human | CHO-K1 | C1217-1 | DC1217-1 | MC1217-1 | |
| Free Fatty Acid | GPR119 | human | CHO-K1 | C1298-1a | DC1298-1a | MC1298-1a |
| GPR119 | human | HEK293T | C1298 | DC1298 | MC1298 | |
| GPR119 | mouse | CHO-K1 | Cm1298-1 | DCm1298-1 | MCm1298-1 | |
| GPR120 | human | HEK293T | C1294 | DC1294 | MC1294 | |
| GPR120 | human | HEK293T Gαqi5 | CG1294 | DCG1294 | MCG1294 | |
| GPR120 | human | CHO-K1 | C1294-1 | DC1294-1 | MC1294-1 | |
| GPR120L | human | HEK293T | C1522 | DC1522 | MC1522 | |
| GPR120L | human | HEK293T β-Arrestin2 | CA1522 | DCA1522 | MCA1522 | |
| GPR120 | mouse | HEK293T Gαqi5 | CGm1294 | DCGm1294 | MCGm1294 | |
| GPR120 | rat | HEK293T | Cr1294 | DCr1294 | MCr1294 | |
| GPR40 | cynomolgus monkey | CHO-K1 | Cpc1101-1 | DCpc1101-1 | MCpc1101-1 | |
| GPR40 | cynomolgus monkey | CHO-K1 | CApr1101-1 | DCApr1101-1 | MCApr1101-1 | |
| GPR40 | cynomolgus monkey | CHO-K1 β-Arrestin2 | CApc1101-1 | DCApc1101-1 | MCApc1101-1 | |
| GPR40 | dog | CHO-K1 | Cd1101-1 | DCd1101-1 | MCd1101-1 | |
| GPR40 | human | HEK293T | C1101 | DC1101 | MC1101 | |
| GPR40 | human | CHO-K1 | C1101-1 | DC1101-1 | MC1101-1 | |
| GPR40 | human | CHO-K1 | C1101-1A | DC1101-1A | MC1101-1A | |
| GPR40 | human | CHO-K1 β-Arrestin2 | CA1101-1 | DCA1101-1 | MCA1101-1 | |
| GPR40 | mouse | HEK293T | Cm1101 | DCm1101 | MCm1101 | |
| GPR40 | rat | HEK293T | Cr1101 | DCr1101 | MCr1101 | |
| GPR40 | rat | CHO-K1 | Cr1101-1 | DCr1101-1 | MCr1101-1 | |
| GPR40 | rhesus monkey | CHO-K1 | Cpr1101-1 | DCpr1101-1 | MCpr1101-1 | |
| GPR40 | rat | CHO-K1 β-Arrestin2 | CAr1101-1 | DCAr1101-1 | MCAr1101-1 | |
| GPR41 | human | HEK293T | C1102 | DC1102 | MC1102 | |
| GPR41 | human | CHO-K1 Gα16 | C1102-1 | DCG1102-1 | MC1102-1 | |
| GPR41 | human | HEK293T Gαqi5 | CG1102 | DCG1102 | MCG1102 | |
| GPR41 | mouse | CHO-K1 Gα16 | CGm1102-1 | DCGm1102-1 | MCGm1102-1 | |
| GPR41 | rat | HEK293T | Cr1102 | DCr1102 | MCr1102 | |
| GPR43 | human | HEK293T | C1104 | DC1104 | MC1104 | |
| GPR43 | human | CHO-K1 | C1104-1 | DC1104-1 | MC1104-1 | |
| GPR43 | human | CHO-K1 Gα16 | HG1104-1 | DHG1104-1 | MHG1104-1 | |
| GPR43 | mouse | HEK293T | Cm1104 | DCm1104 | MCm1104 | |
| GPR43 | rat | HEK293T | Cr1104 | DCr1104 | MCr1104 | |
| GPR43 | dog | CHO-K1 | Cd1104-1A | DCd1104-1A | MCd1104-1A | |
| GPR43 | dog | CHO-K1 | Cd1104-1B | DCd1104-1B | MCd1104-1B | |
| GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1A | DCpc1104-1A | MCpc1104-1A | |
| GPR43 | cynomolgus monkey | CHO-K1 | Cpc1104-1B | DCpc1104-1B | MCpc1104-1B | |
| GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1A | DCpr1104-1A | MCpr1104-1A | |
| GPR43 | rhesus monkey | CHO-K1 | Cpr1104-1B | DCpr1104-1B | MCpr1104-1B | |
| GPR84 | human | CHO-K1 | C1137-1 | DC1137-1 | MC1137-1 | |
| GPR84 | human | CHO-K1 Gαqi5 | CG1137-1 | DCG1137-1 | MCG1137-1 | |
| Frizzled | SMO | human | HEK293T | C1442 | DC1442 | MC1442 |
| SMO | human | HEK293T | H1442 | DH1442 | MH1442 | |
| Galanin | GAL1 | human | CHO-K1 Gαqi5 | CG1178-1 | DCG1178-1 | MCG1178-1 |
| GAL1 | human | HEK293T | C1178 | DC1178 | MC1178 | |
| GAL2 | human | CHO-K1 | C1179-1 | DC1179-1 | MC1179-1 | |
| Ghrelin | Ghrelin | human | HEK293T | C1197b | DC1197b | MC1197b |
| Ghrelin | human | CHO-K1 | C1197-1 | DC1197-1 | MC1197-1 | |
| Ghrelin | mouse | HEK293T | Cm1197 | DCm1197 | MCm1197 | |
| Glucagon | GHRH | human | HEK293T | C1291 | DC1291 | MC1291 |
| GIP | human | HEK293T | C1290 | DC1290 | MC1290 | |
| GIP | human | HEK293T β-Arrestin2 | CA1290 | DCA1290 | MCA1290 | |
| GIP | mouse | HEK293T | Cm1290 | DCm1290 | MCm1290 | |
| GIP | rat | HEK293T | Cr1290 | DCr1290 | MCr1290 | |
| GIP | dog | HEK293T | Cd1290 | DCd1290 | MCd1290 | |
| GIP | dog | HEK293T | Cd1290a | DCd1290a | MCd1290a | |
| GIP | rabbit | HEK293T | Cb1290 | DCb1290 | MCb1290 | |
| GIP | pig | HEK293T | Cp1290 | DCp1290 | MCp1290 | |
| GIP | rhesus monkey | HEK293T | Cpr1290 | DCpr1290 | MCpr1290 | |
| GIP | rhesus monkey | HEK293T | Cpr1290a | DCpr1290a | MCpr1290a | |
| GIP | ferret | HEK293T | Cf1290 | DCf1290 | MCf1290 | |
| GIP | ferret | HEK293T | Cf1290a | DCf1290a | MCf1290a | |
| GLP-1 | human | HEK293T | C1267 | DC1267 | MC1267 | |
| GLP-1 | human | CHO-K1 | C1267-1 | DC1267-1 | MC1267-1 | |
| GLP-1 | human | CHO-K1 | C1267-1a | DC1267-1a | MC1267-1a | |
| GLP-1 | human | CHO-K1 β-Arrestin2 | CA1267-1 | DCA1267-1 | MCA1267-1 | |
| GLP-1 | human | HEK293T β-Arrestin2 | CA1267BA2 | DCA1267BA2 | MCA1267BA2 | |
| GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1 | DCpc1267-1 | MCpc1267-1 | |
| GLP-1 | cynomolgus monkey | CHO-K1 | Cpc1267-1a | DCpc1267-1a | MCpc1267-1a | |
