Synthesis and characterization of [125I]TZ6544, a promising radioligand for investigating sphingosine-1-phosphate receptor 2

Synthesis and characterization of [125I]TZ6544, a promising radioligand for investigating sphingosine-1-phosphate receptor 2 GPCR Target: S1PR4 lysophospholipid receptor membrane Authors: Luo, Z., et al. Journal: Nucl Med Biol. 2020;88-89:52-61. doi:10.1016/j.nucmedbio.2020.07.007…

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The effect of fatty diacid acylation of human PYY3-36 on Y2 receptor potency and half-life in minipigs

The effect of fatty diacid acylation of human PYY3-36 on Y2 receptor potency and half-life in minipigs GPCR Target: CHO cells stably expressing the human Y2R Cat # CG1274 Authors:…

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