Peer-Reviewed Papers

Sphingosine-1-Phosphate Receptor Subtype 1 (S1P1) Modulator IMMH001 Regulates Adjuvant- and Collagen-Induced Arthritis

GPCR Target: S1P1

Authors: Jing Jin, et al.

Company: Chinese Academy of Medical Sciences and Peking Union Medical College

Journal: Front. Pharmacol. 10:1085.

Year Published: 2019

Nucleoside 5′-O-monophosphorothioates as modulators of the P2Y14 receptor and mast cell degranulation

GPCR Target: P2Y14

Authors: Edyta Gendaszewska-Darmach, et al.

Company: Lodz University of Technology / Polish Academy of Sciences

Journal: Oncotarget. October 25, 2016; 7(43): 69358–69370.

Year Published: 2016

Pharmacology of AMG 416 (Velcalcetide), a Novel Peptide Agonist of the Calcium-Sensing Receptor, for the Treatment of Secondary Hyperparathyroidism in Hemodialysis Patients

GPCR Target: hCaSR

Authors: Sarah Walter, et al.

Company: Amgen, Inc.

Journal: Journal of Pharmacology and Experimental Therapeutics August 2013, 346 (2) 229-240

Year Published: 2013

Amelioration of PXR-mediated CYP3A4 induction by mGluR2 modulators

GPCR Target: mGLUR2

Authors: Roy J.Vaza, et al.

Company: Sanofi US

Journal: Bioorganic & Medicinal Chemistry Letters Volume 28, Issue 19, October 15, 2018, 3194-3196

Year Published: 2018

Discovery of Novel and Potent Leukotriene B4 Receptor Antagonists. Part 1

GPCR Target: BLT1/BLT2

Authors: Robert A. Goodnow Jr., et al.

Company: Roche Research Center

Journal: Journal of Medical Chemistry 2010, 53, 9, 3502-3516

Year Published: 2010

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