| GLP-1 | rat | CHO-K1 | Cr1267-1 | DCr1267-1 | MCr1267-1 | |
| GLP-1 | dog | CHO-K1 | Cd1267-1 | DCd1267-1 | MCd1267-1 | |
| GLP-1 | dog | HEK293T | Cd1267-1a | DCd1267-1a | MCd1267-1a | |
| GLP-1 | dog | HEK293T | Cd1267-1b | DCd1267-1b | MCd1267-1b | |
| GLP-1 | mouse | CHO-K1 | Cm1267-1 | DCm1267-1 | MCm1267-1 | |
| GLP-1 | mouse | CHO-K1 | Cm1267-1a | DCm1267-1a | MCm1267-1a | |
| GLP-1 | pig | CHO-K1 | Cp1267-1 | DCp1267-1 | MCp1267-1 | |
| GLP-1 | rabbit | CHO-K1 | Cb1267-1 | DCb1267-1 | MCb1267-1 | |
| GLP-1 | rabbit | CHO-K1 | Cb1267-1a | DCb1267-1a | MCb1267-1a | |
| GLP-2 | human | HEK293T | C1268 | DC1268 | MC1268 | |
| GLP-2 | rat | HEK293T | Cr1268 | DCr1268 | MCr1268 | |
| Glucagon | human | HEK293T | C1266 | DC1266 | MC1266 | |
| Glucagon | dog | HEK293T | Cd1266 | DCd1266 | MCd1266 | |
| Glucagon | pig | HEK293T | Cp1266 | DCp1266 | MCp1266 | |
| Glucagon | rat | HEK293T | Cr1266 | DCr1266 | MCr1266 | |
| Glucagon | human | HEK293T | C1266A | DC1266A | MC1266A | |
| Glucagon | human | CHO-K1 | C1266-1 | DC1266-1 | MC1266-1 | |
| Glucagon | human | CHO-K1 | C1266-1a | DC1266-1a | MC1266-1a | |
| Glucagon | human | CHO-K1 β-Arrestin2 | CA1266-1 | DCA1266-1 | MCA1266-1 | |
| Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1 | DCpc1266-1 | MCpc1266-1 | |
| Glucagon | cynomolgus monkey | CHO-K1 | Cpc1266-1a | DCpc1266-1a | MCpc1266-1a | |
| Glucagon | cynomolgus monkey | HEK293T | Cpc1266 | DCpc1266 | MCpc1266 | |
| Glucagon | cynomolgus monkey | HEK293T | Cpc1266a | DCpc1266a | MCpc1266a | |
| Secretin | human | CHO-K1 | C1228-1 | DC1228-1 | MC1228-1 | |
| Glycoprotein Hormone | TSH | human | HEK293T | H1177 | DH1177 | MH1177 |
| TSH | rat | HEK293T | C1177-1 | DC1177-1 | MC1177-1 | |
| Gonadotrophin-Releasing Hormone | GnRH | human | HEK293T | C1283 | DC1283 | MC1283 |
| GnRH | dog | HEK293T | Cd1283 | DCd1283 | MCd1283 | |
| FSHR | human | HEK293T | C1175 | DC1175 | MC1175 | |
| Histamine | H1 | human | HEK293T | C1027 | DC1027 | MC1027 |
| H1 | mouse | HEK293T | Cm1027 | DCm1027 | MCm1027 | |
| H2 | human | HEK293T | C1028 | DC1028 | MC1028 | |
| H3 | human | HEK293T | C1029 | DC1029 | MC1029 | |
| H3 | human | HEK293T Gαqi5 | CG1029 | DCG1029 | MCG1029 | |
| H3 | mouse | HEK293T | Cm1029 | DCm1029 | MCm1029 | |
| H3 | mouse | CHO-K1 | Cm1029-1 | DCm1029-1 | MCm1029-1 | |
| H4 | human | HEK293T | C1030 | DC1030 | MC1030 | |
| H4 | human | HEK293T Gαqi5 | CG1030 | DCG1030 | MCG1030 | |
| H4 | human | HEK293T β-Arrestin2 | CA1030BA2 | DCA1030BA2 | MCA1030BA2 | |
| H4 | mouse | HEK293T | Cm1030 | DCm1030 | MCm1030 | |
| H4 | mouse | HEK293T Gαqi5 | CGm1030 | DCGm1030 | MCGm1030 | |
| Hydroxycarboxylic acid | GPR81 | human | HEK293T | |||
| KiSS1-Derived Peptide | KiSS1 | human | CHO dhfr- | C1036 | DC1036 | MC1036 |
| KiSS1 | rat | CHO dhfr- | C1036-1 | DC1036-1 | MC1036-1 | |
| Leukotriene/Lipoxin | BLT1 | human | HEK293T | H1165a | DH1165a | H1165a |
| BLT2 | human | HEK293T | C1272 | DC1272 | MC1272 | |
| BLT2 | human | HEK293T | C1272A | DC1272A | MC1272A | |
| BLT2 | human | HEK293T | C1272b | DC1272b | MC1272b | |
| BLT2 | human | HEK293T | C1272c | DC1272c | MC1272c | |
| BLT2 | monkey | HEK293T | Cp1272a | DCp1272a | MCp1272a | |
| BLT2 | monkey | HEK293T | Cp1272 | DCp1272 | MCp1272 | |
| BLT2 | mouse | HEK293T | Cm1272a | DCm1272a | MCm1272a | |
| BLT2 | mouse | HEK293T | Cm1272 | DCm1272 | MCm1272 | |
| CysLT1 | human | HEK293T | C1308 | DC1308 | MC1308 | |
| CysLT2 | human | HEK293T | C1307 | DC1307 | MC1307 | |
| OXE | human | HEK293T | ||||
| Lysophospholipid | GPR87 | human | RH7777 | C1140-6 | DC1140-6 | MC1140-6 |
| LPA1 | human | RH7777 | C1048-6 | DC1048-6 | MC1048-6 | |
| LPA1 | mouse | RH7777 | Cm1048-6A | DCm1048-6A | MCm1048-6A | |
| LPA1 | mouse | RH7777 | Cm1048-6B | DCm1048-6B | MCm1048-6B | |
| LPA1 | rat | RH7777 | Cr1048-6B | DCr1048-6B | MCr1048-6B | |
| LPA2 | human | RH7777 | C1050-6 | DC1050-6 | MC1050-6 | |
| LPA3 | human | RH7777 | C1053-6 | DC1053-6 | MC1053-6 | |
| LPA3 | human | RH7777 | C1053-6a | DC1053-6a | MC1053-6a | |
| LPA4 | human | CHO-K1 | C1087-1a | DC1087-1a | MC1087-1a | |
| LPA4 | human | CHO-K1 | C1087-1b | DC1087-1b | MC1087-1b | |
| LPA5 | human | RH7777 | C1145-6 | DC1145-6 | MC1145-6 | |
| LPA5 | mouse | RH7777 | Cm1145-6 | DCm1145-6 | MCm1145-6 | |
| S1P1 | human | CHO-K1 | C1047-1 | DC1047-1 | MC1047-1 | |
| S1P1 | human | CHO-K1 Gαqi5 | CG1047-1 | DCG1047-1 | MCG1047-1 | |
| S1P2 | human | CHO-K1 | C1051-1 | DC1051-1 | MC1051-1 | |
| S1P2 | human | CHO-K1 Gαqi5 | CG1051-1 | DCG1051-1 | MCG1051-1 | |
