Identification and In Vivo Evaluation of Myelination Agent PIPE-3297, a Selective Kappa Opioid Receptor Agonist Devoid of β-Arrestin-2 Recruitment Efficacy

Identification and In Vivo Evaluation of Myelination Agent PIPE-3297, a Selective Kappa Opioid Receptor Agonist Devoid of β-Arrestin-2 Recruitment Efficacy

GPCR Target: Membranes isolated from CHO-K1 cells stably expressing human KORs (cat. no. MC1351-1a), MULTISCREENᵀᴹ β-arrestin-2 recruitment assay

Authors: Schrader, T. O., et al.

Journal: ACS Chemical Neuroscience, 15(3), 685–698. 

Year Published: 2024

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