| S1P2 | mouse | CHO-K1 | Cm1051-1 | DCm1051-1 | MCm1051-1 | |
| S1P2 | rat | CHO-K1 | Cr1051-1 | DCr1051-1 | MCr1051-1 | |
| S1P3 | human | RH7777 | C1049-6 | DC1049-6 | MC1049-6 | |
| S1P3 | human | CHO-K1 | C1049-1 | DC1049-1 | MC1049-1 | |
| S1P3 | human | CHO-K1 Gαqi5 | CG1049-1 | DCG1049-1 | MCG1049-1 | |
| S1P3 | mouse | CHO-K1 Gαqi5 | CGm1049-1 | DCGm1049-1 | MCGm1049-1 | |
| S1P3 | rat | CHO-K1 Gαqi5 | CGr1049-1 | DCGr1049-1 | MCGr1049-1 | |
| S1P4 | human | CHO-K1 Gαqi5 | CG1052-1 | DCG1052-1 | MCG1052-1 | |
| S1P4 | mouse | CHO-K1 Gαqi5 | CGm1052-1 | DCGm1052-1 | MCGm1052-1 | |
| S1P4 | rat | CHO-K1 Gαqi5 | CGr1052-1 | DCGr1052-1 | MCGr1052-1 | |
| S1P5 | human | CHO-K1 | C1054-1 | DC1054-1 | MC1054-1 | |
| S1P5 | human | CHO-K1 Gαqi5 | CG1054-1 | DCG1054-1 | MCG1054-1 | |
| Melanin-Concentrating Hormone | MCH1 | human | HEK293T Gαqi5 | C1031-3 | DC1031-3 | MC1031-3 |
| MCH1 | rat | HEK293T Gαqi5 | C1031-4 | DC1031-4 | MC1031-4 | |
| MCH2 | human | CHO dhfr- | C1032 | DC1032 | MC1032 | |
| Melanocortin | MC1 | human | HEK293T | C1340 | DC1340 | MC1340 |
| MC4 | human | HEK293T | H1343 | H1343 | H1343 | |
| Melatonin | MT1 | human | CHO-K1 | C1223-1 | DC1223-1 | MC1223-1 |
| MT2 | human | HEK293T Gαqi5 | C1224 | DC1224 | MC1224 | |
| MT2 | mouse | HEK293T | Cm1224 | DCm1224 | MCm1224 | |
| MT2 | rat | HEK293T | Cr1224 | DCr1224 | MCr1224 | |
| Metabotropic Glutamate | mGlu1 | human | CHO-K1 | C1188-1 | DC1188-1 | MC1188-1 |
| mGlu2 | human | HEK293T | C1189a | DC1189a | MC1189a | |
| mGlu2 | human | HEK293T Gqi5 | HG1189Gi | DHG1189Gi | MHG1189Gi | |
| mGlu2 | human | HEK293T Gαqi5 | HG1189 | HG1189 | HG1189 | |
| mGlu2 | human | HEK293T Gαqi5 | HG1189a | HG1189a | HG1189a | |
| mGlu2 | rat | HEK293T Gαqi5 | HGr1189b | DHGr1189b | MHGr1189b | |
| mGlu3 | human | HEK293T Gαqi5 | CG1190 | DCG1190 | MCG1190 | |
| mGlu4 | dog | CHO-K1 Gαqi5 | HGd1191-1 | DHGd1191-1 | MHGd1191-1 | |
| mGlu4 | human | HEK293T | C1191a | DC1191a | MC1191a | |
| mGlu4 | human | HEK293T Gαqi5 | CG1191 | DCG1191 | MCG1191 | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1a | DHGm1191-1a | MHGm1191-1a | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1b | DHGm1191-1b | MHGm1191-1b | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1c | DHGm1191-1c | MHGm1191-1c | |
| mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1d | DHGm1191-1d | MHGm1191-1d | |
| mGlu4 | rat | HEK293T | Cr1191 | DCr1191 | MCr1191 | |
| mGlu4 | human | HEK293T Gαqi5 | CG1191a | DCG1191a | MCG1191a | |
| mGlu5 | human | HEK293T | C1192 | DC1192 | MC1192 | |
| mGlu5 | human | HEK293T B-ARRESTIN2 | CA1192BA2 | DCA1192BA2 | MCA1192BA2 | |
| mGlu6 | human | HEK293T | C1193 | DC1193 | MC1193 | |
| mGlu6 | human | HEK293T Gαqi5 | CG1193 | DCG1193 | MCG1193 | |
| mGlu7 | human | HEK293T | C1194 | DC1194 | MC1194 | |
| mGlu7 | human | HEK293T Gαqi5 | CG1194 | DCG1194 | MCG1194 | |
| mGlu8 | human | HEK293T | C1195 | DC1195 | MC1195 | |
| mGlu8 | human | HEK293T | C1195a | DC1195a | MC1195a | |
| mGlu8 | human | HEK293T Gαqi5 | CG1195 | DCG1195 | MCG1195 | |
| mGlu8 | human | CHO-K1 | C1195-1a | DC1195-1a | MC1195-1a | |
| Motilin | motilin | human | HEK293T | H1297 | H1297 | H1297 |
| Muscarinic | M1 | human | CHO-K1 | C1022-1 | DC1022-1 | MC1022-1 |
| M1 | human | CHO-K1 | C1022-1a | DC1022-1a | MC1022-1a | |
| M2 | human | CHO-K1 | C1023-1 | DC1023-1 | MC1023-1 | |
| M3 | human | CHO-K1 | C1024-1 | DC1024-1 | MC1024-1 | |
| M3 | mouse | CHO-K1 | Cm1024-1 | DCm1024-1 | MCm1024-1 | |
| M4 | human | CHO-K1 | C1025-1 | DC1025-1 | MC1025-1 | |
| M4 | human | CHO-K1 Gαqi5 | CG1025-1 | DCG1025-1 | MCG1025-1 | |
| M4 | mouse | CHO-K1 | Cm1025-1 | DCm1025-1 | MCm1025-1 | |
| M5 | human | CHO-K1 | C1026-1 | DC1026-1 | MC1026-1 | |
| N-formylpeptide | FPR1 | human | HEK293T | C1243 | DC1243 | MC1243 |
| FPR1 | human | HEK293T | C1243a | DC1243a | MC1243a | |
| FPR1 | human | HEK293T Gαqi5 | CG1243 | DCG1243 | MCG1243 | |
| FPR2 | human | HEK293T | C1244 | DC1244 | MC1244 | |
| FPR2 | human | HEK293T | C1244a | DC1244a | MC1244a | |
| FPR3 | human | HEK293T | C1245 | DC1245 | MC1245 | |
| Neuromedin U | NMU1 | human | HEK293T | C1122 | DC1122 | MC1122 |
| NMU2 | human | HEK293T | C1213 | DC1213 | MC1213 | |
| Neuropeptide FF/AF | NPFF1 | human | HEK293T | C1363 | DC1363 | MC1363 |
| NPFF2 | human | HEK293T Gαqi5 | CG1364 | DCG1364 | MCG1364 | |
| Neuropeptide S | NPS | mouse | HEK293T | C1355-1 | DC1355-1 | MC1355-1 |
| NPS | human | HEK293T | C1355a | DC1355a | MC1355a | |
| NPS(2) | human | HEK293T | C1356 | DC1356 | MC1356 | |
| NPSIle107 | human | HEK293T | C1355-2 | DC1355-2 | MC1355-2 | |
| Neuropeptide W/B | NPBW1 | rat | HEK293T Gαqi5 | C1124-1 | DC1124-1 | MC1124-1 |
| NPBW1 | human | HEK293T Gαqi5 | C1124 | DC1124 | MC1124 | |
| NPBW2 | human | HEK293T Gαqi5 | C1133 | DC1133 | MC1133 | |
| Neuropeptide Y | Y1 | human | CHO-K1 Gαqi5 | CG1273-1 | DCG1273-1 | MCG1273-1 |
| Y2 | human | CHO-K1 Gαqi5 | CG1274-1 | DCG1274-1 | MCG1274-1 | |
| Y2 | rat | CHO-K1 | Cr1274-1 | DCr1274-1 | MCr1274-1 | |
| Y4 | human | CHO-K1 | C1300-1 | DC1300-1 | MC1300-1 | |
| Y4 | human | CHO-K1 Gαqi5 | CG1300-1 | DCG1300-1 | MCG1300-1 | |
| Y5 | human | HEK293T | C1275a | DC1275a | MC1275a | |
| Y5 | human | HEK293T Gαqi5 | CG1275 | DCG1275 | MCG1275 | |
| Neurotensin | NTS1 | human | CHO-K1 | C1276-1 | DC1276-1 | MC1276-1 |
| NTS2 | human | CHO-K1 | C1277-1 | DC1277-1 | MC1277-1 | |
| NTS2 | human | HEK293T | C1277 | DC1277 | MC1277 | |
| NTS2 | human | HEK293T | C1277a | DC1277a | MC1277a | |
| Nicotinic Acid | GPR109A | human | CHO-K1 | C1370-1 | DC1370-1 | MC1370-1 |
| GPR109B | human | CHO-K1 | C1059-1 | DC1059-1 | MC1059-1 | |
| GPR81 | human | HEK293T | C1134 | DC1134 | MC1134 | |
| Opioid | delta | human | CHO-K1 | C1351-1 | DC1351-1 | MC1351-1 |
| delta | human | CHO-K1 Gαqi5 | CG1351-1 | DCG1351-1 | MCG1351-1 | |
| delta | human | CHO-K1 | CA1351-1 | DCA1351-1 | MCA1351-1 | |
| delta | rat | CHO dhfr- | C1351 | DC1351 | MC1351 | |
| kappa | human | CHO-K1 | C1352-1a | DC1352-1a | MC1352-1a | |
| kappa | human | CHO-K1 Gαqi5 | CG1352-1 | DCG1352-1 | MCG1352-1 | |
| kappa | human | CHO-K1 | CA1352-1a | DCA1352-1a | MCA1352-1a | |
| kappa | human | CHO-K1 β-Arrestin2 | CA1352BA2-1 | DCA1352BA2-1 | MCA1352BA2-1 | |
| kappa | human | HEK293T | C1352 | DC1352 | MC1352 | |
| kappa | rat | CHO dhfr- | C1352-1 | DC1352-1 | MC1352-1 | |
| kappa | rat | CHO dhfr- | Cr1352-8 | DCr1352-8 | MCr1352-8 | |
| mu | human | CHO-K1 | C1350-1a | DC1350-1a | MC1350-1a | |
| mu | human | CHO-K1 Gαqi5 | CG1350-1a | DCG1350-1a | MCG1350-1a | |
| mu | human | CHO-K1 | CA1350-1a | DCA1350-1a | MCA1350-1a | |
| mu | rat | CHO dhfr- | Cr1350-1a | DCr1350-1a | MCr1350-1a | |
| mu Mutant Y150F | human | CHO-K1 | C1350-1MT1 | DC1350-1MT1 | MC1350-1MT1 | |
| mu Mutant Y150A | human | CHO-K1 | C1350-1MT2 | DC1350-1MT2 | MC1350-1MT2 | |
| mu Mutant M153A | human | CHO-K1 | C1350-1MT3 | DC1350-1MT3 | MC1350-1MT3 | |
| mu Mutant H299N | human | CHO-K1 | C1350-1MT4 | DC1350-1MT4 | MC1350-1MT4 | |
| mu Mutant H299A | human | CHO-K1 | C1350-1MT5 | DC1350-1MT5 | MC1350-1MT5 | |
| NOP | human | CHO-K1 | C1354-1 | DC1354-1 | MC1354-1 | |
| NOP | human | CHO-K1 Gαqi5 | CG1354-1 | DCG1354-1 | MCG1354-1 | |
| NOP | human | CHO-K1 β-Arrestin2 | CA1354-1 | DCA1354-1 | MCA1354-1 | |
| NOP | human | HEK293T | C1354a | DC1354a | MC1354a | |
| NOP | rat | CHO dhfr- | Cr1354 | DCr1354 | MCr1354 | |
| Orexin | OX1 | human | CHO-K1 | C1033-1 | DC1033-1 | MC1033-1 |
| OX2 | human | CHO-K1 | C1034-1 | DC1034-1 | MC1034-1 | |
| Orphan | GPR3 | human | HEK293T | C1091 | DC1091 | MC1091 |
| GPR6 | human | HEK293T | C1116 | DC1116 | MC1116 | |
| GPR6 | human | HEK293T | C1116a | DC1116a | MC1116a | |
| GPR15 | human | HEK293T | C1069 | DC1069 | MC1069 | |
| GPR34 | human | HEK293T Gαqi5 | CG1095 | DCG1095 | MCG1095 | |
| GPR35 | dog | HEK293T Gα16 | CGd1096 | DCGd1096 | MCGd1096 | |
| GPR35 | dog | CHO-K1 Gα16 | CGd1096-1 | DCGd1096-1 | MCGd1096-1 | |
| GPR35 | mouse | CHO-K1 | Cm1096-1 | DCm1096-1 | MCm1096-1 | |
| GPR35 | mouse | CHO-K1 Gα16 | CGm1096-1 | DCGm1096-1 | MCGm1096-1 | |
| GPR35 (short form) | human | CHO-K1 | C1096-1 | DC1096-1 | MC1096-1 | |
| GPR35 (short form) | human | CHO-K1 β-Arrestin2 | CA1096-1 | DCA1096-1 | MCA1096-1 | |
| GPR35 (short form) | human | CHO-K1 Gα16 | CG1096-1 | DCG1096-1 | MCG1096-1 | |
| GPR35 (short form) | human | HEK293T Gα16 | CG1096 | DCG1096 | MCG1096 | |
| GPR35 (long form) | human | CHO-K1 β-Arrestin2 | CA1523-1 | DCA1523-1 | MCA1523-1 | |
| GPR35 (long form) T108M Mutant | human | CHO-K1 β-Arrestin2 | CA1524-1 | DCA1524-1 | MCA1524-1 | |
| GPR37L1 | human | HEK293T | C1098 | DC1098 | MC1098 | |
| GPR45 | human | CHO-K1 | CG1106-1 | DCG1106-1 | MCG1106-1 | |
| GPR45 | human | CHO-K1 | CG1106-1a | DCG1106-1a | MCG1106-1a | |
| GPR50 | human | HEK293T | C1110 | DC1110 | MC1110 | |
| GPR52 | human | HEK293T | C1112 | DC1112 | MC1112 | |
| GPR52 | human | HEK293T | C1112a | DC1112a | MC1112a | |
| GPR52 | human | HEK293T β-Arrestin2 | CA1112BA2 | DCA1112BA2 | MCA1112BA2 | |
| GPR61 | human | HEK293T | C1117 | DC1117 | MC1117 | |
| GPR61 | human | HEK293T | C1117a | DC1117a | MC1117a | |
| GPR61 | human | HEK293T | C1117b | DC1117b | MC1117b | |
| GPR75 | human | HEK293T | C1129 | DC1129 | MC1129 | |
| GPR85 | human | HEK293T | C1138 | DC1138 | MC1138 | |
| GPR85 | human | CHO-K1 | C1138-1 | DC1138-1 | MC1138-1 | |
| GPR88 | human | CHO-K1 | C1141-1 | DC1141-1 | MC1141-1 | |
| GPR88 | rat | CHO-K1 | Cr1141-1 | DCr1141-1 | MCr1141-1 | |
| GPR142 | human | HEK293T | C1286 | DC1286 | MC1286 | |
| GPR142 | human | HEK293T | C1286a | DC1286a | MC1286a | |
| GPR151 | human | CHO-K1 Gα16 Gαqi5 | CG1181-1 | DCG1181-1 | MCG1181-1 | |
| GPRC5A | human | HEK293T | CA1525 | DCA1525 | MCA1525 | |
| MRGX1 | human | CHO dhfr-Gαqi5 | C1256 | DC1256 | MC1256 | |
| MRGX1 | human | HEK293T | C1256a | DC1256a | MC1256a | |
| MRGX2 | human | HEK293T Gαqi5 | C1257 | DC1257 | MC1257 | |
| MRGX2 | human | HEK293T | C1257a | DC1257a | MC1257a | |
| MRGX2 | human | HEK293T | C1257b | DC1257b | MC1257b | |
| MRGX2 | rhesus monkey | CHO-K1 | Cpr1257-1 | DCpr1257-1 | MCpr1257-1 | |
| MRGX2 | human | HEK293T β-Arrestin2 | CA1257aBA2 | DCA1257aBA2 | MCA1257aBA2 | |
| MRGX2 | human | HEK293T β-Arrestin2 | CA1257bBA2 | DCA1257bBA2 | MCA1257bBA2 | |
| MRGX4 | human | HEK293T | C1259 | DC1259 | MC1259 | |
| MAS1 | human | HEK293T | C1225 | DC1225 | MC1225 | |
| Oxysterol | EBI2 | human | CHO-K1 Gαqi5 | CG1242-1 | DCG1242-1 | MCG1242-1 |
| EBI2 | mouse | CHO-K1 Gαqi5 | CGm1242-1 | DCGm1242-1 | MCGm1242-1 | |
| EBI2 | mouse | CHO-K1 | Cm1242-1 | DCm1242-1 | MCm1242-1 | |
| Parathyroid Hormone | PTH1 | human | HEK293T | C1301 | DC1301 | MC1301 |
| PTH1 | human | HEK293T | C1301-1 | DC1301-1 | MC1301-1 | |
| PTH2 | human | HEK293T | H1302 | DH1302 | H1302 | |
| Platelet-Activating Factor | PAF | human | HEK293T | C1218 | DC1218 | MC1218 |
| Prokineticin | PK1 | human | CHO-K1 | C1128-1 | DC1128-1 | MC1128-1 |
| PK2 | human | CHO-K1 | C1127-1 | DC1127-1 | MC1127-1 | |
| PK2 | human | CHO-K1 | C1127-1a | DC1127-1a | MC1127-1a | |
| PK2 mutant | human | CHO-K1 | C1127CT-1 | DC1127DCT-1 | MC1127MCT-1 | |
| Prolactin-Releasing Peptide | PrRP | human | CHO dhfr- | C1037 | DC1037 | MC1037 |
| Prostanoid | DP1 | human | HEK293T | C1200 | DC1200 | MC1200 |
| DP2 | human | HEK293T | H1105 | DH1105 | MH1105 | |
| DP2 | human | HEK293T | H1105a | DH1105a | MH1105a | |
| EP1 | human | HEK293T | C1201a | DC1201a | MC1201a | |
| EP2 | human | HEK293T | C1202 | DC1202 | MC1202 | |
| EP2 | mouse | HEK293T | Cm1202 | DCm1202 | MCm1202 | |
| EP2 | mouse | HEK293T | Cm1202-3 | DCm1202-3 | MCm1202-3 | |
| EP2 | rat | HEK293T | Cr1202 | DCr1202 | MCr1202 | |
| EP2 | rat | HEK293T | Cr1202-134 | DCr1202-134 | MCr1202-134 | |
| EP3 | human | CHO-K1 | C1203-1 | DC1203-1 | MC1203-1 | |
| EP3 | human | CHO-K1 | C1203-1a | DC1203-1a | MC1203-1a | |
| EP3 | human | CHO-K1 | C1203-1b | DC1203-1b | MC1203-1b | |
| EP3 | human | CHO-K1 | C1203-1c | DC1203-1DC | MC1203-1MC | |
| EP3 | human | CHO-K1 | C1203-1d | DC1203-1d | MC1203-1d | |
| EP4 | human | HEK293T | C1204 | DC1204 | MC1204 | |
| FP | human | HEK293T | C1205 | DC1205 | MC1205 | |
| IP1 | human | CHO-K1 | C1206-1 | DC1206-1 | MC1206-1 | |
| TP | human | HEK293T | C1365 | DC1365 | MC1365 | |
| TP | human | HEK293T | H1365 | H1365 | H1365 | |
| Protease-Activated | PAR1 | human | CHO-K1 | C1207-1 | DC1207-1 | MC1207-1 |
| PAR1 | human | HeLa | C1207-7 | DC1207-7 | MC1207-7 | |
| PAR2 | human | HeLa | C1208-7 | DC1208-7 | MC1208-7 | |
| PAR4 | human | HeLa | C1210-7 | DC1210-7 | MC1210-7 | |
| Proton-Sensing Receptors | GPR4 | human | HEK293T | C1100 | DC1100 | MC1100 |
| GPR4 | human | HEK293T | CA1100 | DCA1100 | MCA1100 | |
| GPR65 | human | HEK293T | C1121 | DC1121 | MC1121 | |
| GPR65 | human | HEK293T | CA1121 | DCA1121 | MCA1121 | |
| GPR65 | human | HEK293T | C1121a | DC1121a | MC1121a | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP20 | DC1121-CSP20 | MC1121-CSP20 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP23 | DC1121-CSP23 | MC1121-CSP23 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP30 | DC1121-CSP30 | MC1121-CSP30 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP36 | DC1121-CSP36 | MC1121-CSP36 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP38 | DC1121-CSP38 | MC1121-CSP38 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP44 | DC1121-CSP44 | MC1121-CSP44 | |
| GPR65 | human | Mia-Pa-Ca-2 | C1121-CSP75 | DC1121-CSP75 | MC1121-CSP75 | |
| GPR68 | human | HEK293T | C1123 | DC1123 | MC1123 | |
| GPR68 | human | HEK293T | CA1123 | DCA1123 | MCA1123 | |
| GPR132 | human | HEK293T | CA1066 | DCA1066 | MCA1066 | |
| Purinergic | GPR17 (short form) | human | 1321N1 | C1526-3 | DC1526-3 | MC1526-3 |
| GPR17 | mouse | 1321N1 | Cm1526-3 | DCm1526-3 | MCm1526-3 | |
| GPR17 | rat | 1321N1 | Cr1526-3 | DCr1526-3 | MCr1526-3 | |
| GPR17 | rat | 1321N1 | Cr1525-3 | DCr1525-3 | MCr1525-3 | |
| P2Y1 | human | 1321N1 | C1160-3 | DC1160-3 | MC1160-3 | |
| P2Y2 | human | 1321N1 | C1161-3 | DC1161-3 | MC1161-3 | |
| P2Y2 | human | HEK293T | C1161 | DC1161 | MC1161 | |
| P2Y2 | rat | 1321N1 | Cr1161-3 | DCr1161-3 | MCr1161-3 | |
| P2Y4 | human | 1321N1 | C1162-3 | DC1162-3 | MC1162-3 | |
| P2Y6 | human | 1321N1 | C1164-3 | DC1164-3 | MC1164-3 | |
| P2Y11 | human | 1321N1 | C1169-3 | DC1169-3 | MC1169-3 | |
| P2Y12 | human | 1321N1 | C1170-3 | DC1170-3 | MC1170-3 | |
| P2Y12 | human | 1321N1 | C1170-3a | DC1170-3a | MC1170-3a | |
| P2Y12 | rat | CHO dhfr- | C1170-1 | DC1170-1 | MC1170-1 | |
| P2Y13 | human | 1321N1 | C1139-3 | DC1139-3 | MC1139-3 | |
| P2Y14 | human | HEK293T | C1057 | DC1057 | MC1057 | |
| P2Y14 | human | HEK293T Gαqi5 | CG1057 | DCG1057 | MCG1057 | |
| P2Y14 | rat | HEK293T Gαqi5 | CGr1057 | DCGr1057 | MCGr1057 | |
| P2Y14 | monkey | HEK293T Gαqi5 | CGp1057 | DCGp1057 | MCGp1057 | |
| Relaxin | RXFP1 | human | HEK293T | C1287 | DC1287 | MC1287 |
| RXFP1 | human | HEK293T | C1287NTa | DC1287NTa | MC1287NTa | |
| RXFP1 | human | HEK293T | C1287NTb | DC1287NTb | MC1287NTb | |
| RXFP2 | human | HEK293T | C1289NTa | DC1289NTa | MC1289NTa | |
| RXFP2 | human | HEK293T | C1289NTb | DC1289NTb | MC1289NTb | |
| RXFP3 | human | HEK293T | C1306 | DC1306 | MC1306 | |
| SARS-CoV-2 | ACE2 | human | HEK293T | C2006 | DC2006 | MC2006 |
| TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 | |
| Serotonin | 5-HT1A | human | HEK293T | C1319 | DC1319 | MC1319 |
| 5-HT1A | human | HEK293T | C1319a | DC1319a | MC1319a | |
| 5-HT1B | human | HEK293T | C1320 | DC1320 | MC1320 | |
| 5-HT1B | human | HEK293T | C1320a | DC1320a | MC1320a | |
| 5-HT1B | human | HEK293T Gαqi5 | CG1320 | DCG1320 | MCG1320 | |
| 5-HT2A | human | HEK293T | C1324 | DC1324 | MC1324 | |
| 5-HT2A | human | CHO-K1 | C1324-1 | DC1324-1 | MC1324-1 | |
| 5-HT2A | mouse | HEK293T | Cm1324 | DCm1324 | MCm1324 | |
| 5-HT2A | mouse | CHO-K1 | Cm1324-1 | DCm1324-1 | MCm1324-1 | |
| 5-HT2A | dog | HEK293T | Cd1324 | DCd1324 | MCd1324 | |
| 5-HT2B | human | CHO-K1 | C1325-1 | DC1325-1 | MC1325-1 | |
| 5-HT2B | human | HEK293T | C1325 | DC1325 | MC1325 | |
| 5-HT2B | mouse | HEK293T | Cm1325 | DCm1325 | MCm1325 | |
| 5-HT2C | human | CHO-K1 | C1326-1 | DC1326-1 | MC1326-1 | |
| 5-HT4A | human | CHO-K1 | C1518-1 | DC1518-1 | MC1518-1 | |
| 5-HT4A | mouse | CHO-K1 | Cm1518-1 | DCm1518-1 | MCm1518-1 | |
| 5-HT4B | human | CHO-K1 | C1330-1 | DC1330-1 | MC1330-1 | |
| 5-HT4B | human | HEK293T | C1330 | DC1330 | MC1330 | |
| 5-HT4D | human | CHO-K1 | C1520-1 | DC1520-1 | MC1520-1 | |
| 5-HT6 | human | CHO-K1 | C1331-1 | DC1331-1 | MC1331-1 | |
| 5-HT7 | human | HEK293T | C1334 | DC1334 | MC1334 | |
| Somatostatin | sst1 | human | CHO-K1 | C1345-1a | DC1345-1a | MC1345-1a |
| sst1 | human | CHO-K1 Gα16 | CG1345-1 | DCG1345-1 | MCG1345-1 | |
| sst2 | human | CHO-K1 | C1346-1 | DC1346-1 | MC1346-1 | |
| sst2 | human | CHO-K1 Gα16 | CG1346-1 | DCG1346-1 | MCG1346-1 | |
| sst3 | human | CHO-K1 | C1347-1 | DC1347-1 | MC1347-1 | |
| sst3 | human | CHO-K1 Gα16 | CG1347-1 | DCG1347-1 | MCG1347-1 | |
| sst4 | human | CHO-K1 | C1348-1a | DC1348-1a | MC1348-1a | |
| sst4 | human | CHO-K1 Gα16 | CG1348-1 | DCG1348-1 | MCG1348-1 | |
| sst5 | human | CHO-K1 | C1349-1 | DC1349-1 | MC1349-1 | |
| sst5 | human | CHO-K1 Gα16 | CG1349-1 | DCG1349-1 | MCG1349-1 | |
| Tachykinin | NK1 | human | HEK293T | C1303 | DC1303 | MC1303 |
| NK2 | human | HEK293T | C1304 | DC1304 | MC1304 | |
| NK3 | human | HEK293T | C1305 | DC1305 | MC1305 | |
| NK3 | rat | HEK293T | Cr1305 | DCr1305 | MCr1305 | |
| NK3 | mouse | HEK293T | Cm1305 | DCm1305 | MCm1305 | |
| Thyrotropin-Releasing Hormone | TRH | human | HEK293T | |||
| Trace Amine | TA1 | rat | HEK293T | C1357 | DC1357 | MC1357 |
| TA1 | human | HEK293T | C1357a | DC1357a | MC1357a | |
| TA1 | rat | HEK293T Gαqi5 | Cr1357 | DCr1357 | MCr1357 | |
| Urotensin | UT | rat | CHO dhfr- | C1035-1 | DC1035-1 | MC1035-1 |
| UT | human | CHO-K1 | C1035-1a | DC1035-1a | MC1035-1a | |
| Vasoactive Intestinal Peptide | PAC1 | human | HEK293T | C1415 | DC1415 | MC1415 |
| VPAC1 | human | CHO-K1 | C1292-1 | DC1292-1 | MC1292-1 | |
| VPAC2 | human | HEK293T | H1293 | DH1293 | MH1293 | |
| Vasopressin/Oxytocin | OT | human | CHO-K1 | C1299-1 | DC1299-1 | MC1299-1 |
| OT | rabbit | HEK293T | Cb1299 | DCb1299 | MCb1299 | |
| OT | rabbit | HEK293T | Cb1299L | DCb1299L | MCb1299L | |
| V1A | human | CHO-K1 | C1042-1 | DC1042-1 | MC1042-1 | |
| V1A | rabbit | HEK293T | Cb1042 | DCb1042 | MCb1042 | |
| V1B | human | CHO-K1 | C1043-1 | DC1043-1 | MC1043-1 | |
| V1B | rabbit | HEK293T | Cb1043 | DCb1043 | MCb1043 | |
| V1B | rabbit | HEK293T | Cb1043L | DCb1043L | MCb1043L | |
| V2 | human | CHO-K1 | C1044-1 | DC1044-1 | MC1044-1 | |
| V2 | rabbit | HEK293T | Cb1044 | DCb1044 | MCb1044 | |
| V2 | rabbit | HEK293T | Cb1044L | DCb1044L | MCb1044L | |
| V2 | dog | CHO-K1 | Cd1044-1 | DCd1044-1 | MCd1044-1 | |
| Zinc | GPR39 | human | HEK293T | H1099 | DH1099 | MH1099 |
| Target Family | Target | Species | Cells |
|---|---|---|---|
| Kinase | AMPK | human | C2C12 |
| DNA-PK | human | Hela | |
| Aryl Hydrocarbon Receptor (Nuclear Hormone Receptor) | AHR | human | Hep G2 |
| AHR | mouse | Hepa1-6 | |
| AHR | human | HG2L6.1c1 CALUX | |
| AHR | mouse | H1L6.c3 CALUX | |
| Chemokine | CCR4 | human | H9 |
| CCR6 | human | H9 | |
| Calcitonin | CGRP | human | SK-N-MC |
| Free Fatty Acid | GPR40 | mouse | MIN6 |
| Lysophospholipid | LPA | human | Human Fibroblast-Like Synoviocytes-Rheumatoid |
| Melanin-Concentrating Hormone | MCH1 | human | YS35 |
| Opioid | mu | human | SK-N-SH |
| Serotonin | 5-HT | human | Human Heart Valvular Interstitial Cells |
| Receptor Family | Target | Species | Parental | Stable Cell Line | Division-Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Integrin | a V b 1 | human | CHOB2 | C3001-1 | DC3001-1 | MC3001-1 |
| Potassium Channel | TMEM175 | human | HEK293T | C1527 | DC1527 | MC1527 |
| TMEM175 | human | HEK293T | C1527a | DC1527a | MC1527a | |
| Receptor Tyrosine Kinases | TrKA | human | CHO-K1 | CK1001-1 | DCK1001-1 | MCK1001-1 |
| TrKA | human | CHO-K1 | CK1001-1b | DCK1001-1b | MCK1001-1b | |
| TrKA | rat | CHO-K1 | CKr1001-1 | DCKr1001-1 | MCKr1001-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1 | DCK1002-1 | MCK1002-1 | |
| FGFR3 | human | CHO-K1 | CK1002-1a | DCK1002-1a | MCK1002-1a | |
| SARS-CoV-2 | TMPRSS2-ACE2 | human | HEK293T | C2007 | DC2007 | MC2007 |
| Zinc Transporter | ZnT3 | human | Hela | C2001-7 | DC2001-7 | MC2001-7 |
| ZnT8 | human | CHO-K1 | C2002-1 | DC2002-1 | MC2002-1 |
| Parental | Stable Cell Lines | Division-Arrested Cells | Membranes |
|---|---|---|---|
| HEK293T | DC0001 | MC0001 | |
| HEK293T Gαqi5 | CG0001 | DCG0001 | MCG0001 |
| CHO-K1 | DC0001-1 | MC0001-1 | |
| CHO-K1 Gαqi5 | CG0001-1 | DCG0001-1 | MCG0001-1 |
| CHO-K1 Gα16 | CG0002-1 | DCG0002-1 | MCG0002-1 |
| CHO-K1 Gα16 Gαqi5 | CG0003-1 | DCG0003-1 | MCG0003-1 |
| CHO dhfr- | DCD0001-1 | MCD0001-1 | |
| CHO-K1 NFAT | CK0001-1 | DCK0001-1 | MCK0001-1 |
| 1321N1 | DC0001-3 | MC0001-3 | |
| RH7777 | DC0001-6 | MC0001-6 | |
| Hela | DC0001-7 | MC0001-7 |
| Assay Kit | Unit Size (384-well) | Catalog | Description | Data |
|---|---|---|---|---|
| MULTISCREEN™ β-Arrestin Assay Kit | 1 plate 96- well/384-well | MSBAK01-1 | The kits contain the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Validated by MULTISCREEN™ stable cell lines co-expressing target GPCRs and MULTISCREEN™ β-Arrestin sensors. Suitable for any cell line or primary cells co-expressing endogenous or untagged GPCR target and MULTISCREEN™ β-Arrestin sensor. | β-Arrestin Recruitment Dose Response in MULTISCREEN™ MOR β-Arrestin2 CHO-K1 stable cell line (CA1350-1a) measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in assay buffer in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | MSBAK01-10 | |||
| 100 plates 96-well/384-well | MSBAK01-100 | |||
| MULTISCREEN™ β-Arrestin BacMam Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKBM01-1 Or β-Arrestin2 MSBAKBM02-1 | The kits contain BacMam viral particles of MULTISCREEN™ β-Arrestin sensor cDNA, control GFP BacMam viral particle, the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. | β-Arrestin Recruitment Dose Response in MULTISCREEN™ MOR CHO-K1 stable cell line (C1350-1a) infected with β-Arrestin sensor BacMam virus for 48 hours before being measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist DAMGO and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-10 Or β-Arrestin2 MSBAKBM02-10 |
|||
| 100 plates 96-well/384-well | β-Arrestin1 MSBAKBM01-100 Or β-Arrestin2 MSBAKBM02-100 |
|||
| MULTISCREEN™ β-Arrestin HSV Assay Kit | 1 plate 96- well/384-well | β-Arrestin1 MSBAKHSV01-1 Or β-Arrestin2 MSBAKHSV02-1 | The kits contain HSV viral particles of MULTISCREEN™ β-Arrestin sensor cDNA, control GFP HSV viral particle, the substrate for MULTISCREEN™ β-Arrestin sensors and assay buffers. They provide homogeneous luminescence assays for intracellular β-Arrestin translocation detection in 96-well, 384-well and higher multiplexity. Total hands-on time for the assay is less than 30 minutes. Suitable for any cell line or primary cells expressing endogenous or untagged GPCR target. | β-Arrestin Recruitment Dose Response in MULTISCREEN™ KOR HEK293T stable cell line (C1352) infected with β-Arrestin HSV sensor for 48 hours before being measured with MULTISCREEN™ β-Arrestin Assay Kit. Cells were seeded in a 384-well plate, incubated with the MULTISCREEN™ Substrate before being treated with control agonist Dynorphin B and measured by Flexstation 3. |
| 10 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-10 Or β-Arrestin2 MSBAKHSV02-10 |
|||
| 100 plates 96-well/384-well | β-Arrestin1 MSBAKHSV01-100 Or β-Arrestin2 MSBAKHSV02-100 |
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| MULTISCREEN™ Calcium 1.0 No Wash Assay Kit | 1000 tests | MSCA01-1 | MULTISCREEN™ Calcium 1.0 No Wash Assay Kits provide homogeneous fluorescence-based assays for intracellular calcium mobilization detection in 96-well, 384-well and higher multiplexity. Pre-loaded with Calcium 1.0 is taken up by the cells where the lipophilic blocking groups of Calcium 1.0 are cleaved by esterases, resulting in a negatively charged fluorescent dye that stays inside cells. The fluorescence signal is greatly enhanced after binding to intracellular calcium released by cell-stimulation. Long wavelength, high sensitivity, and >100 times fluorescence enhancement make Calcium 1.0 an ideal indicator for intracellular calcium release assays measuring GPCRs, calcium channels and receptor tyrosine kinase signaling. MULTISCREEN™ Calcium 1.0 No Wash Assay Kits are validated by MULTISCREEN™ stable cell lines. | Calcium Dose Response in MULTISCREEN™ A2B-HEK293T stable cell line (C1429) measured with MULTISCREEN™ Calcium 1.0 No Wash Assay Kit. Cells were seeded in assay buffer in a 384-well black wall clear bottom PDL-coated plate, incubated with the MULTISCREEN™ Calcium 1.0 No Wash Assay Kit before being treated with control agonist NECA and measured by FLIPR. |
| 10000 tests | MSCA01-10 | |||
| 100000 tests | MSCA01-100 | |||
| MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kit | 500 tests | MSCM01-1 | MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kits provide a homogenous TR-FRET assay method for adenylyl cyclase activity detection in 96-well, 384-well and higher multiplexity. α-cAMP antibody (Ab) is labeled with MULTISCREEN™Eu while cAMP is labeled with MULTISCREEN™650. In the absence of cAMP, MULTISCREEN™650-cAMP is bound to MULTISCREEN™Eu-α-cAMP-Ab to give a strong TR-FRET Emission at 655 nm. Free cAMP in the test sample competes for binding to the MULTISCREEN™ Eu-α-cAMP-Ab, reducing TR-FRET signal from MULTISCREEN™650-cAMP binding. The MULTISCREEN™650-cAMP only has fluorescence lifetime of nanosecond while MULTISCREEN™Eu-α-cAMP-Ab has much longer fluorescence lifetime value due to TR-FRET. The magnitude of TR-FRET is proportional to the concentration of cAMP in a sample. MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kits are validated by MULTISCREEN™ stable cell lines. | cAMP Dose-Response in MULTISCREEN™ β1-HEK293T stable cell line (C1437-1) measured with MULTISCREEN™ TR-FRET cAMP 1.0 No Wash Assay Kit. Cells were seeded in a 384-well solid white plate, incubated with Isoproterenol and 1mM IBMX before being treated with MULTISCREEN™Eu-α-cAMP-Ab and MULTISCREEN™650-cAMP, and measured by FlexStation 3. |
| 5000 tests | MSCM01-5 | |||
| 25000 tests | MSCM01-25 | |||
| MULTISCREEN™ Cell Viability Assay Kit | 400 tests | MSCV01-1 | The MULTISCREEN™ Cell Viability Assay Kit (DTT free) delivers a fast, simple, and highly sensitive luminescence assay for monitoring cell proliferation, viability, and toxicity in mammalian cells. Using firefly luciferase to detect endogenous ATP, it provides bright, stable signals with sensitivity to detect as low as 50 cells per well. Ready-to-use and compatible with 96- and 384-well plates, the kit ensures reliable, reproducible results and has been validated with MULTISCREEN™ stable cell lines, making it an ideal choice for accurate, efficient cell viability testing. | ATP Dose-Response in MULTISCREEN™ MDA-MB-231 parental cells measured with MULTISCREEN™ Cell Viability Assay Kit. Cells were seeded in a 384-well solid white plate, incubated with compound before addition of MULTISCREEN™ ATP assay reagent, and measured by FlexStation 3. |
| 4000 tests | MSCV01-10 | |||
| 40000 tests | MSCV01-100